Effect of G protein-coupled receptor kinase 2 on the sensitivity of M4 muscarinic acetylcholine receptors to agonist-induced internalization and desensitization in NG108-15 cells

Journal of Neurochemistry

Volumn 73, Issue 3, 1999, Pages 1236-1245

  Holroyd, E W ^a   Szekeres, P G ^a   Whittaker, R D ^a   Kelly, E ^b   Edwardson, J M ^a  

^a UNIVERSITY OF CAMBRIDGE   (United Kingdom)

^b UNIVERSITY OF BRISTOL   (United Kingdom)

Author keywords

Desensitization; Internalization; Muscarinic receptors; NG108 cells; Recycling

Indexed keywords

ADENYLATE CYCLASE; CARBACHOL; CHOLINERGIC RECEPTOR STIMULATING AGENT; CYCLIC AMP; GUANINE NUCLEOTIDE BINDING PROTEIN; MUSCARINIC M4 RECEPTOR; PROTEIN TYROSINE KINASE; SUCROSE;

ANIMAL CELL; ARTICLE; CONTROLLED STUDY; ENDOCYTOSIS; GENE OVEREXPRESSION; INTERNALIZATION; KINETICS; MODULATION; NONHUMAN; PRIORITY JOURNAL; RECEPTOR DOWN REGULATION; RECEPTOR SENSITIVITY; RECYCLING;

ADENYLATE CYCLASE; ALGORITHMS; ANIMALS; BETA-ADRENERGIC RECEPTOR KINASE; CARBACHOL; CATTLE; CELL LINE; CYCLIC AMP-DEPENDENT PROTEIN KINASES; ENDOCYTOSIS; ENZYME INHIBITORS; HYPERTONIC SOLUTIONS; MODELS, BIOLOGICAL; MUSCARINIC AGONISTS; RADIOLIGAND ASSAY; RECEPTOR, MUSCARINIC M4; RECEPTORS, MUSCARINIC; SUCROSE;

EID: 0032817553     PISSN: 00223042     EISSN: None     Source Type: Journal    
DOI: 10.1046/j.1471-4159.1999.0731236.x     Document Type: Article

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