-
3
-
-
0024456087
-
-
(c) Spealman, R. D.; Madras, B. K.; Bergman, J. J. Pharmacol. Exp. Ther. 1989, 251, 142-149.
-
(1989)
J. Pharmacol. Exp. Ther.
, vol.251
, pp. 142-149
-
-
Spealman, R.D.1
Madras, B.K.2
Bergman, J.3
-
4
-
-
0025855256
-
-
2. (a) Kuhar, M. J.; Ritz, M. C.; Boja, J. W. Trends Neurosci. 1991, 14, 299-302;
-
(1991)
Trends Neurosci.
, vol.14
, pp. 299-302
-
-
Kuhar, M.J.1
Ritz, M.C.2
Boja, J.W.3
-
6
-
-
0026566383
-
-
3. Carrol, F. I.; Lewin, A. H.; Boja, J. W.; Kuhar, M. J. J. Med. Chem. 1992, 35, 969-981.
-
(1992)
J. Med. Chem.
, vol.35
, pp. 969-981
-
-
Carrol, F.I.1
Lewin, A.H.2
Boja, J.W.3
Kuhar, M.J.4
-
7
-
-
0027468956
-
-
4. (a) Meltzer, P. C.; Liang, A. Y.; Brownell, A.-L.; Elmaleh, D. R.; Madras, B. K. J. Med. Chem. 1993, 36, 855-862;
-
(1993)
J. Med. Chem.
, vol.36
, pp. 855-862
-
-
Meltzer, P.C.1
Liang, A.Y.2
Brownell, A.-L.3
Elmaleh, D.R.4
Madras, B.K.5
-
8
-
-
0030051988
-
-
(b) Meltzer, P. C.; Liang, A. Y.; Madras, B. K. J. Med. Chem. 1996, 39, 371-379;
-
(1996)
J. Med. Chem.
, vol.39
, pp. 371-379
-
-
Meltzer, P.C.1
Liang, A.Y.2
Madras, B.K.3
-
9
-
-
0027446171
-
-
(c) Davies, H. M.; Saikali, E.; Sexton, T.; Childers, S. R. Eur. J. Pharmacol. Mol. Pharmacol. Sect. 1993, 244, 93-97.
-
(1993)
Eur. J. Pharmacol. Mol. Pharmacol. Sect.
, vol.244
, pp. 93-97
-
-
Davies, H.M.1
Saikali, E.2
Sexton, T.3
Childers, S.R.4
-
10
-
-
0026009418
-
-
5. (a) Carrol, F. I.; Gao, Y.; Rahman, M. A.; Abraham, P.; Lewin, A. H.; Parham, K. A.; Boja, J. W.; Kuhar, M. J. J. Med. Chem. 1991, 35, 2719-2725;
-
(1991)
J. Med. Chem.
, vol.35
, pp. 2719-2725
-
-
Carrol, F.I.1
Gao, Y.2
Rahman, M.A.3
Abraham, P.4
Lewin, A.H.5
Parham, K.A.6
Boja, J.W.7
Kuhar, M.J.8
-
11
-
-
0001630928
-
-
Kozikowski, A. P., Ed., Raven Press, New York
-
(b) Carrol, F. I.; Lewin, A. H.; Boja, J. W.; Kuhar, M. J. In Drug Design for Neuroscience, Kozikowski, A. P., Ed., Raven Press, New York, 1993, pp. 149-166.
-
(1993)
Drug Design for Neuroscience
, pp. 149-166
-
-
Carrol, F.I.1
Lewin, A.H.2
Boja, J.W.3
Kuhar, M.J.4
-
12
-
-
0032504009
-
-
(c) Simoni, D.; Roberti, M.; Andrisano, V.; Manferdini, M.; Rondanin, R.; Kozikowski, A. P. J. Org. Chem. 1998, 63, 4834.
-
(1998)
J. Org. Chem.
, vol.63
, pp. 4834
-
-
Simoni, D.1
Roberti, M.2
Andrisano, V.3
Manferdini, M.4
Rondanin, R.5
Kozikowski, A.P.6
-
13
-
-
0027139321
-
-
(d) Simoni, D.; Stoelwinder, J.; Kozikowski, A. P.; Johnson, K. M.; Bergman, J. S.; Ball, R. G. J. Med. Chem. 1993, 36, 3975-3978.
