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Volumn 123, Issue 7, 1998, Pages 1317-1324

Characterization of the recombinant human prostanoid DP receptor and identification of L-644,698, a novel selective DP agonist

Author keywords

DP; Prostaglandin D2; Prostaglandin J2; Prostanoid receptor; Recombinant; Selective agonist

Indexed keywords

3 BENZYL 5 (6 CARBOXYHEXYL) 1 (2 CYCLOHEXYL 2 HYDROXYETHYLAMINO)HYDANTOIN; 4 (3 (3 (3 HYDROXYOCTYL) 4 OXO 2 THIAZOLIDINYL)PROPYL)BENZOIC ACID; 4 [3 [3 (3 HYDROXYOCTYL) 4 OXO 2 THIAZOLIDINYL]PROPYL]BENZOIC ACID; 5 (6 CARBOXYHEXYL) 1 (3 CYCLOHEXYL 3 HYDROXYPROPYL)HYDANTOIN; 9BETA CHLORO 15 CYCLOHEXYL 9 DEOXY 16,17,18,19,20 PENTANORPROSTAGLANDIN F2 ALPHA; BENZOIC ACID DERIVATIVE; CYCLIC AMP; DELTA12 PROSTAGLANDIN J2; PROSTAGLANDIN D2; PROSTAGLANDIN J2; PROSTANOID RECEPTOR; RECOMBINANT RECEPTOR; UNCLASSIFIED DRUG;

EID: 0031913845     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0701708     Document Type: Article
Times cited : (63)

