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Volumn 13, Issue 6, 1998, Pages 619-624

Comparative mutagenic and genotoxic effects of three antimalarial drugs, chloroquine, primaquine and amodiaquine

Author keywords

[No Author keywords available]

Indexed keywords

AMODIAQUINE; ANTIMALARIAL AGENT; CHLOROQUINE; PRIMAQUINE;

EID: 0031726186     PISSN: 02678357     EISSN: None     Source Type: Journal    
DOI: 10.1093/mutage/13.6.619     Document Type: Article
Times cited : (42)

References (49)
  • 3
    • 0014425983 scopus 로고
    • Methemoglobinemia provoked by malarial chemoprophylaxis in Vietnam
    • Cohen,R.J., Sachs,J.R., Wicker,D.J. and Courad,M.E. (1986) Methemoglobinemia provoked by malarial chemoprophylaxis in Vietnam. New Engl. J. Med., 279, 1127-1131.
    • (1986) New Engl. J. Med. , vol.279 , pp. 1127-1131
    • Cohen, R.J.1    Sachs, J.R.2    Wicker, D.J.3    Courad, M.E.4
  • 4
    • 0000029821 scopus 로고
    • Spectrophotometer studies of the interaction of chloroquine with deoxyribonucleic acid
    • Cohen,S.N. and Yielding,K.L. (1965) Spectrophotometer studies of the interaction of chloroquine with deoxyribonucleic acid. J. Biol. Chem., 240, 3123-3131.
    • (1965) J. Biol. Chem. , vol.240 , pp. 3123-3131
    • Cohen, S.N.1    Yielding, K.L.2
  • 5
    • 0020646740 scopus 로고
    • Mutagenicity of antiamebic and anthelmintic drugs in the Salmonella typhimurium test system
    • Cortinas de Nava,C., Espinosa,J., Garcia,L., Zapata,A.M. and Martinez,E. (1983) Mutagenicity of antiamebic and anthelmintic drugs in the Salmonella typhimurium test system. Mutat. Res., 117, 79-91.
    • (1983) Mutat. Res. , vol.117 , pp. 79-91
    • Cortinas De Nava, C.1    Espinosa, J.2    Garcia, L.3    Zapata, A.M.4    Martinez, E.5
  • 6
    • 0009663357 scopus 로고
    • A multiple comparison procedure for comparing several treatments with the control
    • Dunnett,C.W. (1955) A multiple comparison procedure for comparing several treatments with the control. J. Am. Statist. Assoc., 50, 1096-1121.
    • (1955) J. Am. Statist. Assoc. , vol.50 , pp. 1096-1121
    • Dunnett, C.W.1
  • 7
    • 0024560465 scopus 로고
    • Influence of the Uvr repair system on the mutagenicity of antiparasitic drugs
    • Espinosa-Aguirre,J.J., Ramirez Santos,J. and Cortinas de Nava,C. (1989) Influence of the Uvr repair system on the mutagenicity of antiparasitic drugs. Mutat. Res., 222, 161-166.
    • (1989) Mutat. Res. , vol.222 , pp. 161-166
    • Espinosa-Aguirre, J.J.1    Ramirez Santos, J.2    Cortinas De Nava, C.3
  • 8
    • 0017884861 scopus 로고
    • Inhibition of precursor incorporation into nucleic acids of mammalian tissues by antimalarial aminoquinolins
    • Field,R.C., Bibson,B.R., Holbrook,D.J.,Jr and McCall,B.N. (1978) Inhibition of precursor incorporation into nucleic acids of mammalian tissues by antimalarial aminoquinolins. Br. J. Pharmacol., 62, 159-164.
