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Volumn 123, Issue 4, 1998, Pages 619-623

Crystal structure of human secretory phospholipase A2-IIA complex with the potent indolizine inhibitor 120-1032

(5) Kitadokoro, Kengo a,b Hagishita, Sanji a Sato, Tomohiro a Ohtani, Mitsuaki a Miki, Kunio b

Author keywords

Indolizine inhibitor; Non steroidal anti inflammatory drug; Phospholipase A2; Structure based drug design; X ray crystallography

Indexed keywords

CALCIUM ION; ENZYME INHIBITOR; INDOLIZINE DERIVATIVE; INDOLIZINE INHIBITOR; LY 311299; NONSTEROID ANTIINFLAMMATORY AGENT; PHOSPHOLIPASE A2; UNCLASSIFIED DRUG;

ARTICLE; COMPLEX FORMATION; CONTROLLED STUDY; CRYSTAL STRUCTURE; DRUG PROTEIN BINDING; DRUG STRUCTURE; ENZYME ACTIVE SITE; ENZYME INHIBITION; ENZYME STRUCTURE; HYDROGEN BOND; HYDROPHOBICITY; RHEUMATOID ARTHRITIS; SEPTIC SHOCK; STEREOCHEMISTRY; SYNOVIAL FLUID;

EID: 0031978292 PISSN: 0021924X EISSN: None Source Type: Journal
DOI: 10.1093/oxfordjournals.jbchem.a021982 Document Type: Article

Times cited : (46)

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* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.