Synthesis of [methoxy-11C]PD153035, a selective EGF receptor tyrosine kinase inhibitor

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 41, Issue 7, 1998, Pages 623-629

  Johnström, Peter ^a   Fredriksson, Anna ^a   Thorell, Jan Olov ^a   Stone Elander, Sharon ^a  

^a KAROLINSKA UNIVERSITY HOSPITAL   (Sweden)

Author keywords

Carbon 11; EGF receptor; PD153035; PET; Positron emission tomography; Tyrosine kinase inhibitor

Indexed keywords

AMINO ACIDS; CARBON; ENZYME INHIBITION;

CARBON-11; EGF RECEPTOR; METHOXY; METHYL IODIDE; PD153035; POTENT INHIBITOR; RECEPTOR-TYROSINE KINASE; SPECIFIC ACTIVITY; SPECIFIC INHIBITORS; TYROSINE KINASE INHIBITOR;

POSITRON EMISSION TOMOGRAPHY;

4 (3 BROMOANILINO) 6,7 DIMETHOXYQUINAZOLINE; 4 (3 BROMOANILINO) 6,7 DIMETHOXYQUINAZOLINE C 11; CARBON 11; EPIDERMAL GROWTH FACTOR RECEPTOR KINASE; EPIDERMAL GROWTH FACTOR RECEPTOR KINASE INHIBITOR; UNCLASSIFIED DRUG;

ALKYLATION; ARTICLE; DRUG FORMULATION; LIGAND BINDING; POSITRON EMISSION TOMOGRAPHY; PROTON NUCLEAR MAGNETIC RESONANCE; SIGNAL TRANSDUCTION; SYNTHESIS; THIN LAYER CHROMATOGRAPHY;

EOS;

EID: 0031802624     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1099-1344(199807)41:7<623::AID-JLCR120>3.0.CO;2-Q     Document Type: Article

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