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Volumn 290, Issue 3, 1999, Pages 1013-1018

Z-350, a novel compound with α1-adrenoceptor antagonistic and steroid 5α-reductase inhibitory actions: Pharmacological properties in vivo

Author keywords

[No Author keywords available]

Indexed keywords

4 [3 (4 (1 (4 METHYL PHENYL) 3 [4 (2 METHOXYPHENYL)PIPERAZINE 1 YL]PROPOXY)BENZOYL)INDOLE 1 YL]BUTYRIC ACID; ALPHA ADRENERGIC RECEPTOR BLOCKING AGENT; PHENYLEPHRINE; PRAZOSIN; STEROID 5ALPHA REDUCTASE; STEROID 5ALPHA REDUCTASE INHIBITOR; TAMSULOSIN; TESTOSTERONE; UNCLASSIFIED DRUG;

EID: 0032812925     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (13)

References (39)
  • 2
    • 0023630630 scopus 로고
    • Evaluation of the risk for drug-induced postural hypotension in an experimental model: Investigations with carvedilol, prazosin, labetarol, and guanethdine
    • Bartsch W, Sponer G, Strein K, Böhm E and Hooper RG (1967) Evaluation of the risk for drug-induced postural hypotension in an experimental model: Investigations with carvedilol, prazosin, labetarol, and guanethdine. J Cardiovasc Pharmacol 10 (Suppl 11):S49-S51.
    • (1967) J Cardiovasc Pharmacol , vol.10 , Issue.SUPPL. 11
    • Bartsch, W.1    Sponer, G.2    Strein, K.3    Böhm, E.4    Hooper, R.G.5
  • 3
    • 0014414093 scopus 로고
    • Metabolism of testosterone and action of metabolites on prostate glands grown in organ culture
    • Baulieu EE, Lasnitzki I and Robel P (1968) Metabolism of testosterone and action of metabolites on prostate glands grown in organ culture. Nature (Lond) 219:1155-1156.
    • (1968) Nature (Lond) , vol.219 , pp. 1155-1156
    • Baulieu, E.E.1    Lasnitzki, I.2    Robel, P.3
  • 4
    • 0017076325 scopus 로고
    • The use of alpha-adrenergic blockers in benign prostatic obstruction
    • Caine M, Pfau A and Perlberg S (1976) The use of alpha-adrenergic blockers in benign prostatic obstruction. Br J Urol 48:255-263.
    • (1976) Br J Urol , vol.48 , pp. 255-263
    • Caine, M.1    Pfau, A.2    Perlberg, S.3
  • 9
    • 0020422337 scopus 로고
    • Alpha-adrenergic activity and urethral pressure in prostatic zone in benign prostatic hypertrophy
    • Furuya S, Kumamoto Y, Yokoyama E, Tsukamoto T, Izumi T and Abiko Y (1982) Alpha-adrenergic activity and urethral pressure in prostatic zone in benign prostatic hypertrophy. J Urol 128:836-839.
    • (1982) J Urol , vol.128 , pp. 836-839
    • Furuya, S.1    Kumamoto, Y.2    Yokoyama, E.3    Tsukamoto, T.4    Izumi, T.5    Abiko, Y.6
  • 12
    • 0030109784 scopus 로고    scopus 로고
    • The use of α-adrenoceptor antagonists in the pharmacological management of benign prostatic hypertrophy: An overview
    • Hieble JP and Ruffolo RR Jr (1996) The use of α-adrenoceptor antagonists in the pharmacological management of benign prostatic hypertrophy: An overview. Pharmacol Res 33:145-160.
    • (1996) Pharmacol Res , vol.33 , pp. 145-160
    • Hieble, J.P.1    Ruffolo R.R., Jr.2
  • 13
    • 49549145859 scopus 로고
    • Orthostatic hypotension. Mechanisms and management
    • Ibrahim MM, Tarazi RC and Dustan HP (1975) Orthostatic hypotension. Mechanisms and management. Am Heart J 90:513-520.
