Enhanced dissolution of furosemide by coprecipitating or cogrinding with crospovidone

International Journal of Pharmaceutics

Volumn 175, Issue 1, 1998, Pages 17-24

  Shin, Sang Chul ^a   Oh, In Joon ^a   Lee, Yong Bok ^a   Choi, Hoo Kyun ^b   Choi, Jun Shik ^b  

^a Chonnam National University   (South Korea)

^b Chosun University   (South Korea)

Author keywords

Coprecipitate; Crospovidone; Dissolution; Furosemide; Ground mixture; Physicochemical characterization

Indexed keywords

CROSPOVIDONE; FUROSEMIDE; METHANOL;

ARTICLE; CONTROLLED STUDY; CRYSTAL; DRUG GRANULATION; DRUG SOLUBILITY; INFRARED SPECTROSCOPY; PHYSICAL CHEMISTRY; PRECIPITATION; PRIORITY JOURNAL; STOMACH JUICE; X RAY DIFFRACTION;

EID: 0031791549     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0378-5173(98)00260-9     Document Type: Article

References (22)

1. Ampolsuk, C., Mauro, J., Vyhuis, A.A., Shah, N., Jarowski, C.I., 1974. Influence of dispersion method on dissolution rate of digoxin-lactose and hydrocortisone-lactose triturates. J. Pharm. Sci. 63, 117-118.
2. Arias, M.J., Moyano, J.R., Gines, J.M., 1997. Investigation of the triamterene-β-cyclodextrin system prepared by cogrinding. Int. J. Pharm. 153, 181-189.
3. BASF Corporation, 1996. Kollidon, 3rd ed., BASF Aktiengesellschaft, Germany.
4. Iwata, M., Ueda, H., 1996. Dissolution properties of glibenclamide in combinations with polyvinylpyrrolidone. Drug Dev. Ind. Pharm. 22, 1161-1165.
5. Kai, T., Akiyama, Y., Nomura, S., Sato, M., 1996. Oral absorption improvement of poorly soluble drug using solid dispersion technique. Chem. Pharm. Bull. 44, 569-571.
6. Kigasawa, K., Maruyama, K., Tanaka, M., Watabe, K., Koyama, O., 1981. Biopharmaceutical studies of drugs. V. Dissolution properties and bioavailability of ground mixtures of poorly water soluble drugs and soluble proteins. Yakugaku Zasshi 101, 733.
7. Koh, I.B., Shin, S.C., Lee, Y.B., 1986a. Enhanced dissolution rates of piroxicam from the ground mixtures with chitin or chitosan. Arch. Pharm. Res. 9, 55-61.
8. Koh, I.B., Shin, S.C., Lee, Y.B., 1986b. Enhancement of dissolution properties of ketoprofen from ground mixtures with chitin or chitosan. J. Korean Pharm. Sci. 16, 36-41.
9. Mitrevej, A., Sinchaipanid, N., Junyaprasert, V., Warintournuwat, L., 1996. Effect of grinding of B-cyclodextrin and glibenclamide on tablet properties. Part I. In vitro. Drug Dev. Ind. Pharm. 22, 1237-1241.
10. Nakai, Y., Nakajima, K., Yamamoto, K., Terada, K., Konno, T., 1978. Effects of grinding on physical and chemical properties of crystalline medicinals with microcrystalline cellulose. II. Infrared spectra of medicinals on ground mixture. Chem. Pharm. Bull. 26, 3419.
11. Nagarsenker, M.S., Garad, S.D., 1998. Physical characterization and optimization of dissolution parameters of prochlorperazine maleate coevaporates. Int. J. Pharm. 160, 251-255.
12. Okimoto, K., Miyake, M., Ibiki, R., Yasumura, M., Ohnishi, N., Nakai, T., 1997. Dissolution mechanism and rate of solid dispersion particles of nilvadipine with hydroxypropylmethylcellulose. Int. J. Pharm. 159, 85-93.
13. Oster, G., Immergut, E.H., 1954. Ultraviolet and infrared spectral studies of polyvinylpyrrolidone. J. Am. Chem. Soc. 76, 1393.
14. Shah, N., Pytelewski, R., Eisen, H., Jarowski, C.I., 1974. Influence of dispersion method on dissolution rate and bioavailability of digoxin from triturations and compressed tablets. II. J. Pharm. Sci. 63, 339-344.
15. Shah, J.S., Chen, J.R., Chow, D., 1995. Preformulation study of etoposide: enhanced solubility and dissolution rate by solid-solid dispersions. Int. J. Pharm 113, 103-111.
16. Shin, S.C., 1979a. Dissolution characteristics of furosemide-polymer coprecipitates. Arch. Pharm. Res. 2, 35-48.
17. Shin, S.C., 1979b. Physicochemical characteristics of furosemide-PVP coprecipitates. Arch. Pharm. Res. 2, 49-64.
18. Shin, S.C., Cho, C.W., 1997. Physicochemical characterizations of piroxicam-poloxamer solid dispersion. Pharm. Dev. Technol. 2, 403-407.
19. Sugimoto, M., Okagaki, T., Narisawa, S., Koida, Y., Nakajima, K., 1998. Improvement of dissolution characteristics and bioavailability of poorly water-soluble drugs by novel cogrinding method using water-soluble polymer. Int. J. Pharm 160, 11-19.
20. Yamaguchi, G., Sakomoto, K., 1959. Effects of dry grinding on gibbsite. Bull. Chem. Soc. Jpn. 32, 1364.
21. Yamamoto, K., Nakano, M., Arita, T., Nakai, Y., 1974. Dissolution rate and bioavailability of griseofulvin from a ground mixture with microcrystalline cellulose. J. Pharmacokinet. Biopharm. 2, 487.
22. Yamamoto, K., Nakano, M., Arita, T., Takayama, Y., Nakai, Y., 1976. Dissolution behavior and bioavailability of phenytoin from a ground mixture with microcrystalline cellulose. J. Pharm. Sci. 65, 1484-1488.