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Volumn 124, Issue 3, 1998, Pages 485-492

Pharmacological characterization of the human melatonin Mel(1a), receptor following stable transfection into NIH3T3 cells

Author keywords

35S GTP S binding; Efficacy; G(i) coupled receptors; Human melatonin receptor; Melatonin analogues

Indexed keywords

AMIDE; GUANINE NUCLEOTIDE BINDING PROTEIN; GUANINE NUCLEOTIDE EXCHANGE FACTOR; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); MELATONIN; MELATONIN DERIVATIVE; MELATONIN RECEPTOR; PARTIAL AGONIST; PERTUSSIS TOXIN; SODIUM CHLORIDE; SULFUR 35; TRYPTAMINE DERIVATIVE; UNCOUPLING PROTEIN;

EID: 0031801678     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0701860     Document Type: Article
Times cited : (56)

References (39)
  • 1
    • 0028171745 scopus 로고
    • Evidence for multiple forms of melatonin receptor-G-protein complexes by solubilization and gel electrophoresis
    • BARRETT, P., MACLEAN, A. & MORGAN, P.J. (1994). Evidence for multiple forms of melatonin receptor-G-protein complexes by solubilization and gel electrophoresis. J. Neuroendocrinol., 6, 509-515.
    • (1994) J. Neuroendocrinol. , vol.6 , pp. 509-515
    • Barrett, P.1    Maclean, A.2    Morgan, P.J.3
  • 3
    • 0017184389 scopus 로고
    • A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein dye-binding
    • BRADFORD, M. (1976). A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein dye-binding. Anal. Biochem., 72, 248-254.
    • (1976) Anal. Biochem. , vol.72 , pp. 248-254
    • Bradford, M.1
  • 5
    • 0025238655 scopus 로고
    • Spontaneous association between opioid receptors and GTP-binding regulatory proteins in native membranes: Specific regulation by antagonist and sodium ions
    • COSTA, T., LANG, J., GLESS, C. & HERZ, A. (1990). Spontaneous association between opioid receptors and GTP-binding regulatory proteins in native membranes: specific regulation by antagonist and sodium ions. Mol. Pharmacol., 37, 383-394.
    • (1990) Mol. Pharmacol. , vol.37 , pp. 383-394
    • Costa, T.1    Lang, J.2    Gless, C.3    Herz, A.4
  • 6
    • 0026608113 scopus 로고
    • Drug efficacy at guanine nucleotide-binding regulatory protein-linked receptors: Thermodynamic interpretation of negative antagonism and of receptor activity in the absence of ligand
    • COSTA, T., OGINO, Y., MUNSON, P.J., ONGUN ONARAN, H. & RODBARD, D. (1992). Drug efficacy at guanine nucleotide-binding regulatory protein-linked receptors: thermodynamic interpretation of negative antagonism and of receptor activity in the absence of ligand. Mol. Pharmacol., 41, 549-560.
    • (1992) Mol. Pharmacol. , vol.41 , pp. 549-560
    • Costa, T.1    Ogino, Y.2    Munson, P.J.3    Ongun Onaran, H.4    Rodbard, D.5
  • 7
    • 0018001339 scopus 로고
    • Simultaneous analysis of families of sigmoidal curves: Application to bioassay, radioligand assay, and physiological dose-response curves
    • DE LEAN, A., MUNSON, P.J. & RODBARD, D. (1978). Simultaneous analysis of families of sigmoidal curves: application to bioassay, radioligand assay, and physiological dose-response curves. Am. J. Physiol., 235, E97-E102.
    • (1978) Am. J. Physiol. , vol.235
