Synthesis of (E)-N-(3-bromoprop-2-enyl)-2β-carbomethoxy-3β-(4'-tolyl) nortropane (PE2Br) and radiolabelling of [76Br]PE2Br: A potential ligand for exploration of the dopamine transporter by PET

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 42, Issue 6, 1999, Pages 581-588

  Helfenbein, J ^a   Emond, P ^a   Loc'h, C ^b   Bottlaender, M ^b   Ottaviani, M ^b   Guilloteau, D ^a   Maziere B ^b   Frangin, Y ^a   Chalon, S ^a  

^a INSERM   (France)

^b SERVICE HOSPITALIER FRÉDÉRIC JOLIOT   (France)

Author keywords

76Br; Cocaine analogue; Dopamine transporter

Indexed keywords

AMINES; BROMINE COMPOUNDS; NEUROPHYSIOLOGY;

76BR; COCAINE ANALOG; DOPAMINE TRANSPORTERS; N-BROMOSUCCINIMIDE; PERACETIC ACIDS; POTENTIAL LIGAND; RADIOCHEMICAL PURITY; RADIOCHEMICAL YIELD; RADIOLABELLING; SYNTHESISED;

BRAIN;

BROMINE; BROMINE DERIVATIVE; DOPAMINE TRANSPORTER; N BROMOSUCCINIMIDE; OXIDIZING AGENT; PERACETIC ACID; TRIBUTYLTIN; TROPANE DERIVATIVE;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; AUTORADIOGRAPHY; BRAIN; BRAIN REGION; CORPUS STRIATUM; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; IN VIVO STUDY; ISOTOPE LABELING; NONHUMAN; POSITRON EMISSION TOMOGRAPHY; PURIFICATION; RADIOACTIVITY; RADIOCHEMISTRY; RAT; SYNTHESIS;

ANIMALIA;

EID: 0032998649     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1099-1344(199906)42:6<581::AID-JLCR218>3.0.CO;2-M     Document Type: Article

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