Synthesis and pharmacological activity of thebaine-derived μ-opioid receptor agonists

Pharmaceutica Acta Helvetiae

Volumn 73, Issue 5, 1999, Pages 251-254

  Shafiee, A ^a   Amanlou, M ^a   Farsam, H ^a   Dehpour, A R ^a   Mir Ershadi, F ^a   Mani, A R ^a  

^a TEHRAN UNIVERSITY OF MEDICAL SCIENCES   (Iran)

Author keywords

Diels Alder's reaction; Opioid agonist activity; Thebaine

Indexed keywords

MORPHINE; MU OPIATE RECEPTOR AGONIST; OPIATE AGONIST; SUCCINIMIDE; THEBAINE;

ANIMAL TISSUE; ANTINOCICEPTION; ARTICLE; CONTROLLED STUDY; DRUG SYNTHESIS; GUINEA PIG; ILEUM; MOUSE; NONHUMAN; SMOOTH MUSCLE; STRUCTURE ACTIVITY RELATION; VAS DEFERENS;

ANALGESICS, OPIOID; ANIMALS; GUINEA PIGS; MALE; MICE; MORPHINE; MUSCLE, SMOOTH; NARCOTICS; PAIN MEASUREMENT; RECEPTORS, OPIOID, MU; THEBAINE; VAS DEFERENS;

EID: 0032997460     PISSN: 00316865     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0031-6865(98)00031-4     Document Type: Article

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