    • (1978) Br. J. Pharmacol. , vol.62 , pp. 159-164
    • Field, R.C.1    Bibson, B.R.2    Holbrook Jr., D.J.3    McCall, B.N.4
  • 9
    • 0015410809 scopus 로고
    • Liver microsomal metabolism of aflatoxin B1 to a reactive derivative toxic to Salmonella typhimurium TA1530
    • Garner,R.C., Miller,E.C. and Miller,J.A. (1972) Liver microsomal metabolism of aflatoxin B1 to a reactive derivative toxic to Salmonella typhimurium TA1530. Cancer Res., 32, 2085-2066.
    • (1972) Cancer Res. , vol.32 , pp. 2085-12066
    • Garner, R.C.1    Miller, E.C.2    Miller, J.A.3
  • 11
    • 0029314175 scopus 로고    scopus 로고
    • Genetic toxicology of four commonly used benzodiazepines: A review
    • Giri,A.K. (1996) Genetic toxicology of four commonly used benzodiazepines: a review. Mutat. Res., 340, 93-108.
    • (1996) Mutat. Res. , vol.340 , pp. 93-108
    • Giri, A.K.1
  • 12
    • 0031002998 scopus 로고    scopus 로고
    • Genetic toxicology of epichlorohydrin: A review
    • Giri,A.K. (1997) Genetic toxicology of epichlorohydrin: a review. Mutat. Res., 386, 25-38.
    • (1997) Mutat. Res. , vol.386 , pp. 25-38
    • Giri, A.K.1
  • 13
    • 0024467696 scopus 로고
    • Sister chromatid exchange and chromosome aberrations for four aliphatic epoxides in mice
    • Giri,A.K., Messerly,E.A. and Sinsheimer,J.E. (1989) Sister chromatid exchange and chromosome aberrations for four aliphatic epoxides in mice. Mutat. Res., 224, 253-261.
    • (1989) Mutat. Res. , vol.224 , pp. 253-261
    • Giri, A.K.1    Messerly, E.A.2    Sinsheimer, J.E.3
  • 14
    • 0026514326 scopus 로고
    • Sister chromatid exchange and chromosome aberrations induced by paracetamol in vivo in bone marrow cells of mice
    • Giri,A.K., Sai Sivam,S. and Khan,K.A. (1992) Sister chromatid exchange and chromosome aberrations induced by paracetamol in vivo in bone marrow cells of mice. Mutat. Res., 278, 253-257.
    • (1992) Mutat. Res. , vol.278 , pp. 253-257
    • Giri, A.K.1    Sai Sivam, S.2    Khan, K.A.3
  • 16
    • 0041109123 scopus 로고
    • Drugs used in the chemotherapy of malaria
    • Goodman,L.S. and Gilman,A. (eds), Macmillan Publishing Co. Inc., New York
    • Goodman,X.S. and Gilman,A. (1980) Drugs used in the chemotherapy of malaria. In Goodman,L.S. and Gilman,A. (eds), The Pharmacological Basis of Therapeutics, 6th edn. Macmillan Publishing Co. Inc., New York, pp. 1038-1060.
    • (1980) The Pharmacological Basis of Therapeutics, 6th Edn. , pp. 1038-1060
    • Goodman, X.S.1    Gilman, A.2
  • 17
    • 0030596091 scopus 로고    scopus 로고
    • Mutagenicity of dihydroxy benzenes and dihydroxy naphthalenes for Ames Salmonella tester strains
    • Hakura,A., Tsutsui,Y., Mochida,H., Sugihara,Y., Mikami,T. and Sagami,F. (1996) Mutagenicity of dihydroxy benzenes and dihydroxy naphthalenes for Ames Salmonella tester strains. Mutat. Res., 371, 293-299.
    • (1996) Mutat. Res. , vol.371 , pp. 293-299
    • Hakura, A.1    Tsutsui, Y.2    Mochida, H.3    Sugihara, Y.4    Mikami, T.5    Sagami, F.6
  • 18
    • 1342317031 scopus 로고
    • Acridine antimalarials
    • Acheson,R-M. (ed.), Wiley, New York, NY
    • Henry,D.W. (1973) Acridine antimalarials. In Acheson,R-M. (ed.), Acridines, 2nd Edn. Wiley, New York, NY, pp. 829-850.
