A trypanosome oligopeptidase as a target for the trypanocidal agents pentamidine, diminazene and suramin

FEBS Letters

Volumn 433, Issue 3, 1998, Pages 251-256

  Morty, Rory E ^a   Troeberg, Linda ^a   Pike, Robert N ^b   Jones, Roy ^c   Nickel, Peter ^d   Lonsdale Eccles, John D ^e   Coetzer, Theresa H T ^a  

^a UNIVERSITY OF KWAZULU NATAL   (South Africa)

^b MONASH UNIVERSITY   (Australia)

^c BABRAHAM INSTITUTE   (United Kingdom)

^d UNIVERSITY OF BONN   (Germany)

^e UNIVERSITY OF ALABAMA AT BIRMINGHAM   (United States)

Author keywords

Diminazene; Oligopeptidase; Pentamidine; Protease; Suramin; Trypanosoma brucei

Indexed keywords

TRYPANOSOMA; TRYPANOSOMA BRUCEI;

ANTITRYPANOSOMAL AGENT; DIMINAZENE; DRUG DERIVATIVE; OLIGOPEPTIDASE TB; PENTAMIDINE; SERINE PROTEINASE; SERINE PROTEINASE INHIBITOR; SURAMIN;

ANIMAL; ARTICLE; DRUG EFFECT; ENZYMOLOGY; METABOLISM; STRUCTURE ACTIVITY RELATION; TRYPANOSOMA;

ANIMALS; DIMINAZENE; PENTAMIDINE; SERINE ENDOPEPTIDASES; SERINE PROTEINASE INHIBITORS; STRUCTURE-ACTIVITY RELATIONSHIP; SURAMIN; TRYPANOCIDAL AGENTS; TRYPANOSOMA;

EID: 0032555363     PISSN: 00145793     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-5793(98)00914-4     Document Type: Article

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