Functional and electrophysiological effects of a novel imidazoline-based K(ATP) channel blocker, IMID-4F

British Journal of Pharmacology

Volumn 128, Issue 8, 1999, Pages 1636-1642

  McPherson, Grant A ^a   Bell, Karen L ^a   Favaloro, Joanne L ^a   Kubo, Masahiro ^b   Standen, Nicholas B ^b  

^a MONASH UNIVERSITY   (Australia)

^b UNIVERSITY OF LEICESTER   (United Kingdom)

Author keywords

Imidazolines; K(ATP) channel antagonists; K(ATP) channels; Levcromakalim; Pig coronary artery; Rat mesenteric artery; Smooth muscle relaxation

Indexed keywords

15 HYDROXY 11ALPHA,9ALPHA EPOXYMETHANOPROSTA 5,13 DIENOIC ACID; 2 CYANO 1 (1,1 DIMETHYLPROPYL) 3 (3 PYRIDYL)GUANIDINE; 2 [N (2,6 DICHLOROPHENYL) N (4 FLUOROBENZYL)AMINO]IMIDAZOLINE; ADENOSINE TRIPHOSPHATE; CLONIDINE DERIVATIVE; GLIBENCLAMIDE; IMIDAZOLINE DERIVATIVE; LEMAKALIM; NITROPRUSSIDE SODIUM; POTASSIUM CHANNEL BLOCKING AGENT; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTERY MUSCLE; ARTICLE; CELL MEMBRANE DEPOLARIZATION; CONCENTRATION RESPONSE; CONTROLLED STUDY; CORONARY ARTERY; CORONARY ARTERY DILATATION; DRUG BINDING SITE; DRUG POTENCY; DRUG STRUCTURE; ELECTROPHYSIOLOGY; MALE; MESENTERIC ARTERY; NONHUMAN; PATCH CLAMP; POTASSIUM CURRENT; PRIORITY JOURNAL; RADIORECEPTOR ASSAY; RAT; SWINE; VASODILATATION;

EID: 0033406151     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0702925     Document Type: Article

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