Recognition and activation of the opioid receptor-like ORL1 receptor by nociceptin, nociceptin analogs and opioids

European Journal of Pharmacology

Volumn 321, Issue 1, 1997, Pages 97-103

  Butour, Jean Luc ^a   Moisand, Christiane ^a   Mazarguil, Honoré ^a   Mollereau, Catherine ^a   Meunier, Jean Claude ^a  

^a CNRS   (France)

Author keywords

3H Nociceptin; Adenylylcyclase, inhibition; Drug screening; Nociceptin receptor; Radioreceptor assay

Indexed keywords

3,4 DICHLORO N METHYL N [2 (1 PYRROLIDINYL)CYCLOHEXYL]BENZENEACETAMIDE; ADENYLATE CYCLASE; ALPHA NEOENDORPHIN; CYCLIC AMP; DELTAKEPHALIN; DIPRENORPHINE; DYNORPHIN A; ENKEPHALIN[2 DEXTRO ALANINE 4 METHYLPHENYLALANINE 5 GLYCINE]; ETHYLKETAZOCINE; ETORPHINE; FENTANYL; GUANYLYLIMIDODIPHOSPHATE; LEUCINE ENKEPHALIN; LOFENTANIL; METENKEPHALIN; MORPHINE; NALOXONE; NOCICEPTIN; OPIATE; OPIATE RECEPTOR;

ANIMAL TISSUE; ARTICLE; BINDING SITE; CHO CELL; CONTROLLED STUDY; DRUG RECEPTOR BINDING; HAMSTER; NOCICEPTIVE RECEPTOR; NONHUMAN; PRIORITY JOURNAL; RADIORECEPTOR ASSAY; RECEPTOR AFFINITY; SCREENING;

ADENYLATE CYCLASE; AMINO ACID SEQUENCE; ANALGESICS, OPIOID; ANIMALS; BINDING, COMPETITIVE; CELL MEMBRANE; CHO CELLS; CRICETINAE; ENZYME INHIBITORS; FENTANYL; FORSKOLIN; MOLECULAR SEQUENCE DATA; OPIOID PEPTIDES; RECEPTORS, OPIOID;

EID: 0031577964     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(96)00919-3     Document Type: Article

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