-
1
-
-
0023889603
-
Chimeric alpha 2-, beta 2-adrenergic receptors: delineation of domains involved in effector coupling and ligand binding specificity
-
Kobilka B., Kobilka T., Daniel K., Regan J., Caron M., Lefkowitz R. Chimeric alpha 2-, beta 2-adrenergic receptors: delineation of domains involved in effector coupling and ligand binding specificity. Science 1988; 240: 1310 – 1316
-
(1988)
Science
, vol.240
, pp. 1310-1316
-
-
Kobilka, B.1
Kobilka, T.2
Daniel, K.3
Regan, J.4
Caron, M.5
Lefkowitz, R.6
-
2
-
-
0024519931
-
Structural basis of β-adrenergic receptor function
-
Strader C., Sigal I., Dixon R. Structural basis of β-adrenergic receptor function. FASEB J. 1989; 7: 1825 – 1832
-
(1989)
FASEB J.
, vol.7
, pp. 1825-1832
-
-
Strader, C.1
Sigal, I.2
Dixon, R.3
-
3
-
-
0027297275
-
Constitutive activity of receptors coupled to guanine nucleotide regulatory proteins, Trends Pharmacol
-
Lefkowitz R. J., Coteccia S., Samama P., Costa T. Constitutive activity of receptors coupled to guanine nucleotide regulatory proteins, Trends Pharmacol. Sci. 1993; 14: 303 – 307
-
(1993)
Sci.
, vol.14
, pp. 303-307
-
-
Lefkowitz, R.J.1
Coteccia, S.2
Samama, P.3
Costa, T.4
-
5
-
-
0026015293
-
Primary structure and functional characterization of a human 5-HT1D-type serotonin receptor
-
Hamblin M. W., Metcalf M. A. Primary structure and functional characterization of a human 5-HT1D-type serotonin receptor. Mol. Pharmacol. 1991; 40: 143 – 148
-
(1991)
Mol. Pharmacol.
, vol.40
, pp. 143-148
-
-
Hamblin, M.W.1
Metcalf, M.A.2
-
6
-
-
0027950817
-
The mouse 5-hydroxytryptamine1Breceptor is localized predominantly on axon terminals
-
Boschert U., Amara D. A., Segu L., Hen R. The mouse 5-hydroxytryptamine1Breceptor is localized predominantly on axon terminals. Neuroscience 1994; 58: 167 – 182
-
(1994)
Neuroscience
, vol.58
, pp. 167-182
-
-
Boschert, U.1
Amara, D.A.2
Segu, L.3
Hen, R.4
-
7
-
-
0026651814
-
A human serotonin1Dreceptor variant (5HT1Dβ) encoded by an intronless gene on chromosome 6
-
Demchyshyn L., Sunahara R. K., Miller K., Teitler M., Hoffman B. J., Kennedy J. L., Seeman P., Van Tol H. H.M., Niznik H. B. A human serotonin1Dreceptor variant (5HT1Dβ) encoded by an intronless gene on chromosome 6. Proc. Natl Acad. Sci. U.S.A. 1992; 89: 5522 – 5526
-
(1992)
Proc. Natl Acad. Sci. U.S.A.
, vol.89
, pp. 5522-5526
-
-
Demchyshyn, L.1
Sunahara, R.K.2
Miller, K.3
Teitler, M.4
Hoffman, B.J.5
Kennedy, J.L.6
Seeman, P.7
Van Tol, H.H.M.8
Niznik, H.B.9
-
8
-
-
0027278101
-
Binding-site modeling of the muscarinic m1receptor – a combination of homology-based and indirect approaches
-
Nordvall G., Hacksell U. Binding-site modeling of the muscarinic m1receptor – a combination of homology-based and indirect approaches. J. Med. Chem. 1993; 36: 967 – 976
-
(1993)
