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Volumn 97, Issue 1-2, 1998, Pages 13-19

MGBG analogues as potent inhibitors of S-adenosylmethionine decarboxylase of Onchocerca volvulus

Author keywords

Chemotherapy; Onchocerca volvulus; S adenosylmethionine decarboxylase

Indexed keywords

4 AMIDINO 1 INDANONE 2' AMIDINOHYDRAZONE; ADENOSYLMETHIONINE DECARBOXYLASE; DIMINAZENE ACETURATE; MITOGUAZONE; PUTRESCINE;

EID: 0032583196     PISSN: 01666851     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0166-6851(98)00124-8     Document Type: Article
Times cited : (7)

References (40)
  • 1
    • 0024153483 scopus 로고
    • The polyamine metabolism of filarial worms as chemotherapeutic target
    • Müller S., Wittich R.M., Walter R.D. The polyamine metabolism of filarial worms as chemotherapeutic target. Adv Exp Med Biol. 250:1988;737-743.
    • (1988) Adv Exp Med Biol , vol.250 , pp. 737-743
    • Müller, S.1    Wittich, R.M.2    Walter, R.D.3
  • 2
    • 0025917445 scopus 로고
    • Effect of bis(benzyl)polyamine derivatives on polyamine transport and survival of Brugia pahangi
    • Müller S., Lüchow A., McCann P.P., Walter R.D. Effect of bis(benzyl)polyamine derivatives on polyamine transport and survival of Brugia pahangi. Parasitol Res. 77:1991;612-615.
    • (1991) Parasitol Res , vol.77 , pp. 612-615
    • Müller, S.1    Lüchow, A.2    McCann, P.P.3    Walter, R.D.4
  • 3
    • 0022450919 scopus 로고
    • Recent advances in the biochemistry of polyamines in eukaryotes
    • Pegg A.E. Recent advances in the biochemistry of polyamines in eukaryotes. Biochem J. 234:1986;249-262.
    • (1986) Biochem J , vol.234 , pp. 249-262
    • Pegg, A.E.1
  • 5
    • 0027240277 scopus 로고
    • Diethylglyoxal bis(guanylhydrazone); A potent inhibitor of mammalian S-adenosylmethionine decarboxylase; Effects on cell proliferation and polyamine metabolism in L1210 leukemia cells
    • Svensson F., Kockum I., Persson L. Diethylglyoxal bis(guanylhydrazone); a potent inhibitor of mammalian S-adenosylmethionine decarboxylase; Effects on cell proliferation and polyamine metabolism in L1210 leukemia cells. Mol Cell Biochem. 124:1993;141-147.
    • (1993) Mol Cell Biochem , vol.124 , pp. 141-147
    • Svensson, F.1    Kockum, I.2    Persson, L.3
  • 6
    • 0028931579 scopus 로고
    • Antileishmanial activity of berenil and methylglyoxal bis(guanylhydrazone) and its correlation with S-adenosylmethionine decarboxylase and polyamines
    • Mukhopadhyay R., Madhubala R. Antileishmanial activity of berenil and methylglyoxal bis(guanylhydrazone) and its correlation with S-adenosylmethionine decarboxylase and polyamines. Int J Biochem Cell Biol. 27:1995;55-59.
    • (1995) Int J Biochem Cell Biol , vol.27 , pp. 55-59
    • Mukhopadhyay, R.1    Madhubala, R.2
  • 7
    • 0029901203 scopus 로고    scopus 로고
    • Antileishmanial effect of a potent S-adenosylmethionine decarboxylase inhibitor: CGP 40215A
    • Mukhopadhyay R., Kapoor P., Madhubala R. Antileishmanial effect of a potent S-adenosylmethionine decarboxylase inhibitor: CGP 40215A. Pharmacol Res. 33:1996;67-70.
    • (1996) Pharmacol Res , vol.33 , pp. 67-70
    • Mukhopadhyay, R.1    Kapoor, P.2    Madhubala, R.3
  • 8
    • 0029937062 scopus 로고    scopus 로고
    • In vivo trypanocidal activities of new S-adenosylmethionine decarboxylase inhibitors
    • Bacchi C.J., Brun R., Croft S.L., Alicea K., Buhler Y. In vivo trypanocidal activities of new S-adenosylmethionine decarboxylase inhibitors. Antimicrob Agents Chemother. 40:1996;1448-1453.
