Characterization of FR 172357, a new non-peptide bradykinin B2 receptor antagonist, in human, pig and rabbit preparations

European Journal of Pharmacology

Volumn 386, Issue 1, 1999, Pages 25-31

  Rizzi, Caterina ^a   Rizzi, Anna ^a   Calò, Girolamo ^a   Jorizzo, Gianfranco ^a   Agnello, Giovanni ^a   Mollica, Gioacchino ^a   Inamura, Noriaki ^b   Regoli, Domenico ^a  

^a UNIVERSITY OF FERRARA   (Italy)

^b ASTELLAS PHARMA INC   (Japan)

Author keywords

(Human); (Pig); (Rabbit); Antagonist; Bradykinin B2 receptor; Vessel, isolated

Indexed keywords

ANGIOTENSIN; BRADYKININ B2 RECEPTOR ANTAGONIST; ENDOTHELIN 1; FR 172357; NORADRENALIN; SEROTONIN; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; COMPETITIVE INHIBITION; CONCENTRATION RESPONSE; CONTROLLED STUDY; CORONARY ARTERY; DRUG MECHANISM; DRUG STRUCTURE; FEMALE; HUMAN; HUMAN TISSUE; JUGULAR VEIN; NONHUMAN; PRIORITY JOURNAL; RABBIT; SWINE; UMBILICAL VEIN;

ANIMALS; AORTA, THORACIC; BRADYKININ; CORONARY VESSELS; FEMALE; HUMANS; JUGULAR VEINS; MUSCLE, SMOOTH, VASCULAR; PREGNANCY; PYRIDINES; RABBITS; RECEPTOR, BRADYKININ B2; RECEPTORS, BRADYKININ; SWINE; UMBILICAL VEINS;

EID: 0033462194     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(99)00711-6     Document Type: Article

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