J. Med. Chem.
, vol.36
, pp. 967-976
-
-
Nordvall, G.1
Hacksell, U.2
-
9
-
-
0025292355
-
Model for the structure of bacteriorhodopsin based on high-resolution electron cryo-microscopy
-
Henderson R., Baldwin J. M., Ceska T. A., Zemlin F., Beckmann E., Downing K. H. Model for the structure of bacteriorhodopsin based on high-resolution electron cryo-microscopy. J. Mol. Biol 1990; 213: 899 – 929
-
(1990)
J. Mol. Biol
, vol.213
, pp. 899-929
-
-
Henderson, R.1
Baldwin, J.M.2
Ceska, T.A.3
Zemlin, F.4
Beckmann, E.5
Downing, K.H.6
-
10
-
-
0028339899
-
Functional mapping of the ligand binding sites of G-protein coupled receptors
-
Fong T. M., Strader C. D. Functional mapping of the ligand binding sites of G-protein coupled receptors. Med. Res. Rev. 1994; 14: 387 – 399
-
(1994)
Med. Res. Rev.
, vol.14
, pp. 387-399
-
-
Fong, T.M.1
Strader, C.D.2
-
11
-
-
0026601458
-
Site-directed mutagenesis of virtually any plasmid by eliminating a unique site
-
Deng W. P., Nickoloff J. A. Site-directed mutagenesis of virtually any plasmid by eliminating a unique site. Anal. Biochem. 1992; 200: 81 – 88
-
(1992)
Anal. Biochem.
, vol.200
, pp. 81-88
-
-
Deng, W.P.1
Nickoloff, J.A.2
-
12
-
-
0023447252
-
Lipofection: a highly efficient, lipidmediated DNA-transfection procedure
-
Felgner P., Gadek T., Holm M., Roman R., Chan H., Wenz M., Northrop J., Ringold G., Danielsen M. Lipofection: a highly efficient, lipidmediated DNA-transfection procedure. Proc. Natl Acad. Sci. U.S.A. 1987; 84: 7413 – 7417
-
(1987)
Proc. Natl Acad. Sci. U.S.A.
, vol.84
, pp. 7413-7417
-
-
Felgner, P.1
Gadek, T.2
Holm, M.3
Roman, R.4
Chan, H.5
Wenz, M.6
Northrop, J.7
Ringold, G.8
Danielsen, M.9
-
13
-
-
0018178434
-
A modification of the Lowry procedure to simplify protein determination in membrane and lipoprotein samples
-
Markwell M. A.K., Haas S. M., Bieber L. L., Tolbert N. E. A modification of the Lowry procedure to simplify protein determination in membrane and lipoprotein samples. Anal. Biochem. 1978; 87: 206 – 210
-
(1978)
Anal. Biochem.
, vol.87
, pp. 206-210
-
-
Markwell, M.A.K.1
Haas, S.M.2
Bieber, L.L.3
Tolbert, N.E.4
-
14
-
-
0028180615
-
Structural studies on dopamine D2 receptors – mutation of a histidine residue specifically affects the binding of a subgroup of substituted benzamide drugs
-
Woodward R., Daniell S. J., Strange P. G., Naylor L. H. Structural studies on dopamine D2 receptors – mutation of a histidine residue specifically affects the binding of a subgroup of substituted benzamide drugs. J. Neurochem 1994; 62: 1664 – 1669
-
(1994)
J. Neurochem
, vol.62
, pp. 1664-1669
-
-
Woodward, R.1
Daniell, S.J.2
Strange, P.G.3
Naylor, L.H.4
-
15
-
-
0025881062
-
Three-dimensional models of cationic neurotransmitter G-protein coupled receptors
-
Hibert M. F., Trumpp K. S., Bruinvels A., Hoflack J. Three-dimensional models of cationic neurotransmitter G-protein coupled receptors. Mol. Pharmacol. 1991; 40: 8 – 15
-
(1991)
Mol. Pharmacol.