    • De Lean, A.1    Munson, P.J.2    Rodbard, D.3
  • 8
    • 0028202804 scopus 로고
    • Effect of inducing nocturnal serum melatonin concentrations in daytime on sleep, mood, body temperature, and performance
    • DOLLINS, A.B., ZHDANOVA, I.V., WURTMAN, R.J., LYNCH, H.J. & DENG, M.H. (1994). Effect of inducing nocturnal serum melatonin concentrations in daytime on sleep, mood, body temperature, and performance. Proc. Natl. Acad. Sci. U.S.A., 91, 1824-1828.
    • (1994) Proc. Natl. Acad. Sci. U.S.A. , vol.91 , pp. 1824-1828
    • Dollins, A.B.1    Zhdanova, I.V.2    Wurtman, R.J.3    Lynch, H.J.4    Deng, M.H.5
  • 11
    • 0030218210 scopus 로고    scopus 로고
    • Serotonin and N-acetylserotonin effects on pigment cells of the toad Bufo ictericus: Pharmacological characterization of melatonin receptors
    • FILADELFI, A.M.C. & CASTRUCCI, A.M. (1996). Serotonin and N-acetylserotonin effects on pigment cells of the toad Bufo ictericus: pharmacological characterization of melatonin receptors. Gen. Comp. Endocrinol., 103, 192-199.
    • (1996) Gen. Comp. Endocrinol. , vol.103 , pp. 192-199
    • Filadelfi, A.M.C.1    Castrucci, A.M.2
  • 12
    • 0028970287 scopus 로고
    • Mapping the melatonin receptor. 3. Design and synthesis of melatonin agonists and antagonists derived from 2-phenyltryptamines
    • GARRATT, P.J., JONES, R. & TOCHER, D.A. (1995). Mapping the melatonin receptor. 3. Design and synthesis of melatonin agonists and antagonists derived from 2-phenyltryptamines. J. Med. Chem., 38, 1132-1139.
    • (1995) J. Med. Chem. , vol.38 , pp. 1132-1139
    • Garratt, P.J.1    Jones, R.2    Tocher, D.A.3
  • 13
    • 14444287680 scopus 로고
    • 2 dopamine receptors from high to low affinity for dopamine agonists
    • 2 dopamine receptors from high to low affinity for dopamine agonists. Soc. Neurosci. Abstr., 9, 31.
    • (1983) Soc. Neurosci. Abstr. , vol.9 , pp. 31
    • Grigoriadis, D.1    Seeman, P.2
  • 16
    • 0024787617 scopus 로고
    • Muscarinic acetylcholine receptor-stimulated binding of guanosine 5′-O-(3-thiotriphosphate) to guanine nucleotide-binding proteins in cardiac membranes
    • HILF, G., GIERSHIK, P. & JAKOBS, K.H. (1989). Muscarinic acetylcholine receptor-stimulated binding of guanosine 5′-O-(3-thiotriphosphate) to guanine nucleotide-binding proteins in cardiac membranes. Eur. J. Biochem., 186, 725-731.
    • (1989) Eur. J. Biochem. , vol.186 , pp. 725-731
    • Hilf, G.1    Giershik, P.2    Jakobs, K.H.3
  • 18
    • 0025248152 scopus 로고
    • +, 5′-guanylylimidodiphosphate, amiloride and ethylisopropylamiloride: Evidence for receptor-G protein precoupling
    • +, 5′-guanylylimidodiphosphate, amiloride and ethylisopropylamiloride: evidence for receptor-G protein precoupling. J. Pharmacol. Exp. Ther., 252, 1184-1196.
    • (1990) J. Pharmacol. Exp. Ther. , vol.252 , pp. 1184-1196
    • Jagadeesh, G.1    Cragoe, E.J.2    Deth, R.C.3
  • 19
    • 0027313323 scopus 로고
    • 35S]-GTPγS binding mediated by human muscarinic ml-m4 receptors: Antagonist studies
    • 35S]-GTPγS binding mediated by human muscarinic ml-m4 receptors: antagonist studies. Br. J. Pharmacol. 109, 1120-1127.
    • (1993) Br. J. Pharmacol. , vol.109 , pp. 1120-1127
    • Lazareno, S.1    Birdsall, N.J.2
