First fatty acylated dipeptides to affect muscarinic receptor ligand binding

Bioorganic and Medicinal Chemistry Letters

Volumn 9, Issue 23, 1999, Pages 3363-3368

  Krishnan, Vyjayanthi ^a   Pham, Wellington N ^a   Messer Jr , William S ^a   Peseckis, Steven M ^a  

^a MEDICAL COLLEGE OF OHIO   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

DIPEPTIDE; GUANINE NUCLEOTIDE BINDING PROTEIN; MUSCARINIC AGENT; MUSCARINIC M1 RECEPTOR; MUSCARINIC M2 RECEPTOR;

ARTICLE; BINDING AFFINITY; BINDING SITE; DRUG MECHANISM; DRUG SYNTHESIS; LIGAND BINDING;

EID: 0033530813     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(99)00604-6     Document Type: Article

References (8)

1. Wess, J. FASEB J. 1997, 11, 346-354.
2. Neer, E.J. Cell 1995, 80, 249-257.
3. Resh, M.D. Cell Signall. 1996, 8, 403-412.
4. Wang, S.-S.; Gisin, B.F.; Winter, D.P.; Makofske, R.; Kulesha, I.D.; Tzougraki, C.; Meienhofer, J. J. Org. Chem. 1977, 42, 1286-1290.
5. Philips, R.S. Archiv. Biochem. Biophys. 1987, 256, 1, 302-310.
6. 5: C, 67.50; H, 9.15; N, 6.06. Found: C, 67.70; H, 9.23; N, 5.90.
7. Huang, X.-P.; Williams, F. E.; Peseckis, S.M.; Messer, W. S. Jr. J. Pharmacol. Exp. Thr. 1998, 286, 3, 1129-1139.
8. Huang, X.-P.; Nagy, P.I.; Williams, F.E.; Peseckis, S.M.; Messer, W.S. Jr. Br. J. Pharmacol. 1999, 126, 735-745.