Shared determinants of receptor binding for subtype selective, and dual endothelin-angiotensin antagonists on the AT1 angiotensin II receptor

FEBS Letters

Volumn 423, Issue 1, 1998, Pages 15-18

  Dascal, David ^a   Nirula, Vaneet ^a   Lawus, Kimberly ^a   Yoo, Sung Eun ^b   Walsh, Thomas F ^c   Sandberg, Kathryn ^a  

^a GEORGETOWN UNIVERSITY MEDICAL CENTER   (United States)

^b Korea Research Institute of Chemical Technology   (South Korea)

^c MERCK RESEARCH LABORATORIES   (United States)

Author keywords

Angiotensin; AT1 receptor; Biphenylimidazole; Dual receptor antagonist; Endothelin; Non peptide

Indexed keywords

AMINO ACID; ANGIOTENSIN ANTAGONIST; ANGIOTENSIN RECEPTOR; ENDOTHELIN RECEPTOR ANTAGONIST; L 746072; LIGAND; RECEPTOR SUBTYPE; UNCLASSIFIED DRUG;

AMINO ACID SUBSTITUTION; AMPHIBIA; ANIMAL CELL; ARTICLE; CELL STRAIN COS1; MAMMAL; NONHUMAN; PRIORITY JOURNAL; RECEPTOR BINDING;

AMINO ACID SEQUENCE; ANGIOTENSIN II; ANIMALS; BINDING SITES; COS CELLS; IMIDAZOLES; LIGANDS; MOLECULAR SEQUENCE DATA; MOLECULAR STRUCTURE; MUTAGENESIS, SITE-DIRECTED; PYRIDINES; RATS; RECEPTOR, ANGIOTENSIN, TYPE 1; RECEPTOR, ANGIOTENSIN, TYPE 2; RECEPTORS, ANGIOTENSIN; RECEPTORS, ENDOTHELIN; STRUCTURE-ACTIVITY RELATIONSHIP; TETRAZOLES; XENOPUS LAEVIS;

AMPHIBIA; ANIMALIA; MAMMALIA;

EID: 0032512713     PISSN: 00145793     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-5793(98)00040-4     Document Type: Article

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