  • 20
    • 0029094516 scopus 로고
    • Analysis of competitive agonist-antagonist interactions by nonlinear regression
    • LEW, M.J. & ANGUS, J.A. (1995). Analysis of competitive agonist-antagonist interactions by nonlinear regression. Trends Pharmacol. Sci., 16, 328-337.
    • (1995) Trends Pharmacol. Sci. , vol.16 , pp. 328-337
    • Lew, M.J.1    Angus, J.A.2
  • 21
    • 0001290493 scopus 로고
    • The influence of melatonin on the human circadian clock
    • ed. Fraschini, E., Reiter, R.J. & Stankov, B. Nato Asi Series. New York: Plenum Press
    • LEWY, A.J., SACK, R.L., AHMED, S., BAUER, V.K. & BLOOD, M.L. (1995). The influence of melatonin on the human circadian clock. In The Pineal Gland and Its Hormones: Fundamentals and Clinical Perspectives, ed. Fraschini, E., Reiter, R.J. & Stankov, B. Vol. 277, pp. 173-182, Nato Asi Series. New York: Plenum Press.
    • (1995) The Pineal Gland and Its Hormones: Fundamentals and Clinical Perspectives , vol.277 , pp. 173-182
    • Lewy, A.J.1    Sack, R.L.2    Ahmed, S.3    Bauer, V.K.4    Blood, M.L.5
  • 24
    • 0028054749 scopus 로고
    • Melatonin receptors: Localization, molecular pharmacology and physiological significance
    • MORGAN, P.J., BARRET, P., HOWELL, H.E. & HELLIWELL, R. (1994). Melatonin receptors: localization, molecular pharmacology and physiological significance. Neurochem. Int., 24, 101-146.
    • (1994) Neurochem. Int. , vol.24 , pp. 101-146
    • Morgan, P.J.1    Barret, P.2    Howell, H.E.3    Helliwell, R.4
  • 25
    • 0028972629 scopus 로고
    • 1 adenosine receptor/G protein coupling: Identification of a membrane protein that stabilizes the association of the receptor/G protein complex
    • 1 adenosine receptor/G protein coupling: Identification of a membrane protein that stabilizes the association of the receptor/G protein complex. Mol. Pharmacol., 48, 806-817.
    • (1995) Mol. Pharmacol. , vol.48 , pp. 806-817
    • Nanoff, C.1    Mitterauer, T.2    Roka, F.3    Hohenegger, M.4    Freissmuth, M.5
  • 26
    • 0029295605 scopus 로고
    • Distribution and characterization of the melatonin receptors in the hypothalamus and pituitary gland of three domestic ungulates
    • NONNO, R., CAPSONI, S., LUCINI, V., MOLLER, M., FRASCHINI, F. & STANKOV, B. (1995a). Distribution and characterization of the melatonin receptors in the hypothalamus and pituitary gland of three domestic ungulates. J. Pineal Res., 18, 207-216.
    • (1995) J. Pineal Res. , vol.18 , pp. 207-216
    • Nonno, R.1    Capsoni, S.2    Lucini, V.3    Moller, M.4    Fraschini, F.5    Stankov, B.6
  • 27
    • 0028981592 scopus 로고
    • 125]lodomelatonin binding sites in the bovine hippocampus are not sensitive to guanine nucleotides
    • 125]lodomelatonin binding sites in the bovine hippocampus are not sensitive to guanine nucleotides. Neurosci. Lett., 194, 113-116.
    • (1995) Neurosci. Lett. , vol.194 , pp. 113-116
    • Nonno, R.1    Lucini, V.2    Stankov, B.3    Fraschini, F.4
  • 29
    • 0028018966 scopus 로고
    • Cloning and characterization of a mammalian melatonin receptor that mediates reproductive and circadian responses