, vol.40
, pp. 8-15
-
-
Hibert, M.F.1
Trumpp, K.S.2
Bruinvels, A.3
Hoflack, J.4
-
16
-
-
0026488456
-
The role of conserved aspartate and serine residues in ligand binding and in function of the 5-HT1Areceptor: a site-directed mutation study
-
Ho B. Y., Karschin A., Branchek T., Davidson N., Lester H. A. The role of conserved aspartate and serine residues in ligand binding and in function of the 5-HT1Areceptor: a site-directed mutation study. FEBS Lett. 1992; 312: 259 – 262
-
(1992)
FEBS Lett.
, vol.312
, pp. 259-262
-
-
Ho, B.Y.1
Karschin, A.2
Branchek, T.3
Davidson, N.4
Lester, H.A.5
-
17
-
-
0024344941
-
Identification of two serine residues involved in agonist activation of the β-adrenergic receptor
-
Strader C., Candelore M., Hill W., Sigal I., Dixon R. Identification of two serine residues involved in agonist activation of the β-adrenergic receptor. J. Biol. Chem 1989; 264: 13572 – 13578
-
(1989)
J. Biol. Chem
, vol.264
, pp. 13572-13578
-
-
Strader, C.1
Candelore, M.2
Hill, W.3
Sigal, I.4
Dixon, R.5
-
18
-
-
0026630139
-
Serine mutations in transmembrane V of the dopamine D1receptor affect ligand interactions and receptor activation
-
Pollock N. J., Manelli A. M., Hutchins C. W., Steffey M. E., Mackenzie R. G., Frail D. E. Serine mutations in transmembrane V of the dopamine D1receptor affect ligand interactions and receptor activation. J. Biol. Chem. 1992; 267: 17780 – 17786
-
(1992)
J. Biol. Chem.
, vol.267
, pp. 17780-17786
-
-
Pollock, N.J.1
Manelli, A.M.2
Hutchins, C.W.3
Steffey, M.E.4
Mackenzie, R.G.5
Frail, D.E.6
-
19
-
-
0026729248
-
Contributions of conserved serine residues to the interactions of ligands with dopamine D2receptors
-
Cox B. A., Henningsen R. A., Spanoyannis A., Neve R. L., Neve K. A. Contributions of conserved serine residues to the interactions of ligands with dopamine D2receptors. J. Neurochem. 1992; 59: 627 – 635
-
(1992)
J. Neurochem.
, vol.59
, pp. 627-635
-
-
Cox, B.A.1
Henningsen, R.A.2
Spanoyannis, A.3
Neve, R.L.4
Neve, K.A.5
-
20
-
-
0026940770
-
Site-directed mutagenesis of the human dopamine D2receptor
-
Mansour A., Meng F., Meador-Woodruff J. H., Taylor L. P., Civelli O., Akil H. Site-directed mutagenesis of the human dopamine D2receptor. Eur. J. Pharmacol. 1992; 227: 205 – 214
-
(1992)
Eur. J. Pharmacol.
, vol.227
, pp. 205-214
-
-
Mansour, A.1
Meng, F.2
Meador-Woodruff, J.H.3
Taylor, L.P.4
Civelli, O.5
Akil, H.6
-
21
-
-
0027238736
-
A single point mutation (Phe340→Leu340) of a conserved phenylalanine abolishes 4-[125I]iodo-(2,5-dimethoxy)phenylisopropylamine and [3H]mesulergine but not [3H]ketanserin binding to 5-hydroxytryptamine2receptors
-
Choudhary M. S., Craigo S., Roth B. L. A single point mutation (Phe340→Leu340) of a conserved phenylalanine abolishes 4-[125I]iodo-(2,5-dimethoxy)phenylisopropylamine and [3H]mesulergine but not [3H]ketanserin binding to 5-hydroxytryptamine2receptors. Mol. Pharmacol. 1993; 43: 755 – 761
-
(1993)
Mol. Pharmacol.
