3-amino- and 5-aminopyrazoles with anticonvulsant activity

Archiv der Pharmazie

Volumn 332, Issue 6, 1999, Pages 219-221

  Lankau, Hans Joachim ^a   Menzer, Manfred ^a   Rostock, Angelika ^a   Arnold, Thomas ^a   Rundfeldt, Chris ^a   Unverferth, Klaus ^a  

^a ASTA MEDICA AG   (Germany)

Author keywords

Aminopyrazoles; Anticonvulsant activity; Sodium channel blocker

Indexed keywords

3 AMINO 4 (2 FLUOROPHENYL) 1H PYRAZOLE; 3 AMINO 4 (2 METHYLPHENYL) 5 METHYL 1H PYRAZOLE; 3 AMINO 4 (2 TRIFLUOROMETHYLPHENYL) 1H PYRAZOLE; 3 AMINO 4 (2,4 DICHLOROPHENYL) 1H PYRAZOLE; 3 AMINO 4 (2,4 DICHLOROPHENYL) 5 METHYL 1H PYRAZOLE HYDROCHLORIDE; 3 AMINO 4 (2,6 DICHLOROPHENYL) 1H PYRAZOLE; 3 AMINO 4 (2,6 DIFLUOROPHENYL) 1H PYRAZOLE; 4 BROMOPHENYL 3 (MORPHOLIN 4 YL) 1H PYRAZOLE; 4 CHLOROPHENYL 1 (1 ETHOXYCARBONYLMETHYL) 3 (MORPHOLIN 4 YL) 1H PYRAZOLE; 4 CHLOROPHENYL 1 (2 CHLOROETHYL) 3 (MORPHOLIN 4 YL) 1H PYRAZOLE; 4 CHLOROPHENYL 1 (2 HYDROXYETHYL) 3 (MORPHOLIN 4 YL) 1H PYRAZOLE; 4 CHLOROPHENYL 3 (4 OXO MORPHOLIN 4 YL) 1H PYRAZOLE; 4 CHLOROPHENYL 3 (4 PHENYLPIPERAZIN 1 YL) 1H PYRAZOLE; 4 CHLOROPHENYL 3 (MORPHOLIN 4 YL) 1H PYRAZOLE; ANTICONVULSIVE AGENT; SODIUM CHANNEL BLOCKING AGENT; UNCLASSIFIED DRUG;

ANIMAL CELL; ANTICONVULSANT ACTIVITY; ANTICONVULSANT THERAPY; ARTICLE; DRUG ACTIVITY; DRUG EFFICACY; ELECTRIC SHOCK; NONHUMAN; PRIORITY JOURNAL; RAT;

ANIMALS; ANTICONVULSANTS; CELL LINE; PYRAZOLES; RATS; SODIUM CHANNELS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0032979205     PISSN: 03656233     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1521-4184(19996)332:6<219::AID-ARDP219>3.0.CO;2-T     Document Type: Article

References (6)

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