Stimulation of L-type Ca2+ current by the endothelin receptor A- selective antagonist, BQ-123, in ventricular cardiomyocytes isolated from rabbit myocardium

Biochemical Pharmacology

Volumn 55, Issue 6, 1998, Pages 897-902

  Kelso, Elizabeth J ^a   Spiers, J Paul ^a   McDermott, Barbara J ^a   Scholfield, C Norman ^a   Silke, Bernard ^a  

^a QUEEN'S UNIVERSITY BELFAST   (United Kingdom)

Author keywords

BQ 123; BQ 788; Ca2+ current; Endothelin 1; ET(A) receptor antagonist; PD145065; PD155080; Ventricular cardiomyocytes

Indexed keywords

3 BENZYL 4 (4 METHOXYPHENYL) 2 (3,4 METHYLENEDIOXYPHENYL) 4 OXO 2 BUTENOIC ACID; CYCLO(DEXTRO TRYPTOPHYL DEXTRO ASPARTYLPROLYL DEXTRO VALYLLEUCYL); ENDOTHELIN RECEPTOR ANTAGONIST; N (2,6 DIMETHYLPIPERIDINOCARBONYL) 4 METHYLLEUCYL DEXTRO (1 METHOXYCARBONYLTRYPTOPHANYL) DEXTRO NORLEUCINE; N ACETYL 10,11 DIHYDRO 5H DIBENZO[A,D]CYCLOHEPTEN 5 YLGLYCYLLEUCYLASPARTYLISOLEUCYLISOLEUCYLTRYPTOPHAN; RECEPTOR SUBTYPE;

ACTION POTENTIAL; ANIMAL TISSUE; ARTICLE; CALCIUM CURRENT; CONTROLLED STUDY; DRUG MECHANISM; DRUG SELECTIVITY; ELECTROPHYSIOLOGY; HEART MUSCLE CELL; NONHUMAN; POTASSIUM CURRENT; PRIORITY JOURNAL; RABBIT; RECEPTOR AFFINITY; RECEPTOR BLOCKING;

ACTION POTENTIALS; ANIMALS; CALCIUM CHANNELS; CELL SEPARATION; DIOXOLES; HEART VENTRICLES; MALE; OLIGOPEPTIDES; PATCH-CLAMP TECHNIQUES; PEPTIDES, CYCLIC; RABBITS; RECEPTORS, ENDOTHELIN; STIMULATION, CHEMICAL;

EID: 0032520671     PISSN: 00062952     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0006-2952(97)00581-9     Document Type: Article

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