메뉴 건너뛰기




Volumn 30, Issue 1, 1998, Pages 49-55

RTI-113 administration reduces cocaine self-administration at high occupancy of dopamine transporter

Author keywords

Agonist; Dopamine transporter inhibitor; Drug abuse; Psychostimulant

Indexed keywords

3BETA [4 (4 CHLOROPHENYL)TROPAN] 2BETA CARBOXYLIC ACID PHENYL ESTER; COCAINE; DOPAMINE TRANSPORTER; UNCLASSIFIED DRUG;

EID: 0031828427     PISSN: 08874476     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1098-2396(199809)30:1<49::AID-SYN6>3.0.CO;2-K     Document Type: Article
Times cited : (31)

References (26)
  • 1
    • 0001894665 scopus 로고
    • Subjects and Instrumentation
    • Iverson, S. and Lattal, A., eds. Elsevier, New York
    • Ator, N. A. (1991) Subjects and Instrumentation. In: Experimental Analysis of Behavior. Iverson, S. and Lattal, A., eds. Elsevier, New York, pp. 1-62.
    • (1991) Experimental Analysis of Behavior , pp. 1-62
    • Ator, N.A.1
  • 2
    • 0028903389 scopus 로고
    • Novel 2-substituted cocaine analogs: Uptake and ligand binding studies at dopamine, serotonin and norepinephrine transport sites in the rat brain
    • Bennett, B.A., Wichems, C.H., Hollingsworth, C.K., Davies, H.M.L., Thornley, C., Sexton, T., and Childers, S.R. (1995) Novel 2-substituted cocaine analogs: Uptake and ligand binding studies at dopamine, serotonin and norepinephrine transport sites in the rat brain. J.P.E.T., 272:1176-1186.
    • (1995) J.P.E.T. , vol.272 , pp. 1176-1186
    • Bennett, B.A.1    Wichems, C.H.2    Hollingsworth, C.K.3    Davies, H.M.L.4    Thornley, C.5    Sexton, T.6    Childers, S.R.7
  • 3
    • 0029063953 scopus 로고
    • Cocaine and 3beta-(4'Substituted phenyl )-2beta-carboxylic acid ester and amide analogs. New high affinity and selective compounds for the dopamine transporter
    • Carroll, F.I., Kotian, P., Dehghani, A., Gray, J. L., Kuzemko, M. A., Parham, K. A., Abraham, P., Lewin,A. H., Boja, J. W., and Kuhar, M. J. (1995) Cocaine and 3beta-(4'Substituted phenyl )-2beta-carboxylic acid ester and amide analogs. New high affinity and selective compounds for the dopamine transporter. J. Med. Chem., 38:379-388.
    • (1995) J. Med. Chem. , vol.38 , pp. 379-388
    • Carroll, F.I.1    Kotian, P.2    Dehghani, A.3    Gray, J.L.4    Kuzemko, M.A.5    Parham, K.A.6    Abraham, P.7    Lewin, A.H.8    Boja, J.W.9    Kuhar, M.J.10
  • 4
    • 0002379639 scopus 로고    scopus 로고
    • Dopamine transporter uptake blockers: Structure activity relationships
    • M A Reith, ed. Humana Press Inc., Totowa, NJ
    • Carroll, F.I., Lewin, A.., and Kuhar, M.J. (1997) Dopamine transporter uptake blockers: Structure activity relationships. In: Neurotrnamitter Transporters: Structure, Function and Regulation. M A Reith, ed. Humana Press Inc., Totowa, NJ, pp 263-295.
    • (1997) Neurotrnamitter Transporters: Structure, Function and Regulation , pp. 263-295
    • Carroll, F.I.1    Lewin, A.2    Kuhar, M.J.3
  • 5
    • 0026720452 scopus 로고
    • Behavioral effects of novel cocaine analogs: A comparison with in vivo receptor binding potency
    • Cline, E.J., Scheffel, U., Boja, J.W., Carroll, F.I., Katz, J.L., and Kuhar, M.J. (1992) Behavioral effects of novel cocaine analogs: A comparison with in vivo receptor binding potency. J.P.E.T., 260:1174-1179.
    • (1992) J.P.E.T. , vol.260 , pp. 1174-1179
    • Cline, E.J.1    Scheffel, U.2    Boja, J.W.3    Carroll, F.I.4    Katz, J.L.5    Kuhar, M.J.6
  • 6
    • 0027446171 scopus 로고
    • Novel 2-substituted cocaine analogs: Binding properties at dopamine transport sites in rat striatum
