4-hydroxy-1-[3-(5-(1,2,4-triazol-4-yl)-1H-indol-3-yl)propyl]piperidines: Selective h5-HT(1D) agonists for the treatment of migraine

Bioorganic and Medicinal Chemistry Letters

Volumn 9, Issue 23, 1999, Pages 3369-3374

  Bourrain, Sylvie ^a   Neduvelil, Joseph G ^a   Beer, Margaret S ^a   Stanton, Josephine A ^a   Showell, Graham A ^a   Macleod, Angus M ^a  

^a NEUROSCIENCE RESEARCH CENTRE   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

4 HYDROXY 1 [3 (5 (1,2,4 TRIAZOL 4 YL) 1H INDOL 3 YL)PROPYL]PIPERIDINE; ANTIMIGRAINE AGENT; NARATRIPTAN; RIZATRIPTAN; SEROTONIN 1D AGONIST; SEROTONIN 1D RECEPTOR; SUMATRIPTAN; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; DRUG MECHANISM; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; DRUG STRUCTURE; MIGRAINE;

EID: 0033530881     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(99)00614-9     Document Type: Article

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