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Superimposition was calculated by Molecular Modeling System SYBYL, Version 6.2; Tripos Associates, Inc.
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14. Fragments of colon 26 tumor (5mg) were inoculated sc into CD2F1 mice. Test compounds were given iv or sc on days 7, 11 and 15. On day 21, the tumor weights were measured. The inhibition ratio was evaluated as (1-T/C)X100 (%) (T; the mean tumor weight of the treated group, C; the mean tumor weight of the control group). Each group consisted of 5 mice.
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