-
(1993)
J. Med. Chem.
, vol.36
, pp. 3975-3978
-
-
Simoni, D.1
Stoelwinder, J.2
Kozikowski, A.P.3
Johnson, K.M.4
Bergman, J.S.5
Ball, R.G.6
-
14
-
-
0028077861
-
-
6. Yang, B.; Wright, J.; Eldefrawi, M. E.; Pou, S.; MacKerell, A. D. J. Am. Chem. Soc. 1994, 116, 8722-8732.
-
(1994)
J. Am. Chem. Soc.
, vol.116
, pp. 8722-8732
-
-
Yang, B.1
Wright, J.2
Eldefrawi, M.E.3
Pou, S.4
MacKerell, A.D.5
-
15
-
-
0028062672
-
-
7. Kozikowski, A. P.; Saiah, M. K. E.; Bergman, J. S.; Johnson, K. M. J. Med. Chem. 1994, 37, 3440-3442.
-
(1994)
J. Med. Chem.
, vol.37
, pp. 3440-3442
-
-
Kozikowski, A.P.1
Saiah, M.K.E.2
Bergman, J.S.3
Johnson, K.M.4
-
16
-
-
0029965036
-
-
8. (a) Madras, B. K.; Pristupa, Z. B.; Niznik, H. B.; Liang A. Y.; Blundell, P.; Gonzales, M. D.; Meltzer, P. C. Synapse 1996, 24, 340-348;
-
(1996)
Synapse
, vol.24
, pp. 340-348
-
-
Madras, B.K.1
Pristupa, Z.B.2
Niznik, H.B.3
Liang, A.Y.4
Blundell, P.5
Gonzales, M.D.6
Meltzer, P.C.7
-
17
-
-
0030837830
-
-
(b) Meltzer, P. C.; Liang A. Y.; Blundell, P.; Gonzales, M. D.; Chen, Z.; George, C.; Madras, B. K. J. Med. Chem. 1997, 40, 2661-2673.
-
(1997)
J. Med. Chem.
, vol.40
, pp. 2661-2673
-
-
Meltzer, P.C.1
Liang, A.Y.2
Blundell, P.3
Gonzales, M.D.4
Chen, Z.5
George, C.6
Madras, B.K.7
-
20
-
-
37049091394
-
-
11. Ansell, M. F.; Mason, J. S.; Caton, M. P. J. Chem. Soc., Perkin Trans. I 1984, 1061-1068.
-
(1984)
J. Chem. Soc., Perkin Trans. I
, pp. 1061-1068
-
-
Ansell, M.F.1
Mason, J.S.2
Caton, M.P.3
-
21
-
-
0019945851
-
-
12. Carrol, F. I.; Coleman, M. L.; Lewin, A. H. J. Org. Chem. 1982, 47, 13-19.
-
(1982)
J. Org. Chem.
, vol.47
, pp. 13-19
-
-
Carrol, F.I.1
Coleman, M.L.2
Lewin, A.H.3
-
22
-
-
0001762573
-
-
13. Shirai, R.; Tanaka, M.; Koga, K. J. Am. Chem. Soc. 1986, 108, 543-545.
-
(1986)
J. Am. Chem. Soc.
, vol.108
, pp. 543-545
-
-
Shirai, R.1
Tanaka, M.2
Koga, K.3
-
23
-
-
0027472613
-
-
14. Bunn, B. J.; Cox, P. J.; Simpkins, N. S. Tetrahedron 1993, 49, 207-218.
-
(1993)
Tetrahedron
, vol.49
, pp. 207-218
-
-
Bunn, B.J.1
Cox, P.J.2
Simpkins, N.S.3
-
25
-
-
0013614053
-
-
3), 86 % ee
-
3), 86 % ee.
-
-
-
-
26
-
-
0021287012
-
-
17. (a) Javitch, J. A.; Blaustein, R. O.; Snyder, S. H. Mol. Pharmacol. 1984, 26, 35-44;
-
(1984)
Mol. Pharmacol.
, vol.26
, pp. 35-44
-
-
Javitch, J.A.1
Blaustein, R.O.2
Snyder, S.H.3
-
28
-
-
0027054352
-
-
18. Searle, M. S.; William, D. H.; Gerhard, U. J. Am. Chem. Soc. 1992, 114, 10697-10704.
-
(1992)
J. Am. Chem. Soc.
, vol.114
, pp. 10697-10704
-
-
Searle, M.S.1
William, D.H.2
Gerhard, U.3
-
31
-
-
0013623549
-
-
Binding affinities (μM) of (+)-cocaine, WIN 35,428 and its oxa-analogue: 15.8, 0.0075, 0.546
-
21. Binding affinities (μM) of (+)-cocaine, WIN 35,428 and its oxa-analogue: 15.8, 0.0075, 0.546.
-
-
-
|