메뉴 건너뛰기




Volumn 165, Issue 1, 1998, Pages 45-55

Effect of oleic acid/ethanol and oleic acid/propylene glycol on the in vitro percutaneous absorption of 5-fluorouracil and tamoxifen and the macroscopic barrier property of porcine epidermis

Author keywords

5 Fluorouracil; Oleic acid; Percutaneous absorption; Tamoxifen; Transepidermal water loss

Indexed keywords

ALCOHOL; FLUOROURACIL; OLEIC ACID; PROPYLENE GLYCOL; TAMOXIFEN;

EID: 0032550357     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0378-5173(97)00430-4     Document Type: Article
Times cited : (54)

References (51)
  • 2
    • 0023001444 scopus 로고
    • Enhancement of naloxone penetration through human skin in vitro using fatty acids, fatty alcohols, surfactant, sulfoxides and amides
    • Aungst B.J., Rogers N.J., Shefter E. Enhancement of naloxone penetration through human skin in vitro using fatty acids, fatty alcohols, surfactant, sulfoxides and amides. Int. J. Pharm. 33:1986;225-234.
    • (1986) Int. J. Pharm. , vol.33 , pp. 225-234
    • Aungst, B.J.1    Rogers, N.J.2    Shefter, E.3
  • 3
    • 0025906898 scopus 로고
    • Lipid-protein-partitioning theory of skin penetration enhancement
    • Barry B.W. Lipid-protein-partitioning theory of skin penetration enhancement. J. Control. Release. 15:1991;237-248.
    • (1991) J. Control. Release , vol.15 , pp. 237-248
    • Barry, B.W.1
  • 4
    • 0023235207 scopus 로고
    • Effect of penetration enhancers on the permeation of mannitol, hydrocortisone and progesterone throught human skin
    • Barry B.W., Bennett S.L. Effect of penetration enhancers on the permeation of mannitol, hydrocortisone and progesterone throught human skin. J. Pharm. Pharmacol. 39:1987;535-546.
    • (1987) J. Pharm. Pharmacol. , vol.39 , pp. 535-546
    • Barry, B.W.1    Bennett, S.L.2
  • 5
    • 0031003156 scopus 로고    scopus 로고
    • Effect of penetration enhancers and iontophoresis on the FT-IR spectroscopy and LHRH permeability through porcine skin
    • Bhatia K.S., Gao S., Singh J. Effect of penetration enhancers and iontophoresis on the FT-IR spectroscopy and LHRH permeability through porcine skin. J. Control. Release. 47:1997;81-89.
    • (1997) J. Control. Release , vol.47 , pp. 81-89
    • Bhatia, K.S.1    Gao, S.2    Singh, J.3
  • 6
    • 0030765030 scopus 로고    scopus 로고
    • Effect of penetration enhancers and iontophoresis on the ultrastructure and cholecystokinin-8 permeability through porcine skin
    • Bhatia K.S., Gao S., Freeman T.P., Singh J. Effect of penetration enhancers and iontophoresis on the ultrastructure and cholecystokinin-8 permeability through porcine skin. J. Pharm. Sci. 89:1997;1011-1015.
    • (1997) J. Pharm. Sci. , vol.89 , pp. 1011-1015
    • Bhatia, K.S.1    Gao, S.2    Freeman, T.P.3    Singh, J.4
  • 7
    • 0021954919 scopus 로고
    • Optimization of bioavailability of topical steroids: Non-occluded penetration enhancers under thermodynamic control
    • Bennett S.L., Barry B.W., Woodford R. Optimization of bioavailability of topical steroids: non-occluded penetration enhancers under thermodynamic control. J. Pharm. Pharmacol. 37:1985;298-304.
    • (1985) J. Pharm. Pharmacol. , vol.37 , pp. 298-304
    • Bennett, S.L.1    Barry, B.W.2    Woodford, R.3
  • 8
    • 0018093266 scopus 로고
    • The effect of gramicidin A on the temperature dependence of water permeation through liposomal membranes prepared from phosphatidylcholines with different chains lengths
    • Boehler B.A., De Gier J., Van Deenen L.L.M. The effect of gramicidin A on the temperature dependence of water permeation through liposomal membranes prepared from phosphatidylcholines with different chains lengths. Biochim. Biophys. Acta. 512:1978;480-488.
