메뉴 건너뛰기




Volumn , Issue 11, 1999, Pages 1751-1753

A novel strategy for the automated synthesis of bis-amides of 1,2- diamines

Author keywords

Amides; Amines; Combinatorial chemistry; Condensation; Solid phase synthesis

Indexed keywords

AMIDE; DIAMINE DERIVATIVE;

EID: 0032705782     PISSN: 09365214     EISSN: None     Source Type: Journal    
DOI: 10.1055/s-1999-2947     Document Type: Article
Times cited : (8)

References (29)
  • 1
    • 0344225389 scopus 로고    scopus 로고
    • Eur. Pat. April. EP29,602
    • AVS is cerebral vasodilator and antithrombotic agent; Mori, T.; Takaku, S.; Matsuura, F.; Murakami, Y.; Noda, Y.; Yamazaki, T.; Neichi, T.; Nakakimura, H.; Kataoka. S. Eur. Pat. April. EP29,602; CA 95: 168999t; For recent reports as hydrozxyl radical scavenger, see: Komiya, T.; Higurashi, K.; Iizuka, K.; Mizuno, Y. Clin. Neuropharmacol. 1999, 22, 11; Yamanaka, K.; Kumura, E.; Yoshimine, T.; Maruno, M.; Taniguchi, M.; Kosaka, H.; Hayakawa, T. Neurosci. Res. 1998, 31, 347; Yamamoto, K.; Ishikawa, T.; Sakabe, T.; Taguchi, T.; Kawai, S.; Marsala, M. NeuroReport 1998, 9, 1655.
    • Mori, T.1    Takaku, S.2    Matsuura, F.3    Murakami, Y.4    Noda, Y.5    Yamazaki, T.6    Neichi, T.7    Nakakimura, H.8    Kataoka, S.9
  • 2
    • 23544462549 scopus 로고    scopus 로고
    • AVS is cerebral vasodilator and antithrombotic agent; Mori, T.; Takaku, S.; Matsuura, F.; Murakami, Y.; Noda, Y.; Yamazaki, T.; Neichi, T.; Nakakimura, H.; Kataoka. S. Eur. Pat. April. EP29,602; CA 95: 168999t; For recent reports as hydrozxyl radical scavenger, see: Komiya, T.; Higurashi, K.; Iizuka, K.; Mizuno, Y. Clin. Neuropharmacol. 1999, 22, 11; Yamanaka, K.; Kumura, E.; Yoshimine, T.; Maruno, M.; Taniguchi, M.; Kosaka, H.; Hayakawa, T. Neurosci. Res. 1998, 31, 347; Yamamoto, K.; Ishikawa, T.; Sakabe, T.; Taguchi, T.; Kawai, S.; Marsala, M. NeuroReport 1998, 9, 1655.
    • CA , vol.95
  • 3
    • 0032927578 scopus 로고    scopus 로고
    • AVS is cerebral vasodilator and antithrombotic agent; Mori, T.; Takaku, S.; Matsuura, F.; Murakami, Y.; Noda, Y.; Yamazaki, T.; Neichi, T.; Nakakimura, H.; Kataoka. S. Eur. Pat. April. EP29,602; CA 95: 168999t; For recent reports as hydrozxyl radical scavenger, see: Komiya, T.; Higurashi, K.; Iizuka, K.; Mizuno, Y. Clin. Neuropharmacol. 1999, 22, 11; Yamanaka, K.; Kumura, E.; Yoshimine, T.; Maruno, M.; Taniguchi, M.; Kosaka, H.; Hayakawa, T. Neurosci. Res. 1998, 31, 347; Yamamoto, K.; Ishikawa, T.; Sakabe, T.; Taguchi, T.; Kawai, S.; Marsala, M. NeuroReport 1998, 9, 1655.
    • (1999) Clin. Neuropharmacol. , vol.22 , pp. 11
    • Komiya, T.1    Higurashi, K.2    Iizuka, K.3    Mizuno, Y.4
  • 4
    • 0031719584 scopus 로고    scopus 로고
    • AVS is cerebral vasodilator and antithrombotic agent; Mori, T.; Takaku, S.; Matsuura, F.; Murakami, Y.; Noda, Y.; Yamazaki, T.; Neichi, T.; Nakakimura, H.; Kataoka. S. Eur. Pat. April. EP29,602; CA 95: 168999t; For recent reports as hydrozxyl radical scavenger, see: Komiya, T.; Higurashi, K.; Iizuka, K.; Mizuno, Y. Clin. Neuropharmacol. 1999, 22, 11; Yamanaka, K.; Kumura, E.; Yoshimine, T.; Maruno, M.; Taniguchi, M.; Kosaka, H.; Hayakawa, T. Neurosci. Res. 1998, 31, 347; Yamamoto, K.; Ishikawa, T.; Sakabe, T.; Taguchi, T.; Kawai, S.; Marsala, M. NeuroReport 1998, 9, 1655.
    • (1998) Neurosci. Res. , vol.31 , pp. 347