    • Davies, H.M.L., Saikali, E., Sexton, T., and Childers, S.R.(1993) Novel 2-substituted cocaine analogs: binding properties at dopamine transport sites in rat striatum. Eur. J. Pharmacol. Mol. Pharmacol. Sect., 244:93-97.
    • (1993) Eur. J. Pharmacol. Mol. Pharmacol. Sect. , vol.244 , pp. 93-97
    • Davies, H.M.L.1    Saikali, E.2    Sexton, T.3    Childers, S.R.4
  • 7
    • 0028054396 scopus 로고
    • Can stimulant binding and dopamine transport be differentiated? Studies with GBR 12783 derivatives
    • Deutch, H.M., and Schweri, M.M. (1994) Can stimulant binding and dopamine transport be differentiated? Studies with GBR 12783 derivatives. Life Sci., 55:PL115-120.
    • (1994) Life Sci. , vol.55
    • Deutch, H.M.1    Schweri, M.M.2
  • 8
    • 0028897010 scopus 로고
    • Effects of ibogaine on responding maintained by food, cocaine and heroin reinforcement in rats
    • Dworkin, S.I., Gleeson, S., Meloni, D., Koves, T.R., and Martin, T.J.(1995) Effects of ibogaine on responding maintained by food, cocaine and heroin reinforcement in rats. Psychopharmacology, 117:257-261.
    • (1995) Psychopharmacology , vol.117 , pp. 257-261
    • Dworkin, S.I.1    Gleeson, S.2    Meloni, D.3    Koves, T.R.4    Martin, T.J.5
  • 9
    • 0030434485 scopus 로고    scopus 로고
    • Recovery of dopamine transporter binding and function following intrastriatal administation of the irreversible inhibitor RTI-76
    • Fleckenstein, A.E., Pogun, S., Carroll, F.I., and Kuhar, M.J. (1996) Recovery of dopamine transporter binding and function following intrastriatal administation of the irreversible inhibitor RTI-76. J.P.E.T., 279:200-206.
    • (1996) J.P.E.T. , vol.279 , pp. 200-206
    • Fleckenstein, A.E.1    Pogun, S.2    Carroll, F.I.3    Kuhar, M.J.4
  • 10
    • 0029120376 scopus 로고
    • Effects of dopamine reuptake inhibitors on food- and cocaine-maintained responding: II. Comparisons with other drugs and repeated administrations
    • Glowa, J.R., Wojinicki, F.H.E., Matecka, D., Rice, K.C., and Rothman, R.B. (1995) Effects of dopamine reuptake inhibitors on food- and cocaine-maintained responding: II. Comparisons with other drugs and repeated administrations. Exp. Clin. Psychopharmacol., 3:232-239.
    • (1995) Exp. Clin. Psychopharmacol. , vol.3 , pp. 232-239
    • Glowa, J.R.1    Wojinicki, F.H.E.2    Matecka, D.3    Rice, K.C.4    Rothman, R.B.5
  • 11
    • 0030473214 scopus 로고    scopus 로고
    • Sustained decrease in cocaine-maintained responding in rhesus monkeys with 1-[2-[bis (4-fluorophenyl-)methoxy]ethyl]-4-(3-hydroxy-3-phenylpropyl) piperaxinyl decanoate, a long-acting ester derivative of GBR 12909
    • Glowa, J.R., Fantegrossi, W.E., Lewis, D.B., Matecka, D., Rice, K.C., and Rothman, R.B. (1996) Sustained decrease in cocaine-maintained responding in rhesus monkeys with 1-[2-[bis (4-fluorophenyl-)methoxy]ethyl]-4-(3-hydroxy-3-phenylpropyl) piperaxinyl decanoate, a long-acting ester derivative of GBR 12909. J. Med. Chem., 39:4628-4691.
    • (1996) J. Med. Chem. , vol.39 , pp. 4628-4691
    • Glowa, J.R.1    Fantegrossi, W.E.2    Lewis, D.B.3    Matecka, D.4    Rice, K.C.5    Rothman, R.B.6
  • 12
    • 0028337480 scopus 로고
    • Synthesis and characterization of radioiodinated N-(3-Iodopropen-l-yl)-2β-carbomethoxy-3β-(4-chlorophenyl)tropanes Potential dopamine reuptake site imaging agents
    • Goodman, M.M., Kung, M.-P., Kabalka, G.W., Kung, H.F., and Switzer, R. (1994) Synthesis and characterization of radioiodinated N-(3-Iodopropen-l-yl)-2β-carbomethoxy-3β-(4-chlorophenyl)tropanes Potential dopamine reuptake site imaging agents. J. Med. Chem., 37:1535-1542.
    • (1994) J. Med. Chem. , vol.37 , pp. 1535-1542
