G-protein activation at 5-HT(1A) receptors by the 5-ht(1F) ligand LY334370 in guinea-pig brain sections and recombinant cell lines

British Journal of Pharmacology

Volumn 124, Issue 2, 1998, Pages 283-290

  Dupuis, Delphine S ^a   Colpaert, Francis C ^a   Pauwels, Petrus J ^a  

^a INSTITUT DE RECHERCHE PIERRE FABRE   (France)

Author keywords

5 ht(1F) and 5 HT(1A) receptor; 35S GTP S binding and autoradiography; G protein activation; Guinea pig brain; Recombinant h 5 HT(1A) cell lines

Indexed keywords

5 (4 FLUOROBENZAMIDO) 3 (1 METHYL 4 PIPERIDINYL) 1H INDOLE FUMARATE; 5 CARBAMOYLTRYPTAMINE; GUANINE NUCLEOTIDE BINDING PROTEIN; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); IODINE 125; LIGAND; LISURIDE; N [2 [4 (2 METHOXYPHENYL) 1 PIPERAZINYL]ETHYL] N (2 PYRIDYL)CYCLOHEXANECARBOXAMIDE; SEROTONIN 1A RECEPTOR; SEROTONIN 1F RECEPTOR; SULFUR 35; SUMATRIPTAN; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; AUTORADIOGRAPHY; BINDING AFFINITY; BRAIN REGION; CAUDATE NUCLEUS; CELL LINE; CINGULATE GYRUS; CLAUSTRUM; CONTROLLED STUDY; DORSAL RAPHE NUCLEUS; ENTORHINAL CORTEX; GUINEA PIG; HIPPOCAMPUS; MALE; NONHUMAN; PRIORITY JOURNAL; PUTAMEN; SEPTUM PELLUCIDUM; THALAMUS;

AMINOPYRIDINES; ANIMALS; AUTORADIOGRAPHY; BENZAMIDES; BINDING SITES; BINDING, COMPETITIVE; BRAIN; GTP-BINDING PROTEINS; GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE); GUINEA PIGS; HELA CELLS; HIPPOCAMPUS; HUMANS; INDOLES; MALE; PIPERAZINES; PYRIDINES; RAPHE NUCLEI; RECEPTORS, SEROTONIN; RECEPTORS, SEROTONIN, 5-HT1; SEROTONIN; SEROTONIN AGONISTS; SEROTONIN ANTAGONISTS; SUMATRIPTAN;

EID: 0031835564     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0701832     Document Type: Article

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