Total synthesis and protein kinase activity of C(7) methyl derivatives of K252a

Synthesis

Volumn , Issue SPEC. ISS., 1999, Pages 1529-1533

  Wood, John L ^a   Petsch, Dejah T ^a   Stoltz, Brian M ^a   Hawkins, Elizabeth M ^a   Elbaum, Daniel ^b   Stover, David R ^b  

^a YALE UNIVERSITY   (United States)

^b Kinetix Pharmaceuticals Inc ^*  (United States)

Author keywords

Indolocarbazole; K252a; K252a ana logs; Protein kinase; Synthesis

Indexed keywords

CARBAZOLE DERIVATIVE; INDOLE DERIVATIVE; K 252A; METHYL GROUP; PROTEIN TYROSINE KINASE; PROTEIN TYROSINE KINASE INHIBITOR;

ALZHEIMER DISEASE; ARTICLE; CANCER; CARBON NUCLEAR MAGNETIC RESONANCE; DIABETES MELLITUS; DRUG SYNTHESIS; ENZYME ACTIVITY; ENZYME INHIBITION; INFRARED SPECTROSCOPY; MASS SPECTROMETRY; METHYLATION; PROTON NUCLEAR MAGNETIC RESONANCE; RHEUMATOID ARTHRITIS; SYSTEMIC LUPUS ERYTHEMATOSUS;

EID: 0032789939     PISSN: 00397881     EISSN: None     Source Type: Journal    
DOI: 10.1055/s-1999-3652     Document Type: Article

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