    • (1978) Biochim. Biophys. Acta , vol.512 , pp. 480-488
    • Boehler, B.A.1    De Gier, J.2    Van Deenen, L.L.M.3
  • 9
    • 0023926924 scopus 로고
    • Hairless mouse skin is limited as a model for assessing the effects of penetration enhancers in human skin
    • Bond J.R., Barry B.W. Hairless mouse skin is limited as a model for assessing the effects of penetration enhancers in human skin. J. Invest. Dermatol. 90:1988;810-813.
    • (1988) J. Invest. Dermatol. , vol.90 , pp. 810-813
    • Bond, J.R.1    Barry, B.W.2
  • 10
    • 0024467413 scopus 로고
    • Alkyl esters as skin permeation enhancers for indomethacin
    • Catz P., Friend D.R. Alkyl esters as skin permeation enhancers for indomethacin. Int. J. Pharm. 55:1989;17-23.
    • (1989) Int. J. Pharm. , vol.55 , pp. 17-23
    • Catz, P.1    Friend, D.R.2
  • 11
    • 0029807016 scopus 로고    scopus 로고
    • Influence of polyethylene glycol and acetone on the in vitro biotransformation of tamoxifen and alprazolam by human liver microsomes
    • Cotreau-Bibbo M.M., Von Moltke L.L., Greenblatt D.J. Influence of polyethylene glycol and acetone on the in vitro biotransformation of tamoxifen and alprazolam by human liver microsomes. J. Pharm. Sci. 85:1996;1180-1185.
    • (1996) J. Pharm. Sci. , vol.85 , pp. 1180-1185
    • Cotreau-Bibbo, M.M.1    Von Moltke, L.L.2    Greenblatt, D.J.3
  • 12
    • 0001855293 scopus 로고
    • Tansepidermal water loss
    • In: Berardesca, E., Elsner, P., Wilhelm, K.P., Maibach, H.I. (Eds.), CRC Press, Boca Raton
    • Distante, F., Berardesca, E., 1995. Tansepidermal water loss. In: Berardesca, E., Elsner, P., Wilhelm, K.P., Maibach, H.I. (Eds.), Bioengineering of the skin: Methods and Instrumentation. CRC Press, Boca Raton, pp. 1-4.
    • (1995) Bioengineering of the Skin: Methods and Instrumentation , pp. 1-4
    • Distante, F.1    Berardesca, E.2
  • 13
    • 0020608231 scopus 로고
    • Epidermal lipids, barrier function, and desquamation
    • Elias P.M. Epidermal lipids, barrier function, and desquamation. J. Invest. Dermatol. 80:1983;44s-49s.
    • (1983) J. Invest. Dermatol. , vol.80
    • Elias, P.M.1
  • 14
    • 0015030515 scopus 로고
    • Structural approach to partitioning: Estimation of steroid partition coefficients based upon molecular constitution
    • Flynn G.L. Structural approach to partitioning: Estimation of steroid partition coefficients based upon molecular constitution. J. Pharm. Sci. 60:1971;345-353.
    • (1971) J. Pharm. Sci. , vol.60 , pp. 345-353
    • Flynn, G.L.1
  • 15
    • 0002448680 scopus 로고
    • Mechanism of percutaneous absorption from physicochemical evidence
    • In: Bronaugh, R.L., Maibach, H.I. (Eds.), Marcel Dekker, New York
    • Flynn, G.L., 1989. Mechanism of percutaneous absorption from physicochemical evidence. In: Bronaugh, R.L., Maibach, H.I. (Eds.), Percutaneous Absorption. Marcel Dekker, New York, pp. 27-51.
    • (1989) Percutaneous Absorption , pp. 27-51
    • Flynn, G.L.1
  • 16
    • 0024246628 scopus 로고
    • Percutaneous drug penetration: Choosing candidates for transdermal development
    • Flynn G.L., Stewart B. Percutaneous drug penetration: Choosing candidates for transdermal development. Drug Dev. Res. 13:1988;169-185.
    • (1988) Drug Dev. Res. , vol.13 , pp. 169-185
    • Flynn, G.L.1    Stewart, B.2
  • 17
    • 0030787333 scopus 로고    scopus 로고
    • Mechanism of transdermal transport of 5-fluorouracil by terpenes: Carvone, 1,8-cineole and thymol
    • Gao S., Singh J. Mechanism of transdermal transport of 5-fluorouracil by terpenes: carvone, 1,8-cineole and thymol. Int. J. Pharm. 154:1997;67-77.
    • (1997) Int. J. Pharm. , vol.154 , pp. 67-77
    • Gao, S.1    Singh, J.2
  • 18
  • 19
