메뉴 건너뛰기




Volumn 139, Issue 9, 1998, Pages 3736-3742

Effect of the high-affinity estrogen receptor ligand ICI 182,780 on the rat tibia

Author keywords

[No Author keywords available]

Indexed keywords

ANTIESTROGEN; ESTROGEN; FULVESTRANT;

EID: 0031730275     PISSN: 00137227     EISSN: None     Source Type: Journal    
DOI: 10.1210/endo.139.9.6172     Document Type: Article
Times cited : (74)

References (44)
  • 1
    • 0028838468 scopus 로고
    • Tissue-selective actions of estrogen analogs
    • Evans GL, Turner RT 1995 Tissue-selective actions of estrogen analogs. Bone [Suppl] 17:181S-190S
    • (1995) Bone [Suppl] , vol.17
    • Evans, G.L.1    Turner, R.T.2
  • 3
    • 0026395885 scopus 로고
    • A potent specific pure antiestrogen with clinical potential
    • Wakeling AE, Dukes M, Bowler J 1991 A potent specific pure antiestrogen with clinical potential. Cancer Res 51:3867-3873
    • (1991) Cancer Res , vol.51 , pp. 3867-3873
    • Wakeling, A.E.1    Dukes, M.2    Bowler, J.3
  • 4
    • 0027401411 scopus 로고
    • The future of new pure antiestrogens in clinical breast cancer
    • Wakeling AE 1993 The future of new pure antiestrogens in clinical breast cancer. Breast Cancer Res Treat 25:1-9
    • (1993) Breast Cancer Res Treat , vol.25 , pp. 1-9
    • Wakeling, A.E.1
  • 5
    • 0025084510 scopus 로고
    • Inhibition of estrogen receptor DNA binding by the "pure" antiestrogen ICI 163,384 appears to be mediated by impaired receptor dimerization
    • Falwell SE, White R, Hoare S, Syndenham M, Page M, Parker MG 1990 Inhibition of estrogen receptor DNA binding by the "pure" antiestrogen ICI 163,384 appears to be mediated by impaired receptor dimerization. Proc Natl Acad Sci USA 87:6883-6887
    • (1990) Proc Natl Acad Sci USA , vol.87 , pp. 6883-6887
    • Falwell, S.E.1    White, R.2    Hoare, S.3    Syndenham, M.4    Page, M.5    Parker, M.G.6
  • 6
    • 0029038986 scopus 로고
    • Analysis of estrogen receptor function in vitro reveals three distinct classes of antiestrogens
    • McDonnell DP, Clemm DL, Hermann T, Goldman ME, Pike JW 1995 Analysis of estrogen receptor function in vitro reveals three distinct classes of antiestrogens. Mol Endocrinol 9:659-669
    • (1995) Mol Endocrinol , vol.9 , pp. 659-669
    • McDonnell, D.P.1    Clemm, D.L.2    Hermann, T.3    Goldman, M.E.4    Pike, J.W.5
  • 7
    • 0027400930 scopus 로고
    • The efficacy and cost-effectiveness of adjuvant therapy of early breast cancer in premenopausal women
    • Smith TJ, Hillner BE 1993 The efficacy and cost-effectiveness of adjuvant therapy of early breast cancer in premenopausal women. J Clin Oncol 11:771-776
    • (1993) J Clin Oncol , vol.11 , pp. 771-776
    • Smith, T.J.1    Hillner, B.E.2
  • 9
    • 0025043542 scopus 로고
    • Long-term adjuvant tamoxifen therapy for breast cancer
    • Jordan VG 1990 Long-term adjuvant tamoxifen therapy for breast cancer. Breast Cancer Res Treat 15:125-136
    • (1990) Breast Cancer Res Treat , vol.15 , pp. 125-136
    • Jordan, V.G.1
  • 10
    • 0024312674 scopus 로고
    • Tamoxifen therapy in premenopausal breast cancer: Biology, efficacy and side effects
    • Love RR 1989 Tamoxifen therapy in premenopausal breast cancer: biology, efficacy and side effects. J Clin Oncol 7:803-815
