메뉴 건너뛰기




Volumn 36, Issue 11-12, 1997, Pages 1483-1488

A novel kainate receptor ligand [3H]-(2S,4R)-4-methylglutamate: Pharmacological characterization in rabbit brain membranes

Author keywords

Kainate receptors; Rabbit brain synaptic membranes; Radioligand binding; 3H (2S,4R) 4 methylglutamate

Indexed keywords

1 AMINO 1,3 CYCLOPENTANEDICARBOXYLIC ACID; 4 METHYLGLUTAMIC ACID; 6 CYANO 7 NITRO 2,3 QUINOXALINEDIONE; ALPHA AMINO 3 HYDROXY 5 METHYL 4 ISOXAZOLEPROPIONIC ACID; AMPA RECEPTOR; DOMOIC ACID; GLUTAMATE RECEPTOR; GLUTAMIC ACID; ION CHANNEL; