Amino acids and peptides. LVI. Synthesis of pyrazinone ring-containing opioid mimetics and examination of their opioid receptor binding activity

Tetrahedron

Volumn 55, Issue 50, 1999, Pages 14391-14406

  Okada, Yoshio ^a   Fukumizu, Atsuko ^a   Takahashi, Motohiro ^a   Yamazaki, Junpei ^a   Yokoi, Toshio ^a   Tsuda, Yuko ^a   Bryant, Sharon D ^b   Lazarus, Lawrence H ^b  

^a KOBE GAKUIN UNIVERSITY   (Japan)

^b NATIONAL INSTITUTE OF ENVIRONMENTAL HEALTH SCIENCES   (United States)

Author keywords

Cyclization; Dipeptidyl chloromethyl ketone; Opioid mimetics; Pyrazinone ring containing amino acids

Indexed keywords

DELTA OPIATE RECEPTOR; MU OPIATE RECEPTOR; OPIATE AGONIST; PYRAZINE DERIVATIVE;

ANIMAL TISSUE; ARTICLE; BRAIN SYNAPTOSOME; CYCLIZATION; DRUG SYNTHESIS; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR BINDING; STRUCTURE ACTIVITY RELATION;

EID: 0033544785     PISSN: 00404020     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4020(99)00908-4     Document Type: Article

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