    • (1989) J Clin Oncol , vol.7 , pp. 803-815
    • Love, R.R.1
  • 11
    • 0027762610 scopus 로고
    • Type I IGF receptor and acquired tamoxifen resistance in oestrogen-responsive human breast cancer cells
    • Wiseman LR, Johnson MD, Wakeling AE 1993 Type I IGF receptor and acquired tamoxifen resistance in oestrogen-responsive human breast cancer cells. Eur J Cancer 29A:2256-2264
    • (1993) Eur J Cancer , vol.29 A , pp. 2256-2264
    • Wiseman, L.R.1    Johnson, M.D.2    Wakeling, A.E.3
  • 12
    • 0023701360 scopus 로고
    • Novel antioestrogens without partial agonist activity
    • Wakeling AE, Bowler J 1988 Novel antioestrogens without partial agonist activity. J Steroid Biochem 31:654-658
    • (1988) J Steroid Biochem , vol.31 , pp. 654-658
    • Wakeling, A.E.1    Bowler, J.2
  • 13
    • 84995870933 scopus 로고
    • Human estrogen receptor transactivational capacity is determined by both cellular and promoter context and mediated by two functionally distinct intramolecular regions
    • Tzukerman MT, Esty A, Santiso-Mere D, Danielian P, Parker MG, Stein RB, Pike JW, McDonnell DP 1994 Human estrogen receptor transactivational capacity is determined by both cellular and promoter context and mediated by two functionally distinct intramolecular regions. Mol Endocrinol 8:21-30
    • (1994) Mol Endocrinol , vol.8 , pp. 21-30
    • Tzukerman, M.T.1    Esty, A.2    Santiso-Mere, D.3    Danielian, P.4    Parker, M.G.5    Stein, R.B.6    Pike, J.W.7    McDonnell, D.P.8
  • 14
    • 0031039888 scopus 로고    scopus 로고
    • Comparison of the ligand binding specificity and transcript tissue distribution of estrogen receptors α and β
    • Kuiper G, Carlsson B, Grandien K, Enmark E, Häggblad J, Nilsson S, Gustafsson J 1997 Comparison of the ligand binding specificity and transcript tissue distribution of estrogen receptors α and β. Endocrinology 138:863-870
    • (1997) Endocrinology , vol.138 , pp. 863-870
    • Kuiper, G.1    Carlsson, B.2    Grandien, K.3    Enmark, E.4    Häggblad, J.5    Nilsson, S.6    Gustafsson, J.7
  • 15
    • 0027139169 scopus 로고
    • The estrogen antagonist ICI 182,780 reduces cancellous bone volume in female rats
    • Gallagher A, Chambers TJ, Tobias JH 1993 The estrogen antagonist ICI 182,780 reduces cancellous bone volume in female rats. Endocrinology 133:2787-2791
    • (1993) Endocrinology , vol.133 , pp. 2787-2791
    • Gallagher, A.1    Chambers, T.J.2    Tobias, J.H.3
  • 19
    • 0020509916 scopus 로고
    • Relationships between surface, volume and thickness of iliac trabecular bone in aging and osteoporosis: Implications for the microanatomic and cellular mechanisms of bone loss
    • Parfitt AM, Mathews CHE, Villanueva AR, Kleerekoper M, Frame B, Rao DS 1983 Relationships between surface, volume and thickness of iliac trabecular bone in aging and osteoporosis: implications for the microanatomic and cellular mechanisms of bone loss. J Clin Invest 72:1396-1409
    • (1983) J Clin Invest , vol.72 , pp. 1396-1409
    • Parfitt, A.M.1    Mathews, C.H.E.2    Villanueva, A.R.3    Kleerekoper, M.4    Frame, B.5    Rao, D.S.6
  • 20
    • 0030962537 scopus 로고    scopus 로고
