An efficient synthesis of optically active metabolites of platelet adhesion inhibitor OPC-29030 by lipase-catalyzed enantioselective transesterification

Tetrahedron Letters

Volumn 40, Issue 28, 1999, Pages 5235-5238

  Kitano, Kazuyoshi ^a   Matsubara, Jun ^a   Ohtani, Tadaaki ^a   Otsubo, Kenji ^a   Kawano, Yoshikazu ^a   Morita, Seiji ^a   Uchida, Minoru ^a  

^a OTSUKA PHARMACEUTICAL CO LTD   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

3,4 DIHYDRO 6 [3 [1 (2 METHYLPHENYL) 2 IMIDAZOLYLSULFINYL]PROPOXY] 2(1H) QUINOLINONE; 3,4 DIHYDRO 6 [3 [1 (2 TOLYL) 2 IMIDAZOLYL]SULFINYLPROPOXY] 2(1H) QUINOLINONE; ANTITHROMBOCYTIC AGENT; UNCLASSIFIED DRUG;

ARTICLE; DRUG CONFORMATION; DRUG EFFECT; DRUG SYNTHESIS; ENANTIOMER; ESTERIFICATION; STRUCTURE ACTIVITY RELATION; THROMBOCYTE AGGREGATION INHIBITION;

EID: 0033538604     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(99)00946-6     Document Type: Article

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