Syntheses and evaluation of amidinobenzofuran derivatives as tryptase inhibitors

Bioorganic and Medicinal Chemistry Letters

Volumn 9, Issue 23, 1999, Pages 3285-3290

  Ono, Shin'ichiro ^a   Kuwahara, Shigeki ^a   Takeuchi, Masahiro ^a   Sakashita, Hiroshi ^a   Naito, Youichiro ^a   Kondo, Takao ^a  

^a Yoshitomi Pharmaceutical Industries Ltd   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

1,5 BIS[4 (5 AMIDINOBENZOFURAN 2 YLCARBONYL)PIPERAZINYLCARBONYLMETHOXY]CYCLOOCTANE; BENZOFURAN DERIVATIVE; ENZYME INHIBITOR; N (1 HYDROXY 2 NAPHTHOYL)ARGINYLPROLINAMIDE; TRYPTASE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ARTICLE; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; ENZYME SPECIFICITY; NONHUMAN; RAT; STRUCTURE ACTIVITY RELATION;

EID: 0033530812     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(99)00594-6     Document Type: Article

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