    • Characterization of the ovariectomized rat model for the evaluation of estrogen effects on plasma cholesterol levels
    • Lundeen SG, Carver JM, McKean M, Winneker RC 1997 Characterization of the ovariectomized rat model for the evaluation of estrogen effects on plasma cholesterol levels. Endocrinology 138:1552-1558
    • (1997) Endocrinology , vol.138 , pp. 1552-1558
    • Lundeen, S.G.1    Carver, J.M.2    McKean, M.3    Winneker, R.C.4
  • 21
    • 0021189787 scopus 로고
    • Evaluation of pathogenesis of skeletal changes in ovariectomized rats
    • Kalu DN 1984 Evaluation of pathogenesis of skeletal changes in ovariectomized rats. Endocrinology 115:507-512
    • (1984) Endocrinology , vol.115 , pp. 507-512
    • Kalu, D.N.1
  • 22
    • 0028212448 scopus 로고    scopus 로고
    • The effects of raloxifene on tibia histomorphometry in ovariectomized rats
    • Evans GL, Bryant HU, Magee DE, Sato M, Turner RT 1996 The effects of raloxifene on tibia histomorphometry in ovariectomized rats. Endocrinology 134:2283-2288
    • (1996) Endocrinology , vol.134 , pp. 2283-2288
    • Evans, G.L.1    Bryant, H.U.2    Magee, D.E.3    Sato, M.4    Turner, R.T.5
  • 23
    • 0023320347 scopus 로고
    • The effect of ovariectomy and 17β-estradiol on cortical bone histomorphometry in growing rats
    • Turner RT, Vandersteenhoven JJ, Bell NH 1987 The effect of ovariectomy and 17β-estradiol on cortical bone histomorphometry in growing rats. J Bone Miner Res 2:115-122
    • (1987) J Bone Miner Res , vol.2 , pp. 115-122
    • Turner, R.T.1    Vandersteenhoven, J.J.2    Bell, N.H.3
  • 24
    • 0023430358 scopus 로고
    • Tamoxifen prevents the skeletal effects of ovarian hormone deficiency in rats
    • Turner RT, Wakley GK, Hannon KS, Bell NH 1987 Tamoxifen prevents the skeletal effects of ovarian hormone deficiency in rats. J Bone Miner Res 2:449-456
    • (1987) J Bone Miner Res , vol.2 , pp. 449-456
    • Turner, R.T.1    Wakley, G.K.2    Hannon, K.S.3    Bell, N.H.4
  • 25
    • 0017597234 scopus 로고
    • Central action and a special comparison of the estrogenic effects of an antiestrogen on eating and body weight
    • Roy EJ, Maass CA, Wade GN 1977 Central action and a special comparison of the estrogenic effects of an antiestrogen on eating and body weight. Physiol Behav 18:137-140
    • (1977) Physiol Behav , vol.18 , pp. 137-140
    • Roy, E.J.1    Maass, C.A.2    Wade, G.N.3
  • 26
    • 0029618205 scopus 로고
    • Tissue-specific actions of antioestrogens
    • Wakeling AE 1995 Tissue-specific actions of antioestrogens. Mutat Res 333:45-49
    • (1995) Mutat Res , vol.333 , pp. 45-49
    • Wakeling, A.E.1
  • 27
    • 0030933163 scopus 로고    scopus 로고
    • Clomiphene prevents cancellous bone loss from tibia of ovariectomized rats
    • Jimenez MA, Magee DE, Bryant HU, Turner RT 1997 Clomiphene prevents cancellous bone loss from tibia of ovariectomized rats. Endocrinology 138:1794-1800
    • (1997) Endocrinology , vol.138 , pp. 1794-1800
    • Jimenez, M.A.1    Magee, D.E.2    Bryant, H.U.3    Turner, R.T.4
  • 28
    • 0029016173 scopus 로고
    • Droloxifene, a new estrogen antagonist/agonist prevents bone loss in ovariectomized rats
    • Ke HZ, Simmons HA, Pirie CM, Crawford DT, Thompson DD 1995 Droloxifene, a new estrogen antagonist/agonist prevents bone loss in ovariectomized rats. Endocrinology 136:2435-2441