    • 0024804574 scopus 로고
    • Lipid-protein-partitioning (LPP) theory of skin enhancer activity: Finite dose technique
    • Goodman M., Barry B.W. Lipid-protein-partitioning (LPP) theory of skin enhancer activity: finite dose technique. Int. J. Pharm. 57:1989;29-40.
    • (1989) Int. J. Pharm. , vol.57 , pp. 29-40
    • Goodman, M.1    Barry, B.W.2
  • 20
    • 0025242415 scopus 로고
    • Endocrine pharmacology of antiestrogens as antitumor agents
    • Jordan V.C., Murphy C.S. Endocrine pharmacology of antiestrogens as antitumor agents. Endocr. Rev. 11:1990;49-81.
    • (1990) Endocr. Rev. , vol.11 , pp. 49-81
    • Jordan, V.C.1    Murphy, C.S.2
  • 21
    • 0002784494 scopus 로고
    • Update: Breast cancer treatment and prevention with antiestrogens in the 1990s
    • Jordan V.C., Parker C.J., Marrow M. Update: breast cancer treatment and prevention with antiestrogens in the 1990s. Endocr. Rev. 1:1993;82-85.
    • (1993) Endocr. Rev. , vol.1 , pp. 82-85
    • Jordan, V.C.1    Parker, C.J.2    Marrow, M.3
  • 23
    • 0023254185 scopus 로고
    • In vivo relationship between transepidermal water loss and percutaneous penetration of some organic compounds in man: Effect of anatomic site
    • Lotte C., Rougier A., Wilson D.R., Maibach H.I. In vivo relationship between transepidermal water loss and percutaneous penetration of some organic compounds in man: effect of anatomic site. Arch. Dermatol. Res. 279:1987;351-356.
    • (1987) Arch. Dermatol. Res. , vol.279 , pp. 351-356
    • Lotte, C.1    Rougier, A.2    Wilson, D.R.3    Maibach, H.I.4
  • 24
    • 0003143831 scopus 로고
    • Noninvasive techniques for determining skin function
    • In: Drill, V.A., Lazar, P. (Eds.), Raven Press, New York
    • Maibach, H.I., Bronaugh, R., Guy, R., Turr, E., Wilson, D., Jacques, S., Chaing, D., 1984. Noninvasive techniques for determining skin function. In: Drill, V.A., Lazar, P. (Eds.), Cutaneous Toxicity. Raven Press, New York, pp. 63-97.
    • (1984) Cutaneous Toxicity , pp. 63-97
    • Maibach, H.I.1    Bronaugh, R.2    Guy, R.3    Turr, E.4    Wilson, D.5    Jacques, S.6    Chaing, D.7
  • 25
    • 0028861288 scopus 로고
    • Oestradiol permeation across human skin, silastic and snake skin membranes: The effects of ethanol/water co-solvent system
    • Megrab N.A., Williams A.C., Barry B.W. Oestradiol permeation across human skin, silastic and snake skin membranes: the effects of ethanol/water co-solvent system. Int. J. Pharm. 116:1995;101-112.
    • (1995) Int. J. Pharm. , vol.116 , pp. 101-112
    • Megrab, N.A.1    Williams, A.C.2    Barry, B.W.3
  • 26
    • 0029585859 scopus 로고
    • Mechanism of oleic acid-induced skin penetration enhancement in vivo in humans
    • Naik A., Petchtold L.A.R.M., Potts R.O., Guy R.H. Mechanism of oleic acid-induced skin penetration enhancement in vivo in humans. J. Control. Release. 37:1995;299-306.
    • (1995) J. Control. Release , vol.37 , pp. 299-306
    • Naik, A.1    Petchtold, L.A.R.M.2    Potts, R.O.3    Guy, R.H.4
  • 28
    • 0025905320 scopus 로고
    • Evidence that oleic acid exists in a separate phase within stratum corneum lipids
    • Ongpipattanakul B., Burnette R.R., Potts R.O., Francoeur M.L. Evidence that oleic acid exists in a separate phase within stratum corneum lipids. Pharm. Res. 8:1991;350-354.
    • (1991) Pharm. Res. , vol.8 , pp. 350-354
    • Ongpipattanakul, B.1    Burnette, R.R.2    Potts, R.O.3    Francoeur, M.L.4
  • 29
    • 0025372245 scopus 로고
    • Lipid biophysics of water loss through the skin
    • Potts R.O., Francoeur M.L. Lipid biophysics of water loss through the skin. Proc. Natl. Acad. Sci. USA. 87:1990;3871-3873.
    • (1990) Proc. Natl. Acad. Sci. USA , vol.87 , pp. 3871-3873