    • Yamanaka, K.1    Kumura, E.2    Yoshimine, T.3    Maruno, M.4    Taniguchi, M.5    Kosaka, H.6    Hayakawa, T.7
  • 5
    • 0032507591 scopus 로고    scopus 로고
    • AVS is cerebral vasodilator and antithrombotic agent; Mori, T.; Takaku, S.; Matsuura, F.; Murakami, Y.; Noda, Y.; Yamazaki, T.; Neichi, T.; Nakakimura, H.; Kataoka. S. Eur. Pat. April. EP29,602; CA 95: 168999t; For recent reports as hydrozxyl radical scavenger, see: Komiya, T.; Higurashi, K.; Iizuka, K.; Mizuno, Y. Clin. Neuropharmacol. 1999, 22, 11; Yamanaka, K.; Kumura, E.; Yoshimine, T.; Maruno, M.; Taniguchi, M.; Kosaka, H.; Hayakawa, T. Neurosci. Res. 1998, 31, 347; Yamamoto, K.; Ishikawa, T.; Sakabe, T.; Taguchi, T.; Kawai, S.; Marsala, M. NeuroReport 1998, 9, 1655.
    • (1998) NeuroReport , vol.9 , pp. 1655
    • Yamamoto, K.1    Ishikawa, T.2    Sakabe, T.3    Taguchi, T.4    Kawai, S.5    Marsala, M.6
  • 9
    • 0342788369 scopus 로고    scopus 로고
    • John Wiley: New York
    • In Combinatorial Chemistry; Wilson, S. R.; Czarnik, A. W., Eds.; John Wiley: New York, 1997; The Combinatorial Index; Bunin, B. A.; Academic Press: New York, 1998; Solid-Supported Combinatorial and Parallel Synthesis of Small-Molecular-Weight Compound Libraries; Obrecht, D.; Villalgordo, J. M., Eds.; Pergamon: Oxford, 1998.
    • (1997) Combinatorial Chemistry
    • Wilson, S.R.1    Czarnik, A.W.2
  • 10
    • 0342788369 scopus 로고    scopus 로고
    • Academic Press: New York
    • In Combinatorial Chemistry; Wilson, S. R.; Czarnik, A. W., Eds.; John Wiley: New York, 1997; The Combinatorial Index; Bunin, B. A.; Academic Press: New York, 1998; Solid-Supported Combinatorial and Parallel Synthesis of Small-Molecular-Weight Compound Libraries; Obrecht, D.; Villalgordo, J. M., Eds.; Pergamon: Oxford, 1998.
    • (1998) The Combinatorial Index
    • Bunin, B.A.1
  • 13
    • 0028815211 scopus 로고
    • Selective amidation of primary amine in the presence of secondary amine has been reported under the equilibrium of imine and aminoacetal formation. Wang, W.; Liang, T. C.; Zheng, M.; Gao, X. Tetrahedron Lett. 1995, 36, 1181.
    • (1995) Tetrahedron Lett. , vol.36 , pp. 1181
    • Wang, W.1    Liang, T.C.2    Zheng, M.3    Gao, X.4
  • 18
    • 0030057011 scopus 로고    scopus 로고
    • Venkatesan H.; Greenberg, M. M. J. Org. Chem. 1996, 61, 525. Preparation of this linker, Landi, Jr., J. J.; Raming, K. Synth. Commun. 1991, 21, 167.
    • (1996) J. Org. Chem. , vol.61 , pp. 525
    • Venkatesan, H.1    Greenberg, M.M.2
  • 19
    • 0025872821 scopus 로고
    • Venkatesan H.; Greenberg, M. M. J. Org. Chem. 1996, 61, 525. Preparation of this linker, Landi, Jr., J. J.; Raming, K. Synth. Commun. 1991, 21, 167.
    • (1991) Synth. Commun. , vol.21 , pp. 167
    • Landi J.J., Jr.1    Raming, K.2
  • 23
    • 0344225379 scopus 로고    scopus 로고
    • It is essential to use 5% DIEA in dry dichloromethane for washing the resin avoiding cleavage of the diamine from the resin
    • It is essential to use 5% DIEA in dry dichloromethane for washing the resin avoiding cleavage of the diamine from the resin.
  • 28
    • 0345519104 scopus 로고    scopus 로고
    • Nautilus 2400 in Argonaut Technology
    • Nautilus 2400 in Argonaut Technology
  • 29
    • 0344656824 scopus 로고    scopus 로고
    • note
    • 2 313.1665, found 313.1657.


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.