    • (1973) Acridines, 2nd Edn. , pp. 829-850
    • Henry, D.W.1
  • 19
    • 0000437062 scopus 로고
    • Average generation time: A new method for analyzing cellular proliferation kinetics based on bromodeoxyuridine-dependent chromosome differential staining patterns
    • Ivett,J.L. and Tice,R.R. (1982) Average generation time: a new method for analyzing cellular proliferation kinetics based on bromodeoxyuridine-dependent chromosome differential staining patterns. Environ. Mutagen., 4, 358-365.
    • (1982) Environ. Mutagen. , vol.4 , pp. 358-365
    • Ivett, J.L.1    Tice, R.R.2
  • 20
    • 0021688019 scopus 로고
    • Mutagenicity examination of several non steroidal anti-inflammatory drugs in bacterial systems
    • Kadotani,S., Arisawa,M. and Maruyama,H.B. (1984) Mutagenicity examination of several non steroidal anti-inflammatory drugs in bacterial systems. Mutat. Res., 138, 133-136.
    • (1984) Mutat. Res. , vol.138 , pp. 133-136
    • Kadotani, S.1    Arisawa, M.2    Maruyama, H.B.3
  • 21
    • 0000820622 scopus 로고
    • A new tester strain (TA102) with A-T base pairs at the site of mutation detects oxidative mutagens
    • Levin,D.E., Hollstein., Christman,M.F., Schwiers,E.A. and Ames,B.A. (1982) A new tester strain (TA102) with A-T base pairs at the site of mutation detects oxidative mutagens. Proc. Natl Acad. Sci. USA, 79, 7445-7449.
    • (1982) Proc. Natl Acad. Sci. USA , vol.79 , pp. 7445-7449
    • Levin, D.E.1    Hollstein2    Christman, M.F.3    Schwiers, E.A.4    Ames, B.A.5
  • 22
    • 0015849323 scopus 로고
    • Accumulation of drugs on melanin
    • Linquist,N.G. (1973) Accumulation of drugs on melanin. Acta. Radial., 325 (suppl.), 1-92.
    • (1973) Acta. Radial. , vol.325 , Issue.SUPPL. , pp. 1-92
    • Linquist, N.G.1
  • 24
    • 0020533372 scopus 로고
    • Revised methods for Salmonella mutagenicity test
    • Maron,D.M. and Ames,B.N. (1983) Revised methods for Salmonella mutagenicity test. Mutat. Res., 113, 173-215.
    • (1983) Mutat. Res. , vol.113 , pp. 173-215
    • Maron, D.M.1    Ames, B.N.2
  • 25
    • 0023261114 scopus 로고
    • Methemoglobinogenic potential of primaquine and its mutagenicity in Ames test
    • Marrs,T.C., Bright,J.E. and Morris,B.C. (1987) Methemoglobinogenic potential of primaquine and its mutagenicity in Ames test. Toxicol. Lett., 36, 281-287.
    • (1987) Toxicol. Lett. , vol.36 , pp. 281-287
    • Marrs, T.C.1    Bright, J.E.2    Morris, B.C.3
  • 26
    • 85038550535 scopus 로고    scopus 로고
    • J.E.F.Reynolds (ed.). The Pharmaceutical Press, London, UK
    • Martindale,H. (1996) Martindale The Extra Pharmacopoeia. J.E.F.Reynolds (ed.). The Pharmaceutical Press, London, UK, p. 464.
    • (1996) Martindale the Extra Pharmacopoeia , pp. 464
    • Martindale, H.1
  • 27
    • 0010671691 scopus 로고
    • Laboratory studies of the four aminoquinolin antimalarials. I. Some biochemical characteristics of chloroquine, hydrochloroquine and SN-7718
    • McChesney,E.W. and McAnliff,J.P. (1961) Laboratory studies of the four aminoquinolin antimalarials. I. Some biochemical characteristics of chloroquine, hydrochloroquine and SN-7718. Antibiot. Chemother., 11, 800-810.
