Stereoselective synthesis of (R)- and (S)-2-methyl-3-oxo-3,4-dihydro- 2H-1,4-benzoxazine-2-carboxylic acids, -carboxylates and -carboxamides

Tetrahedron Asymmetry

Volumn 10, Issue 1, 1999, Pages 153-167

  Breznik, Matej ^a   Hrast, Valentina ^a   Mrcina, Alenka ^a   Kikelj, Danijel ^a  

^a UNIVERSITY OF LJUBLJANA   (Slovenia)

Author keywords

[No Author keywords available]

Indexed keywords

AMIDE; BENZOXAZINE DERIVATIVE; CARBOXYLIC ACID DERIVATIVE;

ARTICLE; DRUG STRUCTURE; DRUG SYNTHESIS; ENANTIOMER; PRIORITY JOURNAL; STEREOCHEMISTRY; STRUCTURE ANALYSIS;

EID: 0033556594     PISSN: 09574166     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0957-4166(98)00485-6     Document Type: Article

References (11)

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2. Kikelj, D.; Povšič, L.; Pristovšek, P.; Štalc, A.; Kidrič, J. Med. Chem. Res. 1996, 6, 118-127.
3. Goodman, M.; Ro, S. Peptidomimetics for drug design. In Burger's Medicinal Chemistry and Drug Discovery; Wolff, M. E., Ed.; John Wiley & Sons Inc.: New York, 1995; pp. 803-861.
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6. Breznik, M.; Mrcina, A.; Kikelj, D. Tetrahedron: Asymmetry 1998, 9, 1115-1116.
7. Breznik, M.; Kikelj, D. Tetrahedron: Asymmetry 1997, 8, 425-434.
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9. March, J. Advanced Organic Chemistry - 4th Edition; Wiley Interscience: New York, 1992; p. 1218.
10. Schwarz, H.; Arakawa, K. J. Am. Chem. Soc. 1959, 81, 5691-5696.
11. Parker, D.; Taylor, R. J. Analytical methods: determination of enantiomeric purity. In Asymmetric Synthesis; Aitken, R. A.; Kilényi, S. N., Eds; Blackie Academic & Professional: London, 1994; p. 36.