    • Potts, R.O.1    Francoeur, M.L.2
  • 31
    • 0027379355 scopus 로고
    • Electroporation of mammalian skin: A mechanism to enhance transdermal drug delivery
    • Prausnitz M.R., Bose V.G., Langer R., Weaver J.C. Electroporation of mammalian skin: a mechanism to enhance transdermal drug delivery. Proc. Natl. Acad. Sci. USA. 90:1993;10504-10508.
    • (1993) Proc. Natl. Acad. Sci. USA , vol.90 , pp. 10504-10508
    • Prausnitz, M.R.1    Bose, V.G.2    Langer, R.3    Weaver, J.C.4
  • 32
    • 0018142096 scopus 로고
    • The percutaneous absorption of phenolic compounds: The mechanism of diffusion across the stratum corneum
    • Roberts M.S., Anderson R.A., Swarbrick J., Moore D.E. The percutaneous absorption of phenolic compounds: the mechanism of diffusion across the stratum corneum. J. Pharm. Pharmcol. 30:1978;486-490.
    • (1978) J. Pharm. Pharmcol. , vol.30 , pp. 486-490
    • Roberts, M.S.1    Anderson, R.A.2    Swarbrick, J.3    Moore, D.E.4
  • 33
    • 0001010974 scopus 로고
    • In vivo relationship between percutaneous absorption and transepidermal water loss
    • In: Bronaugh, R.L., Maibach, H.I. (Eds), Marcel Dekker, New York
    • Rougier, A., Lotte, C., Maibach, H.I., 1989. In vivo relationship between percutaneous absorption and transepidermal water loss. In: Bronaugh, R.L., Maibach, H.I. (Eds), Percutaneous Absorption. Marcel Dekker, New York, pp. 175-190.
    • (1989) Percutaneous Absorption , pp. 175-190
    • Rougier, A.1    Lotte, C.2    Maibach, H.I.3
  • 34
    • 0001517668 scopus 로고
    • Skin as barrier
    • In: Jarret, A. (Ed.), Academic press, New York
    • Scheuplein, R.J., 1978. Skin as barrier. In: Jarret, A. (Ed.), The physiology and pathophysiology of skin. Academic press, New York, pp. 1693-1730.
    • (1978) The Physiology and Pathophysiology of Skin , pp. 1693-1730
    • Scheuplein, R.J.1
  • 37
    • 0030003515 scopus 로고    scopus 로고
    • Topical iontophoretic drug delivery: Pathways, principles, factors and skin irritation
    • Singh J., Bhatia K.S. Topical iontophoretic drug delivery: pathways, principles, factors and skin irritation. Med. Res. Rev. 16:1996;285-296.
    • (1996) Med. Res. Rev. , vol.16 , pp. 285-296
    • Singh, J.1    Bhatia, K.S.2
  • 38
    • 0025355927 scopus 로고
    • Transdermal delivery of drugs by phonophoresis: A review
    • Singh S., Singh J. Transdermal delivery of drugs by phonophoresis: a review. Drug Des. Deliv. 5:1990;259-265.
    • (1990) Drug Des. Deliv. , vol.5 , pp. 259-265
    • Singh, S.1    Singh, J.2
  • 39
    • 85057221346 scopus 로고
    • Percutaneous penetration enhancers: The fundamental
    • In: Smith, E.W., Maibach, H.I. (Eds.), CRC Press, Boca Raton
    • Smith, E.W., Maibach, H.I., 1995. Percutaneous penetration enhancers: the fundamental. In: Smith, E.W., Maibach, H.I. (Eds.), Percutaneous Penetration Enhancers. CRC Press, Boca Raton, pp 1-4.
    • (1995) Percutaneous Penetration Enhancers , pp. 1-4
    • Smith, E.W.1    Maibach, H.I.2
  • 40
    • 0029025533 scopus 로고
    • Human skin permeability enhancement by lauric acid under equilibrium aqueous conditions
    • Smith S.W., Anderson B.D. Human skin permeability enhancement by lauric acid under equilibrium aqueous conditions. J. Pharm. Sci. 84:1995;551-556.
    • (1995) J. Pharm. Sci. , vol.84 , pp. 551-556
    • Smith, S.W.1    Anderson, B.D.2
  • 41
    • 0027289132 scopus 로고
    • Enhanced delivery of 5-fluorouracil through shed snake skin by two new transdermal penetration enhancers
    • Turunen T.M., Buyuktimkin S., Buyuktimkin N., Urtti A., Paronen P., Rytting J.H. Enhanced delivery of 5-fluorouracil through shed snake skin by two new transdermal penetration enhancers. Int. J. Pharm. 92:1993;89-95.
