Enantioselective synthesis of a key intermediate of Levofloxacin using microbial resolution

Tetrahedron Asymmetry

Volumn 10, Issue 1, 1999, Pages 119-123

  Miyadera, Akihiko ^a   Imura, Akihiro ^a  

^a DAIICHI SANKYO CO   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

7,8 DIFLUORO 2,3 DIHYDRO 3 METHYL 4H 1,4 BENZOXAZINE; AMIDE; BENZOXAZINE DERIVATIVE; LEVOFLOXACIN; UNCLASSIFIED DRUG;

ARTICLE; BACILLUS; DEBARYOMYCES; DRUG SYNTHESIS; ENANTIOMER; LYOPHILISATE; MICROORGANISM; NONHUMAN; PRIORITY JOURNAL; STEREOCHEMISTRY;

EID: 0033556502     PISSN: 09574166     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0957-4166(98)00475-3     Document Type: Article

References (8)

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2. (b) Daiichi Seiyaku, Drugs Future 1992, 17, 559-563.
3. Atarashi, S.; Yokohama, S.; Yamazaki, K.; Sakano, K.; Imamura, M.; Hayakawa, I. Chem. Pharm. Bull. Jpn. 1987, 35, 1896-1902.
4. Atarashi, S.; Tsurumi, H.; Fujiwara, T.; Hayakawa, I. J. Heterocycl. Chem. 1991, 28, 329-331.
5. Kang, S. B.; Ahn, E. J.; Kim, Y.; Kim, Y. H. Tetrahedron Lett. 1996, 37, 9317-9320.
6. Sakano, K.; Yokohama, S.; Hayakawa, I.; Atarashi, S.; Kadoya, S. Agric. Biol. Chem. 1987, 51, 1265-1270.
7. Mori, K.; Iwasawa, H. Tetrahedron 1980, 36, 2209-2213.
8. Chen, C.-S.; Fujimoto, Y.; Girdaukas, G.; Sih, C. J. J. Am. Chem. Soc. 1982, 104, 7292-7299.