    • (1975) Am Heart J , vol.90 , pp. 513-520
    • Ibrahim, M.M.1    Tarazi, R.C.2    Dustan, H.P.3
  • 14
    • 0016359646 scopus 로고
    • Steroid 5α-reductase deficiency in man: An inherited form of male pseudohermaphroditism
    • Imperato-McGinley J, Guerrero L, Gautier T and Peterson RE (1974) Steroid 5α-reductase deficiency in man: An inherited form of male pseudohermaphroditism. Science (Wash DC) 186:1213-1215.
    • (1974) Science (Wash Dc) , vol.186 , pp. 1213-1215
    • Imperato-McGinley, J.1    Guerrero, L.2    Gautier, T.3    Peterson, R.E.4
  • 15
    • 0029034556 scopus 로고
    • Efficacy and safety of tamsulosin in the treatment of benign prostatic hyperplasia
    • Kawabe K (1995) Efficacy and safety of tamsulosin in the treatment of benign prostatic hyperplasia. Br J Urol 76(Suppl 1):63-67.
    • (1995) Br J Urol , vol.76 , Issue.SUPPL. 1 , pp. 63-67
    • Kawabe, K.1
  • 16
    • 0025868129 scopus 로고
    • α-Blocker therapy of hypertension: An unfulfilled promise
    • Khoury AF and Kaplan NM (1991) α-Blocker therapy of hypertension: An unfulfilled promise. JAMA 266:394-398.
    • (1991) JAMA , vol.266 , pp. 394-398
    • Khoury, A.F.1    Kaplan, N.M.2
  • 17
    • 0023225035 scopus 로고
    • Pharmacological characteristics of smooth muscle in benign prostatic hyperplasia and normal prostatic tissue
    • Kitada S and Kumazawa J (1987) Pharmacological characteristics of smooth muscle in benign prostatic hyperplasia and normal prostatic tissue. J Urol 138:158-160.
    • (1987) J Urol , vol.138 , pp. 158-160
    • Kitada, S.1    Kumazawa, J.2
  • 19
    • 0030908877 scopus 로고    scopus 로고
    • Pharmacological characterization of the uroselective alpha-1 antagonist Rec 15/2739 (SB 216469): Role of the alpha-1L adrenoceptor in tissue selectivity, part I
    • Leonardi A, Hieble JP, Guarneri L, Naselsky DP, Poggesi E, Sironi G, Sulpizio AC and Testa R (1997) Pharmacological characterization of the uroselective alpha-1 antagonist Rec 15/2739 (SB 216469): Role of the alpha-1L adrenoceptor in tissue selectivity, part I. J Pharmacol Exp Ther 281:1272-1283.
    • (1997) J Pharmacol Exp Ther , vol.281 , pp. 1272-1283
    • Leonardi, A.1    Hieble, J.P.2    Guarneri, L.3    Naselsky, D.P.4    Poggesi, E.5    Sironi, G.6    Sulpizio, A.C.7    Testa, R.8
  • 23
    • 0030759115 scopus 로고    scopus 로고
    • Comparative alpha-1 adrenoceptor subtype selectivity and functional uroselectivity of alpha-1 adrenoceptor antagonists
    • Martin DJ, Lluel P, Guillot E, Coste A, Jammes D and Angel I (1997) Comparative alpha-1 adrenoceptor subtype selectivity and functional uroselectivity of alpha-1 adrenoceptor antagonists. J Pharmacol Exp Ther 282:228-235.
    • (1997) J Pharmacol Exp Ther , vol.282 , pp. 228-235
    • Martin, D.J.1    Lluel, P.2    Guillot, E.3    Coste, A.4    Jammes, D.5    Angel, I.6
  • 24
    • 0032511109 scopus 로고    scopus 로고
    • Relationship between the effects of alfuzosin on rat urethral and blood pressures and its tissue concentrations
    • Martin DJ, Lluel P, Pouyet T, Rauehi-Desanti C and Angel I (1998) Relationship between the effects of alfuzosin on rat urethral and blood pressures and its tissue concentrations. Life Sci 63:169-176.