    • (1996) Antimicrob Agents Chemother , vol.40 , pp. 1448-1453
    • Bacchi, C.J.1    Brun, R.2    Croft, S.L.3    Alicea, K.4    Buhler, Y.5
  • 9
    • 0029937062 scopus 로고    scopus 로고
    • In vitro trypanocidal activities of new S-adenosylmethionine decarboxylase inhibitors
    • Brun R., Buhler Y., Sandmeier U. et al. In vitro trypanocidal activities of new S-adenosylmethionine decarboxylase inhibitors. Antimicrob Agents Chemother. 40:1996;1442-1447.
    • (1996) Antimicrob Agents Chemother , vol.40 , pp. 1442-1447
    • Brun, R.1    Buhler, Y.2    Sandmeier, U.3
  • 10
    • 0029127116 scopus 로고
    • In vivo effects of 4-amidinoindan-1-one 2′-amidinohydrazone (CGP48664A), and alpha difluoromethylornithine (DFMO) on L1210 growth, cell-cycle phase distribution and polyamine content
    • Dorhout B., Te Velde R.J., Ferwerda H., Kingma A.W., De Hoog E., Muskiet F.A.J. In vivo effects of 4-amidinoindan-1-one 2′-amidinohydrazone (CGP48664A), and alpha difluoromethylornithine (DFMO) on L1210 growth, cell-cycle phase distribution and polyamine content. Int J Cancer. 62:1995;738-742.
    • (1995) Int J Cancer , vol.62 , pp. 738-742
    • Dorhout, B.1    Te Velde, R.J.2    Ferwerda, H.3    Kingma, A.W.4    De Hoog, E.5    Muskiet, F.A.J.6
  • 11
    • 0028925525 scopus 로고
    • In vivo growth inhibition of L1210 leukemia by 4-amidinoindan-1-one 2′-amidinohydrazone (CGP 48664A), a new inhibitor of S-adenosylmethionine decarboxylase
    • Dorhout B., Te Velde R.J., Ferwerda H., Kingma A.W., De Hoog E., Muskiet F.A. In vivo growth inhibition of L1210 leukemia by 4-amidinoindan-1-one 2′-amidinohydrazone (CGP 48664A), a new inhibitor of S-adenosylmethionine decarboxylase. Int J Cancer. 61:1995;214-217.
    • (1995) Int J Cancer , vol.61 , pp. 214-217
    • Dorhout, B.1    Te Velde, R.J.2    Ferwerda, H.3    Kingma, A.W.4    De Hoog, E.5    Muskiet, F.A.6
  • 12
    • 0015505292 scopus 로고
    • Methyl glyoxal bis(guanylhydrazone) as a potent inhibitor of mammalian and yeast S-adenosylmethionine decarboxylases
    • Williams-Ashman H.G., Schenone A. Methyl glyoxal bis(guanylhydrazone) as a potent inhibitor of mammalian and yeast S-adenosylmethionine decarboxylases. Biochem Biophys Res Commun. 46:1972;288-295.
    • (1972) Biochem Biophys Res Commun , vol.46 , pp. 288-295
    • Williams-Ashman, H.G.1    Schenone, A.2
  • 13
    • 0015841716 scopus 로고
    • Effect of methylglyoxal bis(guanylhydrazone) on polyamine metabolism in normal and regenerating rat liver and rat thymus
    • Hölttä E., Hannonen P., Pispa J., Jänne J. Effect of methylglyoxal bis(guanylhydrazone) on polyamine metabolism in normal and regenerating rat liver and rat thymus. Biochem J. 136:1973;669-676.
    • (1973) Biochem J , vol.136 , pp. 669-676
    • Hölttä, E.1    Hannonen, P.2    Pispa, J.3    Jänne, J.4
  • 14
    • 0027097783 scopus 로고
    • S-Adenosylmethionine decarboxylase as an enzyme target for therapy
    • Pegg A.E., McCann P.P. S-Adenosylmethionine decarboxylase as an enzyme target for therapy. Pharmacol Ther. 56:1992;359-377.
    • (1992) Pharmacol Ther , vol.56 , pp. 359-377
    • Pegg, A.E.1    McCann, P.P.2
  • 15
    • 0026775528 scopus 로고
    • New S-adenosylmethionine decarboxylase inhibitors with potent antitumor activity
    • Regenass U., Caravatti G., Mett H. et al. New S-adenosylmethionine decarboxylase inhibitors with potent antitumor activity. Cancer Res. 52:1992;4712-4718.
    • (1992) Cancer Res , vol.52 , pp. 4712-4718
    • Regenass, U.1    Caravatti, G.2    Mett, H.3
  • 16
    • 0028361273 scopus 로고
    • CGP 48664, a new S-adenosylmethionine decarboxylase inhibitor with broad spectrum antiproliferative and antitumor activity
    • Regenass U., Mett H., Stanek J., Mueller M., Kramer D., Porter C.W. CGP 48664, a new S-adenosylmethionine decarboxylase inhibitor with broad spectrum antiproliferative and antitumor activity. Cancer Res. 54:1994;3210-3217.