    • (1961) Antibiot. Chemother. , vol.11 , pp. 800-810
    • McChesney, E.W.1    McAnliff, J.P.2
  • 28
    • 0014083266 scopus 로고
    • Tissue distribution of Chloroquine, hydroxychloroquine and desethyl chloroquine in the rat
    • McChesney,E.W., Banks,W.F.,Jr and Fabian,R.J. (1967) Tissue distribution of Chloroquine, hydroxychloroquine and desethyl chloroquine in the rat. Toxicol. Appl. Pharmacol., 10, 501-513.
    • (1967) Toxicol. Appl. Pharmacol. , vol.10 , pp. 501-513
    • McChesney, E.W.1    Banks Jr., W.F.2    Fabian, R.J.3
  • 29
    • 0020699685 scopus 로고
    • Improved sister chromatid differentiation using paraffin coated bromodeoxyuridine tablets in mice
    • McFee,A.F., Lowe,K. and San Sebastian,J.R. (1983) Improved sister chromatid differentiation using paraffin coated bromodeoxyuridine tablets in mice. Mutat. Res., 119, 83-88.
    • (1983) Mutat. Res. , vol.119 , pp. 83-88
    • McFee, A.F.1    Lowe, K.2    San Sebastian, J.R.3
  • 30
    • 0016176815 scopus 로고
    • Chloroquine inhibition of repair of DNA damage induced in mammalian cells by methyl methane sulphonate
    • Michael,R.O. and William,G.M. (1974) Chloroquine inhibition of repair of DNA damage induced in mammalian cells by methyl methane sulphonate. Mutat. Res., 25, 391-396.
    • (1974) Mutat. Res. , vol.25 , pp. 391-396
    • Michael, R.O.1    William, G.M.2
  • 31
    • 0023025805 scopus 로고
    • Aspects of chloroquine mutagenicity
    • Obaseiki-Ebor,E.E. and Obasi,E.E. (1986) Aspects of chloroquine mutagenicity. Mutat. Res., 175, 51-59.
    • (1986) Mutat. Res. , vol.175 , pp. 51-59
    • Obaseiki-Ebor, E.E.1    Obasi, E.E.2
  • 32
    • 0028167881 scopus 로고
    • Mutagenic evaluation of primaquine, pentaquine and pamaquine in the Salmonella/mammalian microsome assay
    • Ono,T., Norimatsu,M. and Yoshimura,H. (1994) Mutagenic evaluation of primaquine, pentaquine and pamaquine in the Salmonella/mammalian microsome assay. Mutat. Res., 325, 7-10.
    • (1994) Mutat. Res. , vol.325 , pp. 7-10
    • Ono, T.1    Norimatsu, M.2    Yoshimura, H.3
  • 33
    • 0016328318 scopus 로고
    • New Giemsa method for the differential staining of sister chromatids
    • Perry,P. and Wolff,S. (1974) New Giemsa method for the differential staining of sister chromatids. Nature, 251, 156-158.
    • (1974) Nature , vol.251 , pp. 156-158
    • Perry, P.1    Wolff, S.2
  • 34
    • 0030724973 scopus 로고    scopus 로고
    • Comparative mutagenic and genotoxic effects of three propionic acid derivatives ibuprofen, ketoprofen and naproxen
    • Philipose,B., Singh,R., Khan,A.K. and Giri,A.K. (1997) Comparative mutagenic and genotoxic effects of three propionic acid derivatives ibuprofen, ketoprofen and naproxen. Mutat. Res., 393, 123-131.
