메뉴 건너뛰기




Volumn 28, Issue 8, 1998, Pages 759-766

Effect of a new rifamycin derivative, rifalazil, on liver microsomal enzyme induction in rat and dog

Author keywords

[No Author keywords available]

Indexed keywords

CYTOCHROME P450; MICROSOME ENZYME; RIFALAZIL; RIFAMYCIN DERIVATIVE; UNCLASSIFIED DRUG;

EID: 0031691174     PISSN: 00498254     EISSN: None     Source Type: Journal    
DOI: 10.1080/004982598239173     Document Type: Article
Times cited : (35)

References (34)
  • 2
    • 0027971263 scopus 로고
    • Activity of KRM-1648 alone or in combination with ethambutol or clarithromycin against Mycobacterium avium in beige mouse model of disseminated infection
    • BERMUDEZ, L. E., KOLONOSKI, P., YOUNG, L. S. and INDERLIED, C. B., 1994, Activity of KRM-1648 alone or in combination with ethambutol or clarithromycin against Mycobacterium avium in beige mouse model of disseminated infection. Antimicrobial Agents and Chemotherapy, 38, 1844-1848.
    • (1994) Antimicrobial Agents and Chemotherapy , vol.38 , pp. 1844-1848
    • Bermudez, L.E.1    Kolonoski, P.2    Young, L.S.3    Inderlied, C.B.4
  • 3
    • 0022968251 scopus 로고
    • Induction of mixed function oxidase activity in man by rifapentine (MDL 473), a long-acting rifamycin derivative
    • DURAND, D. V., HAMPDEN, C., BOOBIS, A. R., PARK, B. K. and DABIES, D. S., 1986, Induction of mixed function oxidase activity in man by rifapentine (MDL 473), a long-acting rifamycin derivative. British Journal of Clinical Pharmacology, 21, 1-7.
    • (1986) British Journal of Clinical Pharmacology , vol.21 , pp. 1-7
    • Durand, D.V.1    Hampden, C.2    Boobis, A.R.3    Park, B.K.4    Dabies, D.S.5
  • 4
    • 0029681461 scopus 로고    scopus 로고
    • Quantitation of cytochrome P450 enzymes (CYP1A1/2, 2B11, 2C11 and 3A12) in dog liver microsomes by enzyme-linked immunosorbent assay
    • EGUCHI, K., NISHIBE, Y., BABA, T. and OHNO, K., 1996, Quantitation of cytochrome P450 enzymes (CYP1A1/2, 2B11, 2C11 and 3A12) in dog liver microsomes by enzyme-linked immunosorbent assay. Xenobiotica, 26, 755-764.
    • (1996) Xenobiotica , vol.26 , pp. 755-764
    • Eguchi, K.1    Nishibe, Y.2    Baba, T.3    Ohno, K.4
  • 5
    • 0027537219 scopus 로고
    • Therapeutic efficacy of benzoxazinorifamycin KRM-1648 against experimental Mycobacterium avium infection induced in rabbits
    • EMORI, M., SAITO, H., SATO, K., TOMIOKA, H., SETOGAWA, T. and HIDAKA, T., 1993, Therapeutic efficacy of benzoxazinorifamycin KRM-1648 against experimental Mycobacterium avium infection induced in rabbits. Antimicrobial Agents and Chemotherapy, 37, 722-728.
    • (1993) Antimicrobial Agents and Chemotherapy , vol.37 , pp. 722-728
    • Emori, M.1    Saito, H.2    Sato, K.3    Tomioka, H.4    Setogawa, T.5    Hidaka, T.6
  • 6
    • 0042277648 scopus 로고
    • In vitro assays for drug-metabolizing enzymes
    • Glasgow: Blackie Academic & Professional
    • GIBSON, G. G. and SKETT, P., 1994, In vitro assays for drug-metabolizing enzymes. In Introduction to Drug Metabolism, 2nd edn (Glasgow: Blackie Academic & Professional), pp. 217-240.
    • (1994) Introduction to Drug Metabolism, 2nd Edn , pp. 217-240
    • Gibson, G.G.1    Skett, P.2
  • 7
    • 0028031172 scopus 로고
    • Clinically significant drug interactions with antituberculosis agents
    • GRANGE, J. M., WINSTANLEY, P. A. and DAVIES, P. D. O., 1994, Clinically significant drug interactions with antituberculosis agents. Drug Safety, 11, 242-251.
    • (1994) Drug Safety , vol.11 , pp. 242-251
    • Grange, J.M.1    Winstanley, P.A.2    Davies, P.D.O.3
  • 9
    • 0013958297 scopus 로고
    • Evidence for biochemically different types of vehicles in the hepatic microsomal fraction
    • IMAI, Y., ITO, A. and SATO, R., 1966, Evidence for biochemically different types of vehicles in the hepatic microsomal fraction. Journal of Biochemistry, 60, 417-428.
    • (1966) Journal of Biochemistry , vol.60 , pp. 417-428
    • Imai, Y.1    Ito, A.2    Sato, R.3
  • 10
    • 0028114141 scopus 로고