References (45)
  • 4
    • 0024361596 scopus 로고
    • Functional and ligand binding studies suggest heterogeneity of platelet prostacyclin receptors
    • ARMSTRONG, R.A., LAWRENCE, R.A., JONES, R.L., WILSON, N.H. & COLLIER, A. (1989). Functional and ligand binding studies suggest heterogeneity of platelet prostacyclin receptors. Br. J. Pharmacol., 97, 657-668.
    • (1989) Br. J. Pharmacol. , vol.97 , pp. 657-668
    • Armstrong, R.A.1    Lawrence, R.A.2    Jones, R.L.3    Wilson, N.H.4    Collier, A.5
  • 8
    • 0029134144 scopus 로고
    • Molecular cloning and characterization of the human prostanoid DP receptor
    • BOIE, Y., SAWYER, N., SLIPETZ, D.M., METTERS, K.M. & ABRAMOVITZ, M. (1995). Molecular cloning and characterization of the human prostanoid DP receptor. J. Biol. Chem., 270, 18910-18916.
    • (1995) J. Biol. Chem. , vol.270 , pp. 18910-18916
    • Boie, Y.1    Sawyer, N.2    Slipetz, D.M.3    Metters, K.M.4    Abramovitz, M.5
  • 9
    • 0006568229 scopus 로고
    • Heterocyclic prostaglandin analogues. Part 3. The relationship of configuration to biological activity for some hydantoin prostaglandin analogues
    • BROCKWELL, M.A., CALDWELL, A.C., WHITTAKER, N. & BEGLEY, M.J. (1981). Heterocyclic prostaglandin analogues. Part 3. The relationship of configuration to biological activity for some hydantoin prostaglandin analogues. J. Chem. Soc. Perkin Trans., 1, 706-711.
    • (1981) J. Chem. Soc. Perkin Trans. , vol.1 , pp. 706-711
    • Brockwell, M.A.1    Caldwell, A.C.2    Whittaker, N.3    Begley, M.J.4
  • 12
    • 0028183018 scopus 로고
    • VIII. International union of pharmacology classification of prostanoid receptors: Properties, distribution, and structure of the receptors and their subtypes
    • COLEMAN, R.A., SMITH, W.L. & NARUMIYA, S. (1994). VIII. International union of pharmacology classification of prostanoid receptors: properties, distribution, and structure of the receptors and their subtypes. Pharmacol. Rev., 46, 205-229.
    • (1994) Pharmacol. Rev. , vol.46 , pp. 205-229
    • Coleman, R.A.1    Smith, W.L.2    Narumiya, S.3
  • 13
    • 0022632646 scopus 로고
    • Prostaglandin E receptor subtypes in smooth muscle: Agonist activities of stable prostacyclin analogies
    • DONG, Y.J., JONES, R.L. & WILSON, N.H. (1986). Prostaglandin E receptor subtypes in smooth muscle: agonist activities of stable prostacyclin analogies. Br. J. Pharmacol., 87, 97-107.
    • (1986) Br. J. Pharmacol. , vol.87 , pp. 97-107
    • Dong, Y.J.1    Jones, R.L.2    Wilson, N.H.3
  • 14
    • 0015386271 scopus 로고
    • Mathematical theory of complex ligand binding systems at equilibrium: Methods of parameter fitting
    • FELDMAN, H.A. (1972). Mathematical theory of complex ligand binding systems at equilibrium: methods of parameter fitting. Anal. Biochem., 48, 317-338.
    • (1972) Anal. Biochem. , vol.48 , pp. 317-338
    • Feldman, H.A.1
  • 16
    • 0029134947 scopus 로고
    • Functional characterization of the prostanoid DP receptor in human myometrium
    • FERNANDES, B. & CRANKSHAW, D. (1995). Functional characterization of the prostanoid DP receptor in human myometrium. Eur. J. Pharmacol., 283, 73-81.
    • (1995) Eur. J. Pharmacol. , vol.283 , pp. 73-81
    • Fernandes, B.1    Crankshaw, D.2
  • 19
    • 0024547972 scopus 로고
    • The classification of prostaglandin DP-receptors in platelets and vasculature using BW A868C, a novel, selective and potent competitive antagonist
    • GILES, H., LEFF, P., BOLOFO, M.L., KELLY, M.G. & ROBERTSON, A.D. (1989). The classification of prostaglandin DP-receptors in platelets and vasculature using BW A868C, a novel, selective and potent competitive antagonist. Br. J. Pharmacol., 96, 291-300.
    • (1989) Br. J. Pharmacol. , vol.96 , pp. 291-300
    • Giles, H.1    Leff, P.2    Bolofo, M.L.3    Kelly, M.G.4    Robertson, A.D.5
  • 20
    • 0023062991 scopus 로고
    • G proteins: Transducers of receptor-generated signals
    • GILMAN, A.G. (1987). G proteins: transducers of receptor-generated signals. Ann. Rev. Biochem., 56, 615-649.
    • (1987) Ann. Rev. Biochem. , vol.56 , pp. 615-649
    • Gilman, A.G.1
  • 21
    • 0019888760 scopus 로고
    • The regulatory component of adenylate cyclase. Purification and properties of the turkey erythrocyte protein
    • HANSKI, E., STERNWEIS, P.C., NORTHUP, J.K., DROMERICK, A.W. & GILMAN, A.G. (1981). The regulatory component of adenylate cyclase. Purification and properties of the turkey erythrocyte protein. J. Biol. Chem., 256, 12911-12919.
    • (1981) J. Biol. Chem. , vol.256 , pp. 12911-12919
    • Hanski, E.1    Sternweis, P.C.2    Northup, J.K.3    Dromerick, A.W.4    Gilman, A.G.5
  • 23
    • 0027974137 scopus 로고
    • Molecular characterization of a mouse prostaglandin D receptor and functional expression of the cloned gene
    • HIRATA, M., KAKIZUKA, A., AIZAWA, M., USHIKUBI, F. & NARUMIYA, S. (1994). Molecular characterization of a mouse prostaglandin D receptor and functional expression of the cloned gene. Proc. Natl. Acad. Sci. U.S.A., 91, 11192-11196.