    • (1998) Life Sci , vol.63 , pp. 169-176
    • Martin, D.J.1    Lluel, P.2    Pouyet, T.3    Rauehi-Desanti, C.4    Angel, I.5
  • 28
    • 0029849606 scopus 로고    scopus 로고
    • Tamsulosin and chlormadinone for the treatment of benign prostatic hyperplasia
    • Okada H, Kawaida N, Ogawa T, Arakawa S, Matsumoto O, Kamidono S and The Kobe University YM617 Study Group (1996) Tamsulosin and chlormadinone for the treatment of benign prostatic hyperplasia. Scand J Urol Nephrol 30:379-385.
    • (1996) Scand J Urol Nephrol , vol.30 , pp. 379-385
    • Okada, H.1    Kawaida, N.2    Ogawa, T.3    Arakawa, S.4    Matsumoto, O.5    Kamidono, S.6
  • 29
    • 0344138588 scopus 로고
    • Reflex venomotor activity in normal persons and in patients with postural hypotension
    • Page EB, Hickam JB, Sieker HO, McIntoch HD and Pryor WW (1955) Reflex venomotor activity in normal persons and in patients with postural hypotension. Circulation 11:262-270.
    • (1955) Circulation , vol.11 , pp. 262-270
    • Page, E.B.1    Hickam, J.B.2    Sieker, H.O.3    McIntoch, H.D.4    Pryor, W.W.5
  • 31
    • 0014847075 scopus 로고
    • Dihydrotestosterone in prostatic hypertrophy. I. The formation and content of dihydrotestosterone in the hypertrophic prostate of man
    • Siiteri PK and Wilson JD (1970) Dihydrotestosterone in prostatic hypertrophy. I. The formation and content of dihydrotestosterone in the hypertrophic prostate of man. J Clin Invest 49:1737-1745.
    • (1970) J Clin Invest , vol.49 , pp. 1737-1745
    • Siiteri, P.K.1    Wilson, J.D.2
  • 32
    • 0026720615 scopus 로고
    • The clinical effects of a 5α-reductase inhibitor, finasteride, on benign prostatic hyperplasia. The Finasteride Study Group
    • Stoner E (1992) The clinical effects of a 5α-reductase inhibitor, finasteride, on benign prostatic hyperplasia. The Finasteride Study Group. J Urol 147:1298-1302.
    • (1992) J Urol , vol.147 , pp. 1298-1302
    • Stoner, E.1
  • 37
    • 0032568008 scopus 로고    scopus 로고
    • Finasteride to prevent morbidity from benign prostatic hyperplasia
    • Wasson JH (1998) Finasteride to prevent morbidity from benign prostatic hyperplasia. N Engl J Med 338:612-613.
    • (1998) N Engl J Med , vol.338 , pp. 612-613
    • Wasson, J.H.1
  • 38
    • 0023176539 scopus 로고
    • Alpha-1 adrenoceptors in human prostate: Characterization and alteration in benign prostatic hypertrophy
    • Yamada S, Ashizawa N, Ushijima H, Nakayama K, Hayashi E and Honda K (1987) Alpha-1 adrenoceptors in human prostate: Characterization and alteration in benign prostatic hypertrophy. J Pharmacol Exp Ther 242:326-330.
    • (1987) J Pharmacol Exp Ther , vol.242 , pp. 326-330
    • Yamada, S.1    Ashizawa, N.2    Ushijima, H.3    Nakayama, K.4    Hayashi, E.5    Honda, K.6
  • 39
    • 0032571218 scopus 로고    scopus 로고
    • 1-adrenoceptor antagonists for treatment of benign prostatic hyperplasia
    • 1-adrenoceptor antagonists for treatment of benign prostatic hyperplasia. Life Sci 62:1585-1589.
    • (1998) Life Sci , vol.62 , pp. 1585-1589
    • Yamada, S.1    Ohkura, T.2    Kimura, R.3    Kawabe, K.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.