    • (1994) Cancer Res , vol.54 , pp. 3210-3217
    • Regenass, U.1    Mett, H.2    Stanek, J.3    Mueller, M.4    Kramer, D.5    Porter, C.W.6
  • 17
    • 0027324170 scopus 로고
    • 4-Amidinoindan-1-one 2′-amidinohydrazone: A new potent and selective inhibitor of S-Adenosylmethionine decarboxylase
    • Stanek J., Caravatti G., Frei J., Furet P., Mett H., Schneider P., Regenass P. 4-Amidinoindan-1-one 2′-amidinohydrazone: a new potent and selective inhibitor of S-Adenosylmethionine decarboxylase. J Med Chem. 36:1993;2168-2171.
    • (1993) J Med Chem , vol.36 , pp. 2168-2171
    • Stanek, J.1    Caravatti, G.2    Frei, J.3    Furet, P.4    Mett, H.5    Schneider, P.6    Regenass, P.7
  • 18
    • 0027510003 scopus 로고
    • S-adenosylmethionine decarboxylase inhibitors: New aryl and heteroaryl analogues of methylglyoxal bis(guanylhydrazone)
    • Stanek J., Caravatti G., Capraro H. et al. S-adenosylmethionine decarboxylase inhibitors: new aryl and heteroaryl analogues of methylglyoxal bis(guanylhydrazone). J Med Chem. 36:1993;46-54.
    • (1993) J Med Chem , vol.36 , pp. 46-54
    • Stanek, J.1    Caravatti, G.2    Capraro, H.3
  • 19
    • 0029142821 scopus 로고
    • Biochemical and growth-modulatory effects of the new S-adenosylmethionine decarboxylase inhibitor CGP 48664 in malignant and immortalized normal human breast epithelial cells in culture
    • Manni A., Badger B., Wechter R., Kunselman S., Rossini A., Demers L. Biochemical and growth-modulatory effects of the new S-adenosylmethionine decarboxylase inhibitor CGP 48664 in malignant and immortalized normal human breast epithelial cells in culture. Int J Cancer. 62:1995;485-491.
    • (1995) Int J Cancer , vol.62 , pp. 485-491
    • Manni, A.1    Badger, B.2    Wechter, R.3    Kunselman, S.4    Rossini, A.5    Demers, L.6
  • 20
    • 0029004134 scopus 로고
    • Treatment of nude mice with 4-amidinoindan -1- one 2′-amidinohydrazone, a new S-adenosylmethionine decarboxylase inhibitor, delays growth and inhibits metastasis of human melanoma cells
    • Gutman M., Beltran P.J., Fan D. et al. Treatment of nude mice with 4-amidinoindan -1- one 2′-amidinohydrazone, a new S-adenosylmethionine decarboxylase inhibitor, delays growth and inhibits metastasis of human melanoma cells. Melanoma Res. 5:1995;147-154.
    • (1995) Melanoma Res , vol.5 , pp. 147-154
    • Gutman, M.1    Beltran, P.J.2    Fan, D.3
  • 21
    • 0031045715 scopus 로고    scopus 로고
    • CGP 48664, a potent and specific S-adenosylmethionine decarboxylase inhibitor: Effects on regulation and stability of the enzyme
    • Svensson F., Mett H., Persson L. CGP 48664, a potent and specific S-adenosylmethionine decarboxylase inhibitor: effects on regulation and stability of the enzyme. Biochem J. 322:1997;297-302.
    • (1997) Biochem J , vol.322 , pp. 297-302
    • Svensson, F.1    Mett, H.2    Persson, L.3
  • 22
    • 0029853782 scopus 로고    scopus 로고
    • A novel trans-spliced mRNA from O. volvulus encodes a functional S-adenosylmethionine decarboxylase
    • Da'dara A.A., Henkle-Dührsen K., Walter R.D. A novel trans-spliced mRNA from O. volvulus encodes a functional S-adenosylmethionine decarboxylase. Biochem J. 320:1996;519-530.
    • (1996) Biochem J , vol.320 , pp. 519-530
    • Da'dara, A.A.1    Henkle-Dührsen, K.2    Walter, R.D.3
  • 23
    • 0017184389 scopus 로고
    • A rapid and a sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding
    • Bradford M.M. A rapid and a sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding. Anal Biochem. 72:1979;248-254.