    • (1994) Proc. Natl. Acad. Sci. U.S.A. , vol.91 , pp. 11192-11196
    • Hirata, M.1    Kakizuka, A.2    Aizawa, M.3    Ushikubi, F.4    Narumiya, S.5
  • 25
    • 0020398514 scopus 로고
    • Studies on the characterization of prostanoid receptors: A proposed classification
    • KENNEDY, I., COLEMAN, R.A., HUMPHREY, P.P.A., LEVY, G.P. & LUMLEY, P. (1982). Studies on the characterization of prostanoid receptors: a proposed classification. Prostaglandins, 24, 667-689.
    • (1982) Prostaglandins , vol.24 , pp. 667-689
    • Kennedy, I.1    Coleman, R.A.2    Humphrey, P.P.A.3    Levy, G.P.4    Lumley, P.5
  • 26
    • 0028820385 scopus 로고
    • Molecular cloning and expression of multiple isoforms of human prostaglandin E receptor EP3 subtype generated by alternative messenger RNA splicing: Multiple second messenger systems and tissue-specific distributions
    • KOTANI, M., TANAKA, I., OGAWA, Y., UNSUI, T., MORI, K., ICHIKAWA, A., NARUMIYA, S., YOSHIMI, T. & NAKAO, K. (1995). Molecular cloning and expression of multiple isoforms of human prostaglandin E receptor EP3 subtype generated by alternative messenger RNA splicing: multiple second messenger systems and tissue-specific distributions. Mol. Pharmacol., 48, 869-879.
    • (1995) Mol. Pharmacol. , vol.48 , pp. 869-879
    • Kotani, M.1    Tanaka, I.2    Ogawa, Y.3    Unsui, T.4    Mori, K.5    Ichikawa, A.6    Narumiya, S.7    Yoshimi, T.8    Nakao, K.9
  • 30
    • 0028860268 scopus 로고
    • Heterotrimeric G-proteins: Organizers of transmembrane signals
    • NEER, E.J. (1995). Heterotrimeric G-proteins: organizers of transmembrane signals. Cell, 80, 249-257.
    • (1995) Cell , vol.80 , pp. 249-257
    • Neer, E.J.1
  • 31
    • 0025924902 scopus 로고
    • 2 and its mimetic ZK 110.841 are potent inhibitors of receptor-mediated activation of human neutrophils
    • 2 and its mimetic ZK 110.841 are potent inhibitors of receptor-mediated activation of human neutrophils. Eicosanoids, 4, 21-28.
    • (1991) Eicosanoids , vol.4 , pp. 21-28
    • Ney, P.1    Schrör, K.2
  • 32
    • 0029610569 scopus 로고
    • Effects of a selective DP receptor agonist (BW245C) and antagonist (BW A868C) on the canine colonic epithelium: An argument for a different DP receptor
    • RANGACHARI, P.K., BETTI, P.A., PRIOR, E.T. & ROBERTS II, L.J. (1995). Effects of a selective DP receptor agonist (BW245C) and antagonist (BW A868C) on the canine colonic epithelium: an argument for a different DP receptor. J. Pharmacol. Exp. Ther., 275, 611-617.
    • (1995) J. Pharmacol. Exp. Ther. , vol.275 , pp. 611-617
    • Rangachari, P.K.1    Betti, P.A.2    Prior, E.T.3    Roberts II, L.J.4
  • 33
    • 0028948767 scopus 로고
    • Alternative splicing produces a divergent cytoplasmic tail in the human endothelial thromboxane A2 receptor
    • RAYCHOWDHURY, M.K., YUKAWA, M., COLLINS, L.J., MCGRAIL, S.H., KENT, K.C. & WARE, J.C. (1995). Alternative splicing produces a divergent cytoplasmic tail in the human endothelial thromboxane A2 receptor. J. Biol. Chem., 270, 7011-7014.
    • (1995) J. Biol. Chem. , vol.270 , pp. 7011-7014
    • Raychowdhury, M.K.1    Yukawa, M.2    Collins, L.J.3    Mcgrail, S.H.4    Kent, K.C.5    Ware, J.C.6
  • 35
    • 0022416536 scopus 로고
    • Regulation of glucagon receptor binding. Lack of effect of Mg and preferential role for GDP
    • ROJAS, F.J. & BIRMBAUMER, L. (1985). Regulation of glucagon receptor binding. Lack of effect of Mg and preferential role for GDP. J. Biol. Chem., 260, 7829-7835.
    • (1985) J. Biol. Chem. , vol.260 , pp. 7829-7835
    • Rojas, F.J.1    Birmbaumer, L.2
  • 38
    • 0026698153 scopus 로고
    • In vitro characterization of prostanoid FP-, DP-, IP- and TP-receptors on the non-pregnant human myometrium
    • SENIOR, J., SANGHA, R., BAXTER, G.S., MARSHALL, K., & CLAYTON, J.K. (1992). In vitro characterization of prostanoid FP-, DP-, IP-and TP-receptors on the non-pregnant human myometrium. Br. J. Pharmacol., 107, 215-221.
    • (1992) Br. J. Pharmacol. , vol.107 , pp. 215-221
    • Senior, J.1    Sangha, R.2    Baxter, G.S.3    Marshall, K.4    Clayton, J.K.5
  • 40
    • 0019888557 scopus 로고
    • The regulatory component of adenylate cyclase. Purification and properties
    • STERNWEIS, P.C., NORTHUP, J.K., SMIGEL, M.D. & OILMAN, A.G. (1981). The regulatory component of adenylate cyclase. Purification and properties. J. Biol. Chem., 256, 11517-11526.
    • (1981) J. Biol. Chem. , vol.256 , pp. 11517-11526
    • Sternweis, P.C.1    Northup, J.K.2    Smigel, M.D.3    Oilman, A.G.4
  • 44
    • 0020959862 scopus 로고
    • Platelet and cardiovascular activity of the hydantoin BW245C, a potent prostaglandin analogue
    • WHITTLE, B.J.R., MONCADA, S., MULLANE, K. & VANE, J.R. (1983). Platelet and cardiovascular activity of the hydantoin BW245C, a potent prostaglandin analogue. Prostaglandins, 25, 205-223.
    • (1983) Prostaglandins , vol.25 , pp. 205-223
    • Whittle, B.J.R.1    Moncada, S.2    Mullane, K.3    Vane, J.R.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.