, vol.43
, pp. 755-761
-
-
Choudhary, M.S.1
Craigo, S.2
Roth, B.L.3
-
22
-
-
0030899598
-
High-affinity binding is not sufficient for agonist efficacy at 5-hydroxytryptamine2Areceptors: evidence in favor of a modified ternary complex model
-
Roth B. L., Choudhary M. S., Khan N., Uluer A. High-affinity binding is not sufficient for agonist efficacy at 5-hydroxytryptamine2Areceptors: evidence in favor of a modified ternary complex model. J. Pharmacol. Exp. Ther. 1997; 280: 576 – 583
-
(1997)
J. Pharmacol. Exp. Ther.
, vol.280
, pp. 576-583
-
-
Roth, B.L.1
Choudhary, M.S.2
Khan, N.3
Uluer, A.4
-
23
-
-
0028971630
-
Hydrophobic residues of the D2dopamine receptor are important for binding and signal transduction
-
Cho W., Taylor L. P., Mansour A., Akil H. Hydrophobic residues of the D2dopamine receptor are important for binding and signal transduction. J. Neurochem. 1995; 65: 2105 – 2115
-
(1995)
J. Neurochem.
, vol.65
, pp. 2105-2115
-
-
Cho, W.1
Taylor, L.P.2
Mansour, A.3
Akil, H.4
-
24
-
-
0024150228
-
Structure-function analysis of the β-adrenergic receptor, Cold Spring Harbor Symp
-
Dixon R. A.F., Sigal I. S., Strader C. D. Structure-function analysis of the β-adrenergic receptor, Cold Spring Harbor Symp. Quant. Biol. 1988; 53: 487 – 497
-
(1988)
Quant. Biol.
, vol.53
, pp. 487-497
-
-
Dixon, R.A.F.1
Sigal, I.S.2
Strader, C.D.3
-
25
-
-
0027513982
-
A mutational-induced activated state of the β2-adrenergic receptor
-
Samama P., Coteccia S., Costa T., Lefkowitz R. J. A mutational-induced activated state of the β2-adrenergic receptor. J. Biol. Chem. 1993; 268: 4625 – 4636
-
(1993)
J. Biol. Chem.
, vol.268
, pp. 4625-4636
-
-
Samama, P.1
Coteccia, S.2
Costa, T.3
Lefkowitz, R.J.4
-
26
-
-
0027959963
-
High agonist-independent activity is a distinguishing feature of the dopamine D1Breceptor subtype
-
Tiberi M., Caron M. G. High agonist-independent activity is a distinguishing feature of the dopamine D1Breceptor subtype. J. Biol. Chem. 1994; 269: 27925 – 27931
-
(1994)
J. Biol. Chem.
, vol.269
, pp. 27925-27931
-
-
Tiberi, M.1
Caron, M.G.2
-
27
-
-
0026592357
-
Constitutive activation of the α1B-adrenergic receptor by all amino acid substitutions at a single site
-
Kjelsberg M. A., Cotecchia S., Ostrowski J., Caron M. G., Lefkowitz R. J. Constitutive activation of the α1B-adrenergic receptor by all amino acid substitutions at a single site. J. Biol. Chem. 1992; 267: 1430 – 1433
-
(1992)
J. Biol. Chem.
, vol.267
, pp. 1430-1433
-
-
Kjelsberg, M.A.1
Cotecchia, S.2
Ostrowski, J.3
Caron, M.G.4
Lefkowitz, R.J.5
-
28
-
-
0028987979
-
Pharmacological characterisation of [35S]-GTPΓS binding to chinese hamster ovary cell membranes stably expressing cloned human 5-HT1Dreceptor subtypes
-
Thomas D. R., Faruq S. A., Balcarek J. M., Brown A. M. Pharmacological characterisation of [35S]-GTPΓS binding to chinese hamster ovary cell membranes stably expressing cloned human 5-HT1Dreceptor subtypes. J. Receptor Signal Transduct. Res. 1995; 15: 199 – 211
-
(1995)
J. Receptor Signal Transduct. Res.
, vol.15
, pp. 199-211
-
-
Thomas, D.R.1
Faruq, S.A.2
Balcarek, J.M.3
Brown, A.M.4
|