GR196429: A nonindolic agonist at high-affinity melatonin receptors

Journal of Pharmacology and Experimental Therapeutics

Volumn 285, Issue 3, 1998, Pages 1239-1245

  Beresford, Isabel J M ^a   Browning, Christopher ^a   Starkey, Sarah J ^a   Brown, Jason ^a   Foord, Steven M ^a   Coughlan, Josephine ^a   North, Peter C ^a   Dubocovich, Margarita L ^a,b   Hagan, Russell M ^a  

^a GLAXOSMITHKLINE   (United Kingdom)

^b Dept Molec Pharmacol Biol Chem ^*  (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AGOMELATINE; HORMONE RECEPTOR STIMULATING AGENT; LUZINDOLE; MELATONIN; MELATONIN DERIVATIVE; MELATONIN RECEPTOR; N [2 (2,3,7,8 TETRAHYDRO 1H FURO[2,3 G]INDOL 1 YL)ETHYL]ACETAMIDE; N ACETYLSEROTONIN; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; CHO CELL; CIRCADIAN RHYTHM; DRUG RECEPTOR BINDING; GUINEA PIG; LIGAND BINDING; MALE; NONHUMAN; PRIORITY JOURNAL; RECEPTOR AFFINITY; SUPERIOR COLLICULUS; SUPRACHIASMATIC NUCLEUS;

ANIMALS; BINDING SITES; BRAIN; CHO CELLS; CRICETINAE; DOSE-RESPONSE RELATIONSHIP, DRUG; ELECTROPHYSIOLOGY; GUINEA PIGS; HUMANS; INDOLES; MALE; RABBITS; RATS; RECEPTORS, CELL SURFACE; RECEPTORS, CYTOPLASMIC AND NUCLEAR; RECEPTORS, MELATONIN; RETINA;

EID: 0031863947     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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