    • (1997) Mutat. Res. , vol.393 , pp. 123-131
    • Philipose, B.1    Singh, R.2    Khan, A.K.3    Giri, A.K.4
  • 35
    • 0023281076 scopus 로고
    • Mammalian in vivo cytogenetic assays: Analysis of chromosome aberrations in bone marrow cells
    • Preston,R.J., Dean,B.J., Galloway,S., Holden,H., McFee,A.F. and Shelby,M. (1987) Mammalian in vivo cytogenetic assays: analysis of chromosome aberrations in bone marrow cells. Mutat. Res., 189, 157-165.
    • (1987) Mutat. Res. , vol.189 , pp. 157-165
    • Preston, R.J.1    Dean, B.J.2    Galloway, S.3    Holden, H.4    McFee, A.F.5    Shelby, M.6
  • 36
    • 0018895141 scopus 로고
    • Simultaneous detection of chromosomal aberrations and sister chromatid exchange: Experience with DNA intercalating agents
    • Raj,S.A. and Heddle,J.A. (1980) Simultaneous detection of chromosomal aberrations and sister chromatid exchange: experience with DNA intercalating agents. Mutat. Res., 78, 253-260.
    • (1980) Mutat. Res. , vol.78 , pp. 253-260
    • Raj, S.A.1    Heddle, J.A.2
  • 37
    • 0026674717 scopus 로고
    • Acute intramuscular haemolysis in vanuater following a single dose of primaquine in individuals with glucose-6-phosphate deficiency
    • Reever,P.A., Toalin,H., Kaneko,A., Hall,J.J. and Ganczakowski,M. (1992) Acute intramuscular haemolysis in vanuater following a single dose of primaquine in individuals with glucose-6-phosphate deficiency. J. Trop. Med. Hyg., 95, 349-351.
    • (1992) J. Trop. Med. Hyg. , vol.95 , pp. 349-351
    • Reever, P.A.1    Toalin, H.2    Kaneko, A.3    Hall, J.J.4    Ganczakowski, M.5
  • 38
    • 0018396446 scopus 로고
    • Mutagenicity evaluation of the two antimalarial agents chloroquine and mefloquine using a bacterial fluctuation test
    • Schupbach,M.E. (1979) Mutagenicity evaluation of the two antimalarial agents chloroquine and mefloquine using a bacterial fluctuation test. Mutat. Res., 68, 41-49.
    • (1979) Mutat. Res. , vol.68 , pp. 41-49
    • Schupbach, M.E.1
  • 39
    • 0022453403 scopus 로고
    • Sister chromatid exchange and chromosome aberration analyses in mice after in vivo exposure to acrylonitrile, styrene, or butadiene monoxide
    • Sharief,Y., Brown,A.M., Backer,L.C., Campbell,A.J., Westbrook-Collins,B., Stead,A.G. and Allen,J.W. (1986) Sister chromatid exchange and chromosome aberration analyses in mice after in vivo exposure to acrylonitrile, styrene, or butadiene monoxide. Environ. Mutagen., 8, 439-448.
    • (1986) Environ. Mutagen. , vol.8 , pp. 439-448
    • Sharief, Y.1    Brown, A.M.2    Backer, L.C.3    Campbell, A.J.4    Westbrook-Collins, B.5    Stead, A.G.6    Allen, J.W.7
  • 40
    • 0024326905 scopus 로고
    • Toxicological consequences of chloroquine and ethanol on the developing foetus
    • Sharma,A. and Rawat,A.K. (1989) Toxicological consequences of chloroquine and ethanol on the developing foetus. Pharmacol. Biochem. Behav., 34, 77-82.
    • (1989) Pharmacol. Biochem. Behav. , vol.34 , pp. 77-82
    • Sharma, A.1    Rawat, A.K.2
  • 41
    • 0022965360 scopus 로고
    • Comparison of the Ames assay and the induction of sister chromatid exchanges: Results with ten pharmaceuticals and five selected agents
    • Shubber,E.K., Jacobson-Kram,D. and Williams,J.R. (1986) Comparison of the Ames assay and the induction of sister chromatid exchanges: results with ten pharmaceuticals and five selected agents. Cell. biol. Toxicol., 2, 379-399.
