Construction of a high-affinity receptor site for dihydropyridine agonists and antagonists by single amino acid substitutions in a non-L-type Ca2+ channel

Proceedings of the National Academy of Sciences of the United States of America

Volumn 94, Issue 26, 1997, Pages 14906-14911

  Hockerman, Gregory H ^a   Peterson, Blaise Z ^a   Sharp, Elizabeth ^a   Tanada, Timothy N ^a   Scheuer, Todd ^a   Catterall, William A ^a  

^a UNIVERSITY OF WASHINGTON SCHOOL OF MEDICINE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

1,4 DIHYDRO 2,6 DIMETHYL 5 NITRO 4 [2 (TRIFLUOROMETHYL)PHENYL] 3 PYRIDINECARBOXYLIC ACID METHYL ESTER; AMINO ACID; BARIUM; CALCIUM CHANNEL; CALCIUM ION; DIHYDROPYRIDINE; ISRADIPINE; RECEPTOR;

ALPHA CHAIN; AMINO ACID SUBSTITUTION; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; ENERGY; HUMAN; HUMAN CELL; LIGAND BINDING; POLYMERASE CHAIN REACTION; PRIORITY JOURNAL; VOLTAGE CLAMP;

AMINO ACID SUBSTITUTION; AMINO ACIDS; BINDING SITES; CALCIUM CHANNELS; CALCIUM CHANNELS, L-TYPE; CELL LINE; DIHYDROPYRIDINES; HUMANS;

EID: 0031434472     PISSN: 00278424     EISSN: None     Source Type: Journal    
DOI: 10.1073/pnas.94.26.14906     Document Type: Article

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