Characterization of a new AMPA receptor radioligand, [3H]2-amino-3-(3-carboxy-5-methyl-4-isoxazolyl)propionic acid

European Journal of Pharmacology

Volumn 373, Issue 2-3, 1999, Pages 251-262

  Stensbøl, Tine B ^a   Sløk, Frank A ^a   Trometer, Joseph ^b   Hurt, Stephen ^b   Ebert, Bjarke ^c   Kjøller, Connie ^d   Egebjerg, Jan ^e   Madsen, Ulf ^a   Diemer, Nils H ^d   Krogsgaard Larsen, Povl ^a  

^a UNIVERSITY OF COPENHAGEN   (Denmark)

^b Medical Products   (United States)

^c PharmaBiotec Neurosci Res Center   (Denmark)

^d UNIVERSITY OF COPENHAGEN   (Denmark)

^e AARHUS UNIVERSITY   (Denmark)

Author keywords

ACPA ((RS) 2 amino 3 (3 carboxy 5 methyl 4 isoxazolyl)propionic acid); AMPA receptor; Receptor autoradiography; Thiocyanate

Indexed keywords

2 AMINO 3 (3 CARBOXY 5 METHYL 4 ISOXAZOLYL)PROPIONIC ACID; AMPA RECEPTOR; AMPA RECEPTOR AGONIST; RADIOLIGAND; RADIOPHARMACEUTICAL AGENT; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BINDING KINETICS; BRAIN MEMBRANE; DISSOCIATION CONSTANT; DRUG DISTRIBUTION; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; MALE; NONHUMAN; PRIORITY JOURNAL; RAT;

ANIMALS; AUTORADIOGRAPHY; BINDING, COMPETITIVE; BRAIN; CALCIUM CHLORIDE; CELL LINE; EXCITATORY AMINO ACID AGONISTS; ISOXAZOLES; KINETICS; LIGANDS; MALE; MEMBRANES; RADIOLIGAND ASSAY; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, AMPA; RECEPTORS, GLUTAMATE; RECOMBINANT PROTEINS; THIOCYANATES;

EID: 0033021196     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(99)00269-1     Document Type: Article

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