Complexation between local anaesthetics and β-cyclodextrin derivatives relationship between stability constants and in vitro membrane permeability of bupivacaine and lidocaine from their complexes

S.T.P. Pharma Sciences

Volumn 8, Issue 3, 1998, Pages 189-195

  Dollo, G ^a   Le Corre, P ^a   Chevanne, F ^a   Le Verge, R ^a  

^a UNIVERSITÉ DE RENNES 1   (France)

Author keywords

Cellulose membrane permeation; Cyclodextrins; Inclusion complexes; Local anaesthetics; Permeability coefficients; Stability constants

Indexed keywords

2 HYDROXYPROPYL BETA CYCLODEXTRIN; BETA CYCLODEXTRIN DERIVATIVE; BETA CYCLODEXTRIN SULFOBUTYL ETHER; BUPIVACAINE; LIDOCAINE; LOCAL ANESTHETIC AGENT; UNCLASSIFIED DRUG;

ARTICLE; COMPARTMENT MODEL; COMPLEX FORMATION; DERIVATIZATION; DRUG BINDING; DRUG SOLUBILITY; DRUG STABILITY; LOCAL ANESTHESIA; MEMBRANE PERMEABILITY; SPECTROPHOTOMETRY;

EID: 0031798707     PISSN: 11571489     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (18)

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