    • Goodman, M.M.1    Kung, M.-P.2    Kabalka, G.W.3    Kung, H.F.4    Switzer, R.5
  • 13
    • 0029049225 scopus 로고
    • Comparison of a novel tropane analog of cocaine, 2β-propanoyl-3β-(4-tolyl) tropane with cocaine HCl in rats: Nucleus accumbens extracellular dopamine concentration and motor activ-ity
    • Hemby, S.E., Co, C., Reboussin, D., Davies HML, Dworkin, S.I., and Smith, J.E. (1995) Comparison of a novel tropane analog of cocaine, 2β-propanoyl-3β-(4-tolyl) tropane with cocaine HCl in rats: nucleus accumbens extracellular dopamine concentration and motor activ-ity. J.P.E.T., 273:656-666.
    • (1995) J.P.E.T. , vol.273 , pp. 656-666
    • Hemby, S.E.1    Co, C.2    Reboussin, D.3    Davies, H.M.L.4    Dworkin, S.I.5    Smith, J.E.6
  • 14
    • 0029824217 scopus 로고    scopus 로고
    • 3α-4'-substituted phenylOtropane-2β-carboxylic acid methyl esters: Novel ligands with high affinity and selectivity at the dopamine transporter
    • Holmquist, C.R., Keverline-Frantz, K.I., Abraham, P., Boja, J.W., Kuhar, M.J., and Carroll, F.I.(1996) 3α-(4'-substituted phenylOtropane-2β-carboxylic acid methyl esters: Novel ligands with high affinity and selectivity at the dopamine transporter. J. Med. Chem., 39:4139-4141.
    • (1996) J. Med. Chem. , vol.39 , pp. 4139-4141
    • Holmquist, C.R.1    Keverline-Frantz, K.I.2    Abraham, P.3    Boja, J.W.4    Kuhar, M.J.5    Carroll, F.I.6
  • 15
    • 0029899173 scopus 로고    scopus 로고
    • Synthesis, ligand binding and quantitative structure-activity relationship study of 3β-(4'-substituted phenyl)-2β (heterocyclic)tropanes: Evidence for an electrostatic interaction at the 2 beta position
    • Kotian, P., Mascarella, S.W., Abraham, P., Lewin, A. H., Boja, J.W., Kuhar, M.J., and Carroll, F.I. (1996) Synthesis, ligand binding and quantitative structure-activity relationship study of 3β-(4'-substituted phenyl)-2β (heterocyclic)tropanes: Evidence for an electrostatic interaction at the 2 beta position. J. Med. Chem., 39:2753-2763.
    • (1996) J. Med. Chem. , vol.39 , pp. 2753-2763
    • Kotian, P.1    Mascarella, S.W.2    Abraham, P.3    Lewin, A.H.4    Boja, J.W.5    Kuhar, M.J.6    Carroll, F.I.7
  • 16
    • 0002259674 scopus 로고
    • The Otto Krayer Award Lecture: Neurotransmitter transporters as drug targets: Recent research with a focus on the dopamine transporter
    • Kuhar, M.J. (1993) The Otto Krayer Award Lecture: Neurotransmitter transporters as drug targets: Recent research with a focus on the dopamine transporter. Pharmacologist 35:28-33.
    • (1993) Pharmacologist , vol.35 , pp. 28-33
    • Kuhar, M.J.1
  • 17
    • 0024464860 scopus 로고
    • Effects of cocaine and related drugs in nonhuman primates I. [3H]cocaine binding sites in caudate-putamen
    • 1989
    • Madras, B.K., Fahey, M.A., Bergman, J., Canfield, D.R., and Spealman, R.D. (1989) Effects of cocaine and related drugs in nonhuman primates I. [3H]cocaine binding sites in caudate-putamen. J.P.E.T., 251:1310-1141, 1989.
    • (1989) J.P.E.T. , vol.251 , pp. 1310-11141
    • Madras, B.K.1    Fahey, M.A.2    Bergman, J.3    Canfield, D.R.4    Spealman, R.D.5
  • 18
    • 0031055081 scopus 로고    scopus 로고
    • Heteroaromatic analogs of 1-[2-(diphenylmethoxy)ethyl]- and 1-[2-[bis (4-fluorophenyl) methoxy]thyl] -4-(3-phenylpropyl) piperazines (GBR 12935 and GBR 12909) as high-affinity dopamine reuptake inhibitors
    • Matecka, D., Lewis, D., Rothman, R.B., Dersch, C.M., Wojnicki, F.H., Glowa, J.R., DeVries, A.C., Pert, A., and Rice, K.C. (1997) Heteroaromatic analogs of 1-[2-(diphenylmethoxy)ethyl]- and 1-[2-[bis (4-fluorophenyl) methoxy]thyl] -4-(3-phenylpropyl) piperazines (GBR 12935 and GBR 12909) as high-affinity dopamine reuptake inhibitors. J. Med. Chem., 40:705-716.