    • (1986) Cell. Biol. Toxicol. , vol.2 , pp. 379-399
    • Shubber, E.K.1    Jacobson-Kram, D.2    Williams, J.R.3
  • 42
    • 0014549424 scopus 로고
    • Nuclear magnetic resonance studies of the interaction of chloroquine diphosphate with adenosine diphosphate and other nucleotides
    • Sternglanz,H., Yielding,K.C. and Pruitt,K.M. (1969) Nuclear magnetic resonance studies of the interaction of chloroquine diphosphate with adenosine diphosphate and other nucleotides. Mol. Pharmacol., 5, 376-381.
    • (1969) Mol. Pharmacol. , vol.5 , pp. 376-381
    • Sternglanz, H.1    Yielding, K.C.2    Pruitt, K.M.3
  • 43
    • 0023493481 scopus 로고
    • Frameshift mutagenesis by chloroquine in e coli and S. typhimurium
    • Thomas,S.M., Silburn,K.A. and MacPhee,D.G. (1987) Frameshift mutagenesis by chloroquine in E coli and S. typhimurium. Mutat. Res., 192, 233-237.
    • (1987) Mutat. Res. , vol.192 , pp. 233-237
    • Thomas, S.M.1    Silburn, K.A.2    MacPhee, D.G.3
  • 44
    • 0014945759 scopus 로고
    • Variation of the supercoils in closed circular DNA by binding of antibiotics and drugs. Evidence for molecular models involving interaction
    • Waring,M. (1970) Variation of the supercoils in closed circular DNA by binding of antibiotics and drugs. Evidence for molecular models involving interaction. J. Mol. Biol., 54, 247-279.
    • (1970) J. Mol. Biol. , vol.54 , pp. 247-279
    • Waring, M.1
  • 45
    • 0001890401 scopus 로고    scopus 로고
    • Malaria and other diseases caused by red blood cell parasites
    • Fauci,A., Braunwald,E., Isselbacher,K.J., Wilson,J.D., Martin,J.B., Kasper,D.L., Hauser,S.L. and Longo,D.L. (eds), McGraw-Hill, New York, NY
    • White,N.J. and Breman,J.G. (1998) Malaria and other diseases caused by red blood cell parasites. In Fauci,A., Braunwald,E., Isselbacher,K.J., Wilson,J.D., Martin,J.B., Kasper,D.L., Hauser,S.L. and Longo,D.L. (eds), Harrison's Principles of Internal Medicine, 14th Edn. McGraw-Hill, New York, NY, Vol. 1, p. 1187.
    • (1998) Harrison's Principles of Internal Medicine, 14th Edn. , vol.1 , pp. 1187
    • White, N.J.1    Breman, J.G.2
  • 46
    • 0015513032 scopus 로고
    • The inhibition in vitro of bacterial DNA polymerase and RNA polymerase by antimalarial 8-aminoquinolines and by chloroquine
    • Wichard,L.P., Washington,M.E. and Holbrook,D.J.,Jr (1972) The inhibition in vitro of bacterial DNA polymerase and RNA polymerase by antimalarial 8-aminoquinolines and by chloroquine. Biochim. Biophys. Acta, 287, 52-67.
    • (1972) Biochim. Biophys. Acta , vol.287 , pp. 52-67
    • Wichard, L.P.1    Washington, M.E.2    Holbrook Jr., D.J.3
  • 48
    • 0022398120 scopus 로고
    • Testing of chloroquine and quinacrine for mutagenicity in Drosophila melanogater
    • Xamena,N., Creus,A., Velazqez,A. and Marcos,R. (1985) Testing of chloroquine and quinacrine for mutagenicity in Drosophila melanogater. Mutat. Res., 158, 177-180.
    • (1985) Mutat. Res. , vol.158 , pp. 177-180
    • Xamena, N.1    Creus, A.2    Velazqez, A.3    Marcos, R.4


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