    • Activity of the benzoxazinorifamycin KRM-1648 against the Mycobacterium avium complex in vitro and in macrophages
    • INDERLIED, C. B., BARBARA-BURNHAM, L., WU, M., YOUNG, L. and BERMUDEZ, L. E., 1994, Activity of the benzoxazinorifamycin KRM-1648 against the Mycobacterium avium complex in vitro and in macrophages. Antimicrobial Agents and Chemotherapy, 38, 1838-1843.
    • (1994) Antimicrobial Agents and Chemotherapy , vol.38 , pp. 1838-1843
    • Inderlied, C.B.1    Barbara-Burnham, L.2    Wu, M.3    Young, L.4    Bermudez, L.E.5
  • 11
    • 0028093427 scopus 로고
    • Activity of KRM-1648, a new benzoxazinorifamycin, against Mycobacterium tuberculosis in a murine model
    • KLEMENS, S. P., GROSSI, M. A. and CYNAMON, M. H., 1994, Activity of KRM-1648, a new benzoxazinorifamycin, against Mycobacterium tuberculosis in a murine model. Antimicrobial Agents and Chemotherapy, 38, 2245-2248.
    • (1994) Antimicrobial Agents and Chemotherapy , vol.38 , pp. 2245-2248
    • Klemens, S.P.1    Grossi, M.A.2    Cynamon, M.H.3
  • 12
    • 0025977668 scopus 로고
    • In vitro activities of new rifamycin derivatives against mycobacteria
    • KUZE, F., YAMAMOTO, T., AMITANI, R. and SUZUKI, K., 1991, In vitro activities of new rifamycin derivatives against mycobacteria. Kekkaku, 66, 7-12.
    • (1991) Kekkaku , vol.66 , pp. 7-12
    • Kuze, F.1    Yamamoto, T.2    Amitani, R.3    Suzuki, K.4
  • 15
    • 0028835430 scopus 로고
    • In vitro activity of the benzoxazinorifamycin KRM-1648 against drug-susceptible and multidrug-resistant tubercle bacilli
    • LUNA-HERRERA, J., REDDY, M. V. and GANGADHAHAM, P. R. J., 1995, In vitro activity of the benzoxazinorifamycin KRM-1648 against drug-susceptible and multidrug-resistant tubercle bacilli. Antimicrobial Agents and Chemotherapy, 39, 440-444.
    • (1995) Antimicrobial Agents and Chemotherapy , vol.39 , pp. 440-444
    • Luna-Herrera, J.1    Reddy, M.V.2    Gangadhaham, P.R.J.3
  • 16
    • 0029822605 scopus 로고    scopus 로고
    • In vitro metabolism of a rifamycin derivative by animal and human liver microsomes, whole blood and expressed human CYP3a isoform
    • MAE, T., HOSOE, K., FUJII, K., YAMASHITA, K., YAMANE, T., HIDAKA, T. and OHASHI, T., 1996, In vitro metabolism of a rifamycin derivative by animal and human liver microsomes, whole blood and expressed human CYP3A isoform. Xenobiotica, 26, 793-802.
    • (1996) Xenobiotica , vol.26 , pp. 793-802
    • Mae, T.1    Hosoe, K.2    Fujii, K.3    Yamashita, K.4    Yamane, T.5    Hidaka, T.6    Ohashi, T.7
  • 18
    • 77049138167 scopus 로고
    • The colorimetric estimation of formaldehyde by means of the Hantzsch reaction
    • NASH, T., 1953, The colorimetric estimation of formaldehyde by means of the Hantzsch reaction. Biochemistry, 55, 416-421.
    • (1953) Biochemistry , vol.55 , pp. 416-421
    • Nash, T.1
  • 19
    • 0029758162 scopus 로고    scopus 로고
    • Inducing properties of rifampicin and rifabutin for selected enzyme activities of the cytochrome P-450 and UDP-glucuronosyltransferase superfamilies in female rat liver
    • OESCH, F., ARAND, M., STROLIN BENEDETTI, CASTELLE, M.G. and DOSTERT, P., 1996, Inducing properties of rifampicin and rifabutin for selected enzyme activities of the cytochrome P-450 and UDP-glucuronosyltransferase superfamilies in female rat liver. Journal of Antimicrobial Chemotherapy, 37, 1111-1119.
    • (1996) Journal of Antimicrobial Chemotherapy , vol.37 , pp. 1111-1119
    • Oesch, F.1    Arand, M.2    Strolin Benedetti3    Castelle, M.G.4    Dostert, P.5
  • 20
    • 50449100139 scopus 로고
    • The carbon monoxide-binding pigment of liver microsomes
    • OMURA, T. and SATO, R., 1964, The carbon monoxide-binding pigment of liver microsomes. Journal of Biological Chemistry, 239, 2379-2385.
    • (1964) Journal of Biological Chemistry , vol.239 , pp. 2379-2385
    • Omura, T.1    Sato, R.2
  • 25
    • 0028567499 scopus 로고
    • Induction and autoinduction properties of rifamycin derivatives : A review of animal and human studies
