Potential intermediates for incorporation of polyhydroxylated prolines into combinatorial libraries

Tetrahedron Letters

Volumn 39, Issue 33, 1998, Pages 6091-6094

  Long, Daniel D ^a   Frederiksen, Signe M ^a   Marquess, Daniel G ^b   Lane, Alexandra L ^a   Watkin, David J ^a   Winkler, David A ^c   Fleet, George W J ^a  

^a UNIVERSITY OF OXFORD   (United Kingdom)

^b GLAXOSMITHKLINE   (United Kingdom)

^c CSIRO   (Australia)

Author keywords

[No Author keywords available]

Indexed keywords

PROLINE DERIVATIVE;

ARTICLE; BACTERIAL CELL WALL; CRYSTAL STRUCTURE; DRUG STRUCTURE; DRUG SYNTHESIS; PROTEIN SECONDARY STRUCTURE;

BACTERIA (MICROORGANISMS);

EID: 0032514434     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(98)01256-8     Document Type: Article

References (15)

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6. 4 Details of the crystal structure of 1 will be reported in a full paper.
7. 3), 62.1 (t, C-6), 59.1, 63.5, 75.7, 82.1 (4 x d, C-2, C-3, C-4, C-5), 173.7 (s, C=O).
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10. 3), 176.4 (s, C=O).
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15. 12 All isolable new compounds have satisfactory CHN analytical or HRMS data. This work has been supported by Glaxo Wellcome and EPSRC.