    • (1995) Endocrinology , vol.136 , pp. 2435-2441
    • Ke, H.Z.1    Simmons, H.A.2    Pirie, C.M.3    Crawford, D.T.4    Thompson, D.D.5
  • 30
    • 0022475934 scopus 로고
    • Histologic evidence for osteopenia and increased bone turnover in ovariectomized rats
    • Wronski TJ, Walsh CC, Ignaszewski LA 1986 Histologic evidence for osteopenia and increased bone turnover in ovariectomized rats. Bone 7:119-123
    • (1986) Bone , vol.7 , pp. 119-123
    • Wronski, T.J.1    Walsh, C.C.2    Ignaszewski, L.A.3
  • 31
    • 0024404114 scopus 로고
    • The differential effects of gonadal insufficiency on bone histomorphometry in male and female rats
    • Turner RT, Hannon KS, Demers L, Buchanan J, Bell NH 1989 The differential effects of gonadal insufficiency on bone histomorphometry in male and female rats. J Bone Miner Res 4:557-563
    • (1989) J Bone Miner Res , vol.4 , pp. 557-563
    • Turner, R.T.1    Hannon, K.S.2    Demers, L.3    Buchanan, J.4    Bell, N.H.5
  • 32
    • 0027400961 scopus 로고
    • Mechanism of action of estrogen on cancellous bone balance in tibiae of ovariectomized growing rats: Inhibition of indices of formation and resorption
    • Turner RT, Evans GL, Wakley GK 1993 Mechanism of action of estrogen on cancellous bone balance in tibiae of ovariectomized growing rats: inhibition of indices of formation and resorption. J Bone Miner Res 8:359-366
    • (1993) J Bone Miner Res , vol.8 , pp. 359-366
    • Turner, R.T.1    Evans, G.L.2    Wakley, G.K.3
  • 33
    • 0023690523 scopus 로고
    • Estrogen treatment prevents osteopenia, and depresses bone turnover in ovariectomized rats
    • Wronski TJ, Cintron M, Doherty AL, Dann LM 1988 Estrogen treatment prevents osteopenia, and depresses bone turnover in ovariectomized rats. Endocrinology 123:681-686
    • (1988) Endocrinology , vol.123 , pp. 681-686
    • Wronski, T.J.1    Cintron, M.2    Doherty, A.L.3    Dann, L.M.4
  • 34
    • 0027955121 scopus 로고
    • Reduced chondroclast differentiation results in increased cancellous bone volume in estrogen-treated growing rats
    • Turner RT, Evans GL, Wakley GK 1994 Reduced chondroclast differentiation results in increased cancellous bone volume in estrogen-treated growing rats. Endocrinology 134:461-466
    • (1994) Endocrinology , vol.134 , pp. 461-466
    • Turner, R.T.1    Evans, G.L.2    Wakley, G.K.3
  • 35
    • 0024199404 scopus 로고
    • Growth plate structure and function
    • Hunziker EB 1988 Growth plate structure and function. Pathol Immunopathol Res 7:9-13
    • (1988) Pathol Immunopathol Res , vol.7 , pp. 9-13
    • Hunziker, E.B.1
  • 36
    • 0002043349 scopus 로고
    • The physiological and clinical significance of bone histomorphometric data
    • Recker RR (ed) CRC Press, Inc, Boca Raton
    • Parfitt AM 1983 The physiological and clinical significance of bone histomorphometric data. In: Recker RR (ed) Bone Histomorphometry. CRC Press, Inc, Boca Raton, pp 143-223
    • (1983) Bone Histomorphometry , pp. 143-223
    • Parfitt, A.M.1
  • 37
    • 0029816177 scopus 로고    scopus 로고
    • Trabecular and endocortical bone surfaces in the rat: Modeling or remodeling?
