Permeability of benzoic acid derivatives in excised guinea pig dorsal skin and effects of L-menthol

International Journal of Pharmaceutics

Volumn 161, Issue 1, 1998, Pages 115-122

  Kitagawa, Shuji ^a   Hosokai, Akio ^a   Kaseda, Yoshiyuki ^a   Yamamoto, Nobuya ^a   Kaneko, Yoh ^a   Matsuoka, Emiko ^a  

^a NIIGATA UNIVERSITY OF PHARMACY AND APPLIED LIFE SCIENCES   (Japan)

Author keywords

Benzoic acid derivatives; ESR; Partition coefficient; Penetration enhancer; Skin penetration

Indexed keywords

ALCOHOL; BENZOIC ACID DERIVATIVE; MENTHOL;

ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; ELECTRON SPIN RESONANCE; GUINEA PIG; LIPOPHILICITY; MALE; NONHUMAN; PARTITION COEFFICIENT; PRIORITY JOURNAL; SKIN PENETRATION; SKIN PERMEABILITY; SPIN LABELING; STRATUM CORNEUM;

EID: 0032498521     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0378-5173(97)00336-0     Document Type: Article

References (23)

1. Barratt M.D. Quantitative structure-activity relationships for skin permeability. Toxic. in Vitro. 9:1995;27-37.
2. Ghanem A.H., Mahmoud H., Higuchi W.I.et al. The effects of ethanol on the transport of β-estradiol and other permeants in hairless mouse skin. II. A new quantitative approach. J. Controlled Release. 6:1987;75-83.
3. Hashida, M., Yamashita, F., 1995. Terpenes as penetration enhancers. In: Smith, E.W., Maibach, H.I. (Eds.), Percutaneous Penetration Enhancers, CRC Press, Boca Raton, FL, pp. 309-321.
4. Hatanaka T., Shimoyama M., Sugibayashi K., Morimoto Y. Concentration- and time-dependent percutaneous absorption enhancing effect of ethanol. Yakuzaigaku. 52:1992;215-223.
5. Itoh T., Xia J., Magavi R., Nishihata T., Rytting J.H. Use of shed snake skin as a model membrane for in vitro percutaneous penetration studies: comparison with human skin. Pharm. Res. 7:1990;1042-1047.
6. Itoh T., Magavi R., Casady R.L., Nishihata T., Rytting J.H. A method to predict the percutaneous permeability of various compounds: shed snake skin as a model membrane. Pharm. Res. 7:1990;1302-1306.
7. Kitagawa S., Kametani F., Tsuchiya K., Sakurai H. ESR analysis with long-chain alkyl spin labels in bovine blood platelets. Relationship between the increase in membrane fluidity by alcohols and phenolic compounds and their inhibitory effects on aggregation. Biochim. Biophys. Acta. 1027:1990;123-129.
8. Kitagawa S., Yokochi N., Murooka N. pH-dependence of phase transition of the lipid bilayer of liposomes of stratum corneum lipids. Int. J. Pharm. 126:1995;49-56.
9. Kitagawa S., Li H., Sato S. Skin permeation of parabens in excised guinea pig dorsal skin, its modification by penetration enhancers and their relationship with n-octanol/water partition coefficients. Chem. Pharm. Bull. 45:1997;1354-1357.
10. Koyama Y., Bando H., Yamashita F., Takakura Y., Sezaki H., Hashida M. Comparative analysis of percutaneous absorption enhancement by D-limonene and oleic acid based on a skin diffusion model. Pharm. Res. 11:1994;377-383.
11. Leo A., Hansch C., Elkins D. Partition coefficients and their uses. Chem. Rev. 71:1971;525-616.
12. Obata Y., Takayama K., Machida Y., Nagai T. Combined effect of cyclic monoterpenes and ethanol on percutaneous absorption of diclofenac sodium. Drug Des. Discov. 8:1991;137-144.
13. Obata Y., Takayama K., Maitani Y., Machida Y., Nagai T. Effect of ethanol on skin permeation of nonionized and ionized diclofenac. Int. J. Pharm. 89:1993;191-198.
14. Potts R.O., Golden G.M., Francoeur M.L., Mak V.H.W., Guy R.H. Mechanism and enhancement of solute transport across the stratum corneum. J. Controlled Release. 15:1991;249-260.
15. Potts R.O., Guy R.H. Predicting skin permeability. Pharm. Res. 9:1992;663-669.
16. Potts R.O., Guy R.H. Structure-permeability relationships in percutaneous penetration. J. Pharm. Sci. 81:1992;603-604.
17. Quan D., Maibach H.I. An electron spin resonance study: I. Effect of azone on 5-doxyl stearic acid-labeled human stratum corneum. Int. J. Pharm. 104:1994;61-72.
18. Quan, D., Maibach, H.I., 1995. Electron spin resonance. In: Smith, E.W., Maibach, H.I. (Eds.), Percutaneous Penetration Enhancers, CRC Press, Boca Raton, FL, pp. 427-439.
19. Sotomatsu T., Shigemura M., Murata Y., Fujita T. Octanol/water partition coefficient of ortho-substituted aromatic solutes. J. Pharm. Sci. 82:1993;776-781.
20. Sugibayashi K., Kobayashi D., Nakagaki E.et al. Differences in enhancing effect of L-menthol, ethanol and their combination between hairless rat and human skin. Int. J. Pharm. 113:1995;189-197.
21. Tayar N.E., Tsai R.-S., Testa B., Carrupt P.-A., Hansch C., Leo A. Percutaneous penetration of drugs: a quantitative structure-permeability relationship study. J. Pharm. Sci. 80:1991;744-749.
22. Walker R.B., Smith E.W. The role of percutaneous penetration enhancers. Adv. Drug Deliv. Rev. 18:1996;295-301.
23. Ward A.I.I., Tallon R. Penetration enhancer incorporation in bilayers. Drug Dev. Ind. Pharm. 9:1988;1155-1166.