    • (1993) Int. J. Pharm. , vol.92 , pp. 89-95
    • Turunen, T.M.1    Buyuktimkin, S.2    Buyuktimkin, N.3    Urtti, A.4    Paronen, P.5    Rytting, J.H.6
  • 42
    • 16344375748 scopus 로고    scopus 로고
    • Dug information for the health care professional
    • USP DI, Rockville, MD
    • USP DI, 1997. Dug information for the health care professional, US Pharmacopeial Convention, Rockville, MD, pp. 1496-1502.
    • (1997) US Pharmacopeial Convention , pp. 1496-1502
  • 43
    • 0016737528 scopus 로고
    • Thermal analysis of human stratum corneum
    • Van Duzee B.F. Thermal analysis of human stratum corneum. J. Invest. Dermatol. 65:1971;404-408.
    • (1971) J. Invest. Dermatol. , vol.65 , pp. 404-408
    • Van Duzee, B.F.1
  • 44
    • 0028347451 scopus 로고
    • Alveolar permeability enhancement by oleic acid and related fatty acids: Evidence for a calcium-dependent mechanism
    • Wang L.Y., Ma J.K., Pan W.F., Toledo-Velasquez D., Malanga C.J., Rojanasakul Y. Alveolar permeability enhancement by oleic acid and related fatty acids: evidence for a calcium-dependent mechanism. Pharm. Res. 11:1994;513-517.
    • (1994) Pharm. Res. , vol.11 , pp. 513-517
    • Wang, L.Y.1    Ma, J.K.2    Pan, W.F.3    Toledo-Velasquez, D.4    Malanga, C.J.5    Rojanasakul, Y.6
  • 45
    • 0020000879 scopus 로고
    • Glycolipids in mammalian epidermis: Structure and function in the water barrier
    • Wertz P.M., Downing D.T. Glycolipids in mammalian epidermis: structure and function in the water barrier. Science. 217:1982;1261-1262.
    • (1982) Science , vol.217 , pp. 1261-1262
    • Wertz, P.M.1    Downing, D.T.2
  • 48
    • 0001951787 scopus 로고
    • A review of transepidermal water loss: physical aspects and measurements as related to infants and adults
    • In: Maibach, H.I., Bouititis, E.K. (Eds.), Marcel Dekker, New York
    • Wilson, D.R., Maibach, H.I., 1982. A review of transepidermal water loss: physical aspects and measurements as related to infants and adults. In: Maibach, H.I., Bouititis, E.K. (Eds.), Neonatal Skin. Marcel Dekker, New York, pp. 83-100.
    • (1982) Neonatal Skin , pp. 83-100
    • Wilson, D.R.1    Maibach, H.I.2
  • 49
    • 0022458160 scopus 로고
    • Relationship between lipid fluidity and water permeability of bovine tracheal epithelial cell apical membranes
    • Worman H.J., Brasitus T.A., Dudeja P.K., Fozzard H.A., Field M. Relationship between lipid fluidity and water permeability of bovine tracheal epithelial cell apical membranes. Biochemistry. 25:1986;1549-1555.
    • (1986) Biochemistry , vol.25 , pp. 1549-1555
    • Worman, H.J.1    Brasitus, T.A.2    Dudeja, P.K.3    Fozzard, H.A.4    Field, M.5
  • 50
    • 0028830178 scopus 로고
    • Effects of terpenes and oleic acid as skin penetration enhancers towards 5-fluorouracil as assessed with time; Permeation, partitioning and differential scanning calorimetry
    • Yamane M.A., William A.C., Barry B.W. Effects of terpenes and oleic acid as skin penetration enhancers towards 5-fluorouracil as assessed with time; permeation, partitioning and differential scanning calorimetry. Int. J. Pharm. 116:1995;237-251.
    • (1995) Int. J. Pharm. , vol.116 , pp. 237-251
    • Yamane, M.A.1    William, A.C.2    Barry, B.W.3
  • 51
    • 0023713886 scopus 로고
    • Percutaneous absorption of nicardipine and ketorolac in rhesus monkeys
    • Yu D., Sanders L.M., Davidson G.W., Marvin M.J., Ling T. Percutaneous absorption of nicardipine and ketorolac in rhesus monkeys. Pharm. Res. 5:1988;457-462.
    • (1988) Pharm. Res. , vol.5 , pp. 457-462
    • Yu, D.1    Sanders, L.M.2    Davidson, G.W.3    Marvin, M.J.4    Ling, T.5


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.