    • Erben RG 1996 Trabecular and endocortical bone surfaces in the rat: modeling or remodeling? Anat Rec 246:39-46
    • (1996) Anat Rec , vol.246 , pp. 39-46
    • Erben, R.G.1
  • 38
    • 0026068145 scopus 로고
    • Skeletal response of ovariectomized rats to low and high doses of 17β-estradiol
    • Kalu DN, Liu CC, Salerno E, Hollis B, Echon R, Ray M 1991 Skeletal response of ovariectomized rats to low and high doses of 17β-estradiol. Bone Miner 14:175-187
    • (1991) Bone Miner , vol.14 , pp. 175-187
    • Kalu, D.N.1    Liu, C.C.2    Salerno, E.3    Hollis, B.4    Echon, R.5    Ray, M.6
  • 39
    • 0030993372 scopus 로고    scopus 로고
    • Estrogen regulates the rate of bone turnover but bone balance in ovariectomized rats is modulated by prevailing mechanical strain
    • Westerlind KC, Wronski TJ, Ritman EL, Luo Z, An K, Bell NH, Turner RT 1997 Estrogen regulates the rate of bone turnover but bone balance in ovariectomized rats is modulated by prevailing mechanical strain. Proc Natl Acad Sci USA 94:4199-4204
    • (1997) Proc Natl Acad Sci USA , vol.94 , pp. 4199-4204
    • Westerlind, K.C.1    Wronski, T.J.2    Ritman, E.L.3    Luo, Z.4    An, K.5    Bell, N.H.6    Turner, R.T.7
  • 40
    • 0021759939 scopus 로고
    • Mechanisms of hormone action: Parallels in receptor-mediated signal propagation for steroid and receptor-mediated signal propagation for steroid and peptide effectors
    • Szego CM 1984 Mechanisms of hormone action: parallels in receptor-mediated signal propagation for steroid and receptor-mediated signal propagation for steroid and peptide effectors. Life Sci 35:2383-2396
    • (1984) Life Sci , vol.35 , pp. 2383-2396
    • Szego, C.M.1
  • 41
    • 15644380245 scopus 로고    scopus 로고
    • Estrogen results in rapid, differential regulation of immediate response, growth factor, and matrix protein genes in bone and uterus of growing rats
    • Minneapolis MN
    • Kidder LS, Zhang M, Wronski TJ, Turner RT Estrogen results in rapid, differential regulation of immediate response, growth factor, and matrix protein genes in bone and uterus of growing rats. Program of the 79th Annual Meeting of The Endocrine Society, Minneapolis MN, 1997, p 547
    • (1997) 79th Annual Meeting of the Endocrine Society , pp. 547
    • Kidder, L.S.1    Zhang, M.2    Wronski, T.J.3    Turner, R.T.4
  • 43
    • 0029841146 scopus 로고    scopus 로고
    • Identification of an estrogen response element activated by metabolites of 17β-estradiol and raloxifene
    • Yang NN, Venugopalan M, Hardikar S, Glasebrook A 1996 Identification of an estrogen response element activated by metabolites of 17β-estradiol and raloxifene. Science 273:1222-1225
    • (1996) Science , vol.273 , pp. 1222-1225
    • Yang, N.N.1    Venugopalan, M.2    Hardikar, S.3    Glasebrook, A.4
  • 44
    • 0030898711 scopus 로고    scopus 로고
    • The quinone reductase gene: A unique estrogen receptor-regulated gene that is activated by antiestrogens
    • Montano MM, Katzenellenbogen BS 1997 The quinone reductase gene: a unique estrogen receptor-regulated gene that is activated by antiestrogens. Proc Natl Acad Sci USA 94:2581-2586
    • (1997) Proc Natl Acad Sci USA , vol.94 , pp. 2581-2586
    • Montano, M.M.1    Katzenellenbogen, B.S.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.