Studies in search of α2 selective ligands for GABA(A)/BzR receptor subtypes. Part I. Evidence for the conservation of pharmacophoric descriptors for DS subtypes

Medicinal Chemistry Research

Volumn 9, Issue 3, 1999, Pages 186-202

  Yu, Shu ^a   He, Xiaohui ^a   Ma, Chunrong ^a   McKernan, Ruth ^b   Cook, James M ^a  

^a UNIVERSITY OF WISCONSIN MILWAUKEE   (United States)

^b Merck Sharp & Dohme Limited   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

2 (4 BROMOPHENYL) 8 TERT BUTYL PYRAZOLOQUINOLIN 3 ONE; 4 AMINOBUTYRIC ACID RECEPTOR; PYRAZOLOQUINOLIN 3 ONE DERIVATIVE; QUINOLINE DERIVATIVE; RECOMBINANT RECEPTOR; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; DRUG SELECTIVITY; HIPPOCAMPUS; LIGAND BINDING; LIPOPHILICITY; PHARMACOPHORE; SHORT TERM MEMORY; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

EID: 0033036172     PISSN: 10542523     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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