3-Amidinophenylalanine-based inhibitors of urokinase

Bioorganic and Medicinal Chemistry Letters

Volumn 9, Issue 21, 1999, Pages 3147-3152

  Stürzebecher, Jörg ^a   Vieweg, Helmut ^b   Steinmetzer, Torsten ^a   Schweinitz, Andrea ^a   Stubbs, Milton T ^c   Renatus, Martin ^d   Wikström, Peter ^b  

^a FRIEDRICH SCHILLER UNIVERSITY JENA   (Germany)

^b Pentapharm Ltd   (Switzerland)

^c PHILIPPS UNIVERSITY MARBURG   (Germany)

^d BURNHAM INSTITUTE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

3 AMIDINOPHENYLALANINE DERIVATIVE; AMIDE; ENZYME INHIBITOR; PLASMIN; TRYPSIN; UNCLASSIFIED DRUG; UROKINASE;

ARTICLE; CHEMICAL MODIFICATION; CRYSTAL STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; ENZYME INHIBITOR INTERACTION; STRUCTURE ACTIVITY RELATION;

BENZAMIDINES; ENZYME INHIBITORS; MODELS, MOLECULAR; MOLECULAR CONFORMATION; MOLECULAR STRUCTURE; PHENYLALANINE; PLASMIN; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONAMIDES; TRYPSIN INHIBITORS; URINARY PLASMINOGEN ACTIVATOR;

EID: 0033231047     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(99)00541-7     Document Type: Article

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