    • REPPERT, S.M., WEAVER, D.R. & EBISAWA, T. (1994). Cloning and characterization of a mammalian melatonin receptor that mediates reproductive and circadian responses. Neuron, 13, 1177-1185.
    • (1994) Neuron , vol.13 , pp. 1177-1185
    • Reppert, S.M.1    Weaver, D.R.2    Ebisawa, T.3
  • 31
    • 0027716547 scopus 로고
    • 2-Substituted 5-methoxy-N-acyltryptamines: Synthesis, binding affinity for the melatonin receptor, and evaluation of the biological activity
    • SPADONI, G., STANKOV, B., DURANTI, A., BIELLA, G., LUCINI, V., SALVATORI, A. & FRASCHINl, F. (1993). 2-Substituted 5-methoxy-N-acyltryptamines: synthesis, binding affinity for the melatonin receptor, and evaluation of the biological activity. J. Med. Chem., 36, 4069-4074.
    • (1993) J. Med. Chem. , vol.36 , pp. 4069-4074
    • Spadoni, G.1    Stankov, B.2    Duranti, A.3    Biella, G.4    Lucini, V.5    Salvatori, A.6    Fraschinl, F.7
  • 32
    • 0025979612 scopus 로고
    • Characterization and mapping of melatonin receptors in the brain of three mammalian species: Rabbit, horse and sheep
    • STANKOV, B., COZZI, B., LUCINI, V., FUMAGALLI, P., SCAGLIONE, F. & FRASCHINI, F. (1991). Characterization and mapping of melatonin receptors in the brain of three mammalian species: rabbit, horse and sheep. Neuroendocrinology, 53, 214-221.
    • (1991) Neuroendocrinology , vol.53 , pp. 214-221
    • Stankov, B.1    Cozzi, B.2    Lucini, V.3    Fumagalli, P.4    Scaglione, F.5    Fraschini, F.6
  • 34
    • 0028176054 scopus 로고
    • 2-adrenergic receptor activation of G proteins: Evidence for a precoupled receptor/G protein state
    • 2-adrenergic receptor activation of G proteins: evidence for a precoupled receptor/G protein state. Mol. Pharmacol., 45, 524-531.
    • (1994) Mol. Pharmacol. , vol.45 , pp. 524-531
    • Tian, W.-N.1    Duzic, E.2    Lanier, S.M.3    Deth, R.C.4
  • 35
    • 0028986870 scopus 로고
    • 35S]thio)triphosphate binding to membranes from human neuroblastoma SH-SY5Y cells
    • 35S]thio)triphosphate binding to membranes from human neuroblastoma SH-SY5Y cells. Mol. Pharmacol., 47, 848-854.
    • (1995) Mol. Pharmacol. , vol.47 , pp. 848-854
    • Traynor, J.R.1    Nahorski, S.R.2
  • 37
    • 0031565267 scopus 로고    scopus 로고
    • Efficacy I: A new method for estimating relative efficacy of full agonists via a newly defined efficacy related parameter
    • VENTER, D.P. (1997). Efficacy I: a new method for estimating relative efficacy of full agonists via a newly defined efficacy related parameter. Eur. J. Pharmacol., 320, 223-231.
    • (1997) Eur. J. Pharmacol. , vol.320 , pp. 223-231
    • Venter, D.P.1
  • 38
    • 0029895791 scopus 로고    scopus 로고
    • 1A melatonin receptor stably expressed in Chinese hamster ovary cells
    • 1A melatonin receptor stably expressed in Chinese hamster ovary cells. Mol. Pharmacol., 50, 166-174.
    • (1996) Mol. Pharmacol. , vol.50 , pp. 166-174
    • Wltt-Enderby, P.A.1    Dubocovich, M.L.2
  • 39
    • 0021697164 scopus 로고
    • 2-dopamine receptor of the anterior pituitary gland
    • 2-dopamine receptor of the anterior pituitary gland. Mol. Pharmacol., 26, 214-227.
    • (1984) Mol. Pharmacol. , vol.26 , pp. 214-227
    • Wreggett, K.A.1    De Lean, A.2


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