Simplified pepstatins: Synthesis and evaluation of N-terminally modified analogues

Journal of Medicinal Chemistry

Volumn 42, Issue 11, 1999, Pages 2041-2045

  Kratzel, Martin ^a   Schlichtner, Birgit ^a   Kirchmayer, Roland ^b   Bernkop Schnürch, Andreas ^b  

^a UNIVERSITY OF VIENNA   (Austria)

^b Inst of Pharmaceutical Technology   (Austria)

Author keywords

[No Author keywords available]

Indexed keywords

EPIDERMAL GROWTH FACTOR; PEPSIN A; PEPSTATIN; POLYMER;

ARTICLE; COST; COVALENT BOND; DRUG ACTIVITY; DRUG DELIVERY SYSTEM; DRUG EFFECT; DRUG SYNTHESIS; ENZYME INHIBITION; HUMAN; ORAL DRUG ADMINISTRATION; PROTEIN MODIFICATION; STOMACH ULCER;

ANTI-ULCER AGENTS; DRUG DELIVERY SYSTEMS; EPIDERMAL GROWTH FACTOR; PEPSTATINS; PROTEASE INHIBITORS;

EID: 0033519695     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm9807306     Document Type: Article

References (7)

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5. Kratzel, M.; Hiessböck, R.; Bernkop-Schnürch, A. Auxiliary Agents for the Peroral Administration of Peptide and Protein Drugs: Synthesis and Evaluation of Novel Pepstatin Analogues. J. Med. Chem. 1998, 41, 2339-2344.
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