    • (1979) Anal Biochem , vol.72 , pp. 248-254
    • Bradford, M.M.1
  • 24
    • 0023908603 scopus 로고
    • Ascaris suum and O. volvulus: S-adenosylmethionine decarboxylase
    • Rathaur S., Wittich R.M., Walter R.D. Ascaris suum and O. volvulus: S-Adenosylmethionine decarboxylase. Exp Parasitol. 65:1988;277-281.
    • (1988) Exp Parasitol , vol.65 , pp. 277-281
    • Rathaur, S.1    Wittich, R.M.2    Walter, R.D.3
  • 25
    • 0015327378 scopus 로고
    • A linear equation that describes the steady-state kinetics of enzymes and subcellular particles interacting with tightly bound inhibitors
    • Henderson P.J.F. A linear equation that describes the steady-state kinetics of enzymes and subcellular particles interacting with tightly bound inhibitors. Biochem J. 127:1972;321-333.
    • (1972) Biochem J , vol.127 , pp. 321-333
    • Henderson, P.J.F.1
  • 26
    • 73649151319 scopus 로고
    • Esters of methanesulfonic acid as irreversible inhibitors of acetylcholinesterase
    • Kitz R, Wilson IB. Esters of methanesulfonic acid as irreversible inhibitors of acetylcholinesterase, J Biol Chem 1962;237:3245-9.
    • (1962) J Biol Chem , vol.237 , pp. 3245-3249
    • Kitz, R.1    Wilson, I.B.2
  • 27
    • 0016236847 scopus 로고
    • Purification of rat liver S-adenosylmethionine decarboxylase
    • Pegg A.E. Purification of rat liver S-adenosylmethionine decarboxylase. Biochem J. 141:1974;581-583.
    • (1974) Biochem J , vol.141 , pp. 581-583
    • Pegg, A.E.1
  • 28
    • 0023140148 scopus 로고
    • Putrescine-activated S-adenosylmethionine decarboxylase from Acanthamoeba culbertsoni
    • Gupta S., Shukla O.P., Walter R.D. Putrescine-activated S-adenosylmethionine decarboxylase from Acanthamoeba culbertsoni. Mol Biochem Parasitol. 23:1987;247-252.
    • (1987) Mol Biochem Parasitol , vol.23 , pp. 247-252
    • Gupta, S.1    Shukla, O.P.2    Walter, R.D.3
  • 29
    • 0027438385 scopus 로고
    • S-adenosyl-L-methionine decarboxylase of Acanthamoeba castellanii (Neff): Purification and properties
    • Hugo E.R., Byers T.J. S-adenosyl-L-methionine decarboxylase of Acanthamoeba castellanii (Neff): purification and properties. Biochem J. 295:1993;203-209.
    • (1993) Biochem J , vol.295 , pp. 203-209
    • Hugo, E.R.1    Byers, T.J.2
  • 31
    • 0022454288 scopus 로고
    • Characterization of Trypanosoma brucei brucei S-adenosyl-L-methionine decarboxylase and its inhibition by berenil; Pentamidine and methylglyoxal bis(guanylhydrazone)
    • Bitonti A.J., Dumont J.A., McCann P.P. Characterization of Trypanosoma brucei brucei S-adenosyl-L-methionine decarboxylase and its inhibition by berenil; pentamidine and methylglyoxal bis(guanylhydrazone). Biochem J. 237:1986;685-689.
    • (1986) Biochem J , vol.237 , pp. 685-689
    • Bitonti, A.J.1    Dumont, J.A.2    McCann, P.P.3
  • 32
    • 0020805604 scopus 로고
    • Comparison of inhibitors of S-adenosylmethionine decarboxylase from different species
    • Pegg A.E., Jacob G. Comparison of inhibitors of S-adenosylmethionine decarboxylase from different species. Biochem J. 213:1983;495-502.
    • (1983) Biochem J , vol.213 , pp. 495-502
    • Pegg, A.E.1    Jacob, G.2
  • 33
    • 0022553584 scopus 로고
    • Inhibition of diamine oxidase and S-adenosylmethionine decarboxylase by diminacene aceturate (berenil)
    • Balana-Fouce R., Garzon Pulido T., Ordonez-Escudero D., Garrido-Pertierra A. Inhibition of diamine oxidase and S-adenosylmethionine decarboxylase by diminacene aceturate (berenil). Biochem Pharmacol. 35:1986;1597-1600.
