Synthesis of ABT-378, an HIV protease inhibitor candidate: Avoiding the use of carbodiimides in a difficult peptide coupling

Organic Process Research and Development

Volumn 3, Issue 2, 1999, Pages 145-148

  Stoner, Eric J ^a   Stengel, Peter J ^a   Cooper, Arthur J ^a  

^a ABBOTT LABORATORIES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0033417984     PISSN: 10836160     EISSN: None     Source Type: Journal    
DOI: 10.1021/op980214p     Document Type: Article

References (5)

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3. (a) Molla, A.; Korneyeva, M.; Gao, Q.; Vasavanonda, S.; Schipper, P. J.; Mo, H.-M.; Markowitz, M.; Chernyavskiy, T.; Niu, P.; Lyonns, N.; Hsu, A.; Granneman, G. R.; Ho, D. D.; Boucher, C. A. B.; Leonard, J. M.; Norbeck, D. W.; Kempf, D. J. Nat. Med. (N. Y.) 1996, 2 (7), 760.
4. (b) Schmit, J.-C.; Ruiz, L.; Clotet, B.; Raventos, A.; Tor, J.; Leonard, J.; Desmyter, J.; De Clercq, E.; Vandamme, A.-M. AIDS 1996, 10, 995.
5. Sham, H. L.; Chen, X. Exp. Opin. Invest. Drugs 1996, 5 (8), 977.