Synthesis and transporter binding properties of (R)-2β,3β- and (R)- 2α,3α-diaryltropanes

Bioorganic and Medicinal Chemistry Letters

Volumn 8, Issue 24, 1998, Pages 3689-3692

  Jiang, Songchun ^a   Chang, An Chih ^a   Abraham, Philip ^a   Kuhar, Michael J ^b   Carroll, F Ivy ^a  

^a RTI INTERNATIONAL   (United States)

^b EMORY UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

2 CARBOMETHOXY 3 TROPINONE; 3BETA (4 METHYLPHENYL) 2BETA PHENYLTROPANE; COCAINE; DOPAMINE TRANSPORTER; NORADRENALIN; RADIOLIGAND; SEROTONIN TRANSPORTER; TROPANE DERIVATIVE; TROPARIL; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; DRUG POTENCY; STEREOISOMERISM; SYNTHESIS;

CARRIER PROTEINS; DOPAMINE; DOPAMINE PLASMA MEMBRANE TRANSPORT PROTEINS; MEMBRANE GLYCOPROTEINS; MEMBRANE TRANSPORT PROTEINS; NERVE TISSUE PROTEINS; NOREPINEPHRINE; NOREPINEPHRINE PLASMA MEMBRANE TRANSPORT PROTEINS; PROTEIN BINDING; RADIOLIGAND ASSAY; SEROTONIN; SEROTONIN PLASMA MEMBRANE TRANSPORT PROTEINS; SYMPORTERS; TROPANES;

EID: 0032534885     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(98)00673-8     Document Type: Article

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