Combined histamine H1/H2 receptor antagonists: Part II. Pharmacological hybrids with pheniramine- and tiotidine-like substructures

European Journal of Pharmaceutical Sciences

Volumn 6, Issue 3, 1998, Pages 187-196

  Wolf, Cornelia ^a   Schulze, Frank R ^a   Buschauer, Armin ^b   Schunack, Walter ^a  

^a FREIE UNIVERSITÄT BERLIN   (Germany)

^b UNIVERSITY OF REGENSBURG   (Germany)

Author keywords

2 Guanidinothiazole; Histamine; Histamine H1 receptor antagonists; Histamine H2 receptor antagonists; Pheniramine

Indexed keywords

HISTAMINE H1 RECEPTOR; HISTAMINE H1 RECEPTOR ANTAGONIST; HISTAMINE H2 RECEPTOR; HISTAMINE H2 RECEPTOR ANTAGONIST; ICOTIDINE; PHENIRAMINE; TIOTIDINE; CIMETIDINE; DRUG DERIVATIVE;

ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; GUINEA PIG; HEART RIGHT ATRIUM; ILEUM; IN VITRO STUDY; NONHUMAN; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; PKA; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION; ANIMAL; DRUG EFFECT; HEART ATRIUM; HEART ATRIUM FUNCTION; PHYSIOLOGY; SYNTHESIS;

ANIMALS; ATRIAL FUNCTION; CIMETIDINE; GUINEA PIGS; HEART ATRIA; HISTAMINE H1 ANTAGONISTS; HISTAMINE H2 ANTAGONISTS; ILEUM; PHENIRAMINE; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0031593477     PISSN: 09280987     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0928-0987(97)10017-3     Document Type: Article

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