    • (1997) J. Med. Chem. , vol.40 , pp. 705-716
    • Matecka, D.1    Lewis, D.2    Rothman, R.B.3    Dersch, C.M.4    Wojnicki, F.H.5    Glowa, J.R.6    DeVries, A.C.7    Pert, A.8    Rice, K.C.9
  • 19
    • 0027468956 scopus 로고
    • Substituted 3-phenyltropane analogs of cocaine: Synthe-sis, inhibition of binding at cocaine recognition sites, and positron emission tomography imaging
    • Meltzer, P.C., Liang, A.Y., Brownell, A.-L., Elmaleh, D.R., and Madras, B.K. (1993) Substituted 3-phenyltropane analogs of cocaine: synthe-sis, inhibition of binding at cocaine recognition sites, and positron emission tomography imaging. J. Med. Chem., 36:855-862.
    • (1993) J. Med. Chem. , vol.36 , pp. 855-862
    • Meltzer, P.C.1    Liang, A.Y.2    Brownell, A.-L.3    Elmaleh, D.R.4    Madras, B.K.5
  • 20
    • 0030899415 scopus 로고    scopus 로고
    • The reinforcing and discriminative stimulus effects of the novel cocaine analog 2 -propanoyl-3 -94-tolyl-tropane in rhesus monkeys
    • Nader, M.A., Grant, K.A., Davies, H.M.L., Mach, R.H., and Childers, S.R. (1997) The reinforcing and discriminative stimulus effects of the novel cocaine analog 2 -propanoyl-3 -94-tolyl)-tropane in rhesus monkeys. J.P.E.T., 280:541-550.
    • (1997) J.P.E.T. , vol.280 , pp. 541-550
    • Nader, M.A.1    Grant, K.A.2    Davies, H.M.L.3    Mach, R.H.4    Childers, S.R.5
  • 21
    • 0028104102 scopus 로고
    • Novel 3α-(diphenylmethoxy) tropane analogs: Potent dopamine uptake inhibitors without cocaine-like behavioral profiles
    • Newman, A.H., Allen, A.C., Izenwasser, S., and Katz, J.L. (1994) Novel 3α-(diphenylmethoxy) tropane analogs: Potent dopamine uptake inhibitors without cocaine-like behavioral profiles. J. Med. Chem., 37:2258-2261.
    • (1994) J. Med. Chem. , vol.37 , pp. 2258-2261
    • Newman, A.H.1    Allen, A.C.2    Izenwasser, S.3    Katz, J.L.4
  • 22
    • 0023265754 scopus 로고
    • Cocaine receptors on dopamine transporters are related to self-administration of cocaine
    • Ritz, M.C., Lamb, R.J., Goldberg, S.R., and Kuhar, M.J.(1987) Cocaine receptors on dopamine transporters are related to self-administration of cocaine. Science, 237:1219-1223.
    • (1987) Science , vol.237 , pp. 1219-1223
    • Ritz, M.C.1    Lamb, R.J.2    Goldberg, S.R.3    Kuhar, M.J.4
  • 23
    • 0026469291 scopus 로고
    • Cocaine and GBR 12909 produce equivalent motoric responses at different occupancy of the dopamine transporter
    • Rothman, R.B., Grieg, N., Kim, A., DeCosta, B.R., Rice, K.C., Carroll, F., and Pert, A. (1992) Cocaine and GBR 12909 produce equivalent motoric responses at different occupancy of the dopamine transporter. Pharmacol. Biochem. Behav. 43:1135-1142.
    • (1992) Pharmacol. Biochem. Behav. , vol.43 , pp. 1135-1142
    • Rothman, R.B.1    Grieg, N.2    Kim, A.3    DeCosta, B.R.4    Rice, K.C.5    Carroll, F.6    Pert, A.7
  • 25
    • 0027464060 scopus 로고
    • In vivo occupancy of the striatal dopamine uptake complex by various inhibitors does not predict their effects on locomotion
    • Vaugeois, J.-M., Bonnet, J.-J., Duterte-Boucher, D., and Costentin, J. (1993) In vivo occupancy of the striatal dopamine uptake complex by various inhibitors does not predict their effects on locomotion. Eur. J. Pharmacol., 230:195-201.
    • (1993) Eur. J. Pharmacol. , vol.230 , pp. 195-201
    • Vaugeois, J.-M.1    Bonnet, J.-J.2    Duterte-Boucher, D.3    Costentin, J.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.