Neutral acylation (protection) of the indole nitrogen: A simple synthesis of indole-1-carboxylates, indole-1-thiocarboxylates and indole-1- carboxamides

Tetrahedron Letters

Volumn 40, Issue 14, 1999, Pages 2733-2736

  Macor, John E ^a   Cuff, Alison ^a   Cornelius, Lyndon ^a  

^a Pharmaceutical Research Institute   (United States)

Author keywords

Acylation; Carbonyl compounds; Indoles; Protecting groups

Indexed keywords

INDOLE 1 CARBOXYAMIDE; INDOLE 1 CARBOXYLATE; INDOLE 1 THIOCARBOXYLATE; INDOLE DERIVATIVE; NITROGEN; UNCLASSIFIED DRUG;

ACYLATION; ARTICLE; CHEMICAL MODIFICATION; CHEMICAL REACTION; MOLECULAR STABILITY; SYNTHESIS;

EID: 0033515870     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(99)00352-4     Document Type: Article

References (5)

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