    • STROLIN BENEDETTI, M. and DOSTERT, P., 1994, Induction and autoinduction properties of rifamycin derivatives : a review of animal and human studies. Environmental Health Perspectives, 102(suppl. 9), 101-105.
    • (1994) Environmental Health Perspectives , vol.102 , Issue.9 SUPPL. , pp. 101-105
    • Strolin Benedetti, M.1    Dostert, P.2
  • 27
    • 0027446212 scopus 로고
    • In vitro antimicrobial activity of benzoxazinorifamycin, KRM-1648, against Mycobacterium avium complex determined by the radiometric method
    • TOMIOKA, H., SAITO, H., FUJII, K., SATO, K and HIDAKA, T., 1993, In vitro antimicrobial activity of benzoxazinorifamycin, KRM-1648, against Mycobacterium avium complex determined by the radiometric method. Antimicrobial Agents and Chemotherapy, 37, 67-70.
    • (1993) Antimicrobial Agents and Chemotherapy , vol.37 , pp. 67-70
    • Tomioka, H.1    Saito, H.2    Fujii, K.3    Sato, K.4    Hidaka, T.5
  • 28
    • 0026515252 scopus 로고
    • Chemotherapeutic efficacy of a newly synthesized benzoxazinorifamycin, KRM-1648, against Mycobacterium avium complex infection induced in mice
    • TOMIOKA, H., SAITO, H., SATO, K., YAMANE, T., YAMASHITA, K., HOSOE, K., FUJII, K. and HIDAKA, T., 1992, Chemotherapeutic efficacy of a newly synthesized benzoxazinorifamycin, KRM-1648, against Mycobacterium avium complex infection induced in mice. Antimicrobial Agents and Chemotherapy, 36, 387-393.
    • (1992) Antimicrobial Agents and Chemotherapy , vol.36 , pp. 387-393
    • Tomioka, H.1    Saito, H.2    Sato, K.3    Yamane, T.4    Yamashita, K.5    Hosoe, K.6    Fujii, K.7    Hidaka, T.8
  • 29
    • 0026531077 scopus 로고
    • Pharmacokinetic drug interactions with rifampicin
    • VENKATESAN, K., 1992, Pharmacokinetic drug interactions with rifampicin. Clinical Pharmacokinetics, 22, 47-65.
    • (1992) Clinical Pharmacokinetics , vol.22 , pp. 47-65
    • Venkatesan, K.1
  • 30
    • 0028915901 scopus 로고
    • Reduced serum levels of clarithromycin in patients treated with multidrug regimens including rifampin or rifabutin for Mycobacterium avium-M. intracellulare infection
    • WALLACE, R. J. JR, BROWN, B. A., GRIFFITH, D. E., GIRARD, W. and TANAKA, K., 1995, Reduced serum levels of clarithromycin in patients treated with multidrug regimens including rifampin or rifabutin for Mycobacterium avium-M. intracellulare infection. Journal of Infectious Diseases, 171, 747-750.
    • (1995) Journal of Infectious Diseases , vol.171 , pp. 747-750
    • Wallace Jr., R.J.1    Brown, B.A.2    Griffith, D.E.3    Girard, W.4    Tanaka, K.5
  • 31
    • 0026341321 scopus 로고
    • Site of action of substrates requiring cytochrome b5 for oxidation by cytochrome P450
    • WASKELL, L. A., VIGNE, J. L. and VERGERES, G., 1991, Site of action of substrates requiring cytochrome b5 for oxidation by cytochrome P450. Methods in Enzymology, 206, 523-529.
    • (1991) Methods in Enzymology , vol.206 , pp. 523-529
    • Waskell, L.A.1    Vigne, J.L.2    Vergeres, G.3
  • 32
    • 0025634037 scopus 로고
    • In vitro activities of new rifamycin derivatives against Mycobacterium tuberculosis and M. avium complex
    • YAMAMOTO, T., AMITANI, R., KUZE, F. and SUZUKI, K., 1990, In vitro activities of new rifamycin derivatives against Mycobacterium tuberculosis and M. avium complex. Kekkaku, 65, 805-810.
    • (1990) Kekkaku , vol.65 , pp. 805-810
    • Yamamoto, T.1    Amitani, R.2    Kuze, F.3    Suzuki, K.4
  • 34
    • 0030029958 scopus 로고    scopus 로고
    • Erythromycin as a specific substrate for cytochrome P4503a isozymes and identification of a high-affinity erythromycin N-demethylase in adult female rats
    • ZHANG, X. J. and THOMAS, P. E., 1996, Erythromycin as a specific substrate for cytochrome P4503A isozymes and identification of a high-affinity erythromycin N-demethylase in adult female rats. Drug Metabolism and Disposition, 24, 23-27.
    • (1996) Drug Metabolism and Disposition , vol.24 , pp. 23-27
    • Zhang, X.J.1    Thomas, P.E.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.