    • (1986) Biochem Pharmacol , vol.35 , pp. 1597-1600
    • Balana-Fouce, R.1    Garzon Pulido, T.2    Ordonez-Escudero, D.3    Garrido-Pertierra, A.4
  • 34
    • 0026532347 scopus 로고
    • Purification and characterization of polyamine oxidase from Ascaris suum
    • Müller S., Walter R.D. Purification and characterization of polyamine oxidase from Ascaris suum. Biochem J. 283:1992;75-80.
    • (1992) Biochem J , vol.283 , pp. 75-80
    • Müller, S.1    Walter, R.D.2
  • 35
    • 0024809887 scopus 로고
    • 5′-{[(Z)-4-Amino-2-butenyl]methylamino}-5′-deoxyadenosine: A potent enzyme-activated irreversible inhibitor of S-adenosylmethionine decarboxylase from E. coli
    • Casara P., Marchal P., Wagner J., Danzin C. 5′-{[(Z)-4-Amino-2-butenyl]methylamino}-5′-deoxyadenosine: a potent enzyme-activated irreversible inhibitor of S-adenosylmethionine decarboxylase from E. coli. J Am Chem Soc. 111:1989;9111-9113.
    • (1989) J Am Chem Soc , vol.111 , pp. 9111-9113
    • Casara, P.1    Marchal, P.2    Wagner, J.3    Danzin, C.4
  • 36
    • 0024999490 scopus 로고
    • Irreversible inhibition of rat S-adenosylmethionine decarboxylase by 5′-{[(Z)-4-amino-2-butenyl]methylamino}-5′-deoxyadenosine
    • Danzin C., Marchal P., Casara P. Irreversible inhibition of rat S-adenosylmethionine decarboxylase by 5′-{[(Z)-4-amino-2-butenyl]methylamino}-5′-deoxyadenosine. Biochem Pharmacol. 40:1990;1499-1503.
    • (1990) Biochem Pharmacol , vol.40 , pp. 1499-1503
    • Danzin, C.1    Marchal, P.2    Casara, P.3
  • 37
    • 0025180260 scopus 로고
    • Cure of Trypanosoma brucei brucei and Trypanosoma brucei rhodesiense infections in mice with an irreversible inhibitor of S-adenosylmethionine decarboxylase
    • Bitonti A.J., Byers T.L., Bush T.L. et al. Cure of Trypanosoma brucei brucei and Trypanosoma brucei rhodesiense infections in mice with an irreversible inhibitor of S-adenosylmethionine decarboxylase. Antimicrob Agents Chemother. 34:1990;1485-1490.
    • (1990) Antimicrob Agents Chemother , vol.34 , pp. 1485-1490
    • Bitonti, A.J.1    Byers, T.L.2    Bush, T.L.3
  • 38
    • 0026033857 scopus 로고
    • Antitrypanosomal effects of polyamine biosynthesis inhibitors correlate with increases in Trypanosoma brucei brucei S-adenosyl-L-methionine
    • Byers T.L., Bush T.L., McCann P.P., Bitonti A.J. Antitrypanosomal effects of polyamine biosynthesis inhibitors correlate with increases in Trypanosoma brucei brucei S-adenosyl-L-methionine. Biochem J. 274:1991;527-533.
    • (1991) Biochem J , vol.274 , pp. 527-533
    • Byers, T.L.1    Bush, T.L.2    McCann, P.P.3    Bitonti, A.J.4
  • 39
    • 0025780218 scopus 로고
    • Irreversible inhibition of S-adenosylmethionine decarboxylase in Plasmodium falciparum-infected erythrocytes: Growth inhibition in vitro
    • Wright P.S., Byers T.L., Cross-Doersen D.E. Irreversible inhibition of S-adenosylmethionine decarboxylase in Plasmodium falciparum-infected erythrocytes: growth inhibition in vitro. Biochem Pharmacol. 41:1991;1713-1718.
    • (1991) Biochem Pharmacol , vol.41 , pp. 1713-1718
    • Wright, P.S.1    Byers, T.L.2    Cross-Doersen, D.E.3
  • 40
    • 0002861247 scopus 로고
    • Modulation of antineoplastic drug action by inhibitors of polyamine biosynthesis
    • McCann PP, Pegg AE, Sjoerdsma A, editors. San Diego: Academic Press
    • Porter CW, Jänne J. Modulation of antineoplastic drug action by inhibitors of polyamine biosynthesis. In: McCann PP, Pegg AE, Sjoerdsma A, editors. Inhibition of Polyamine Metabolism, Biological Significance and Basis for New Therapies. San Diego: Academic Press, 1987:203-248.
    • (1987) Inhibition of Polyamine Metabolism, Biological Significance and Basis for New Therapies , pp. 203-248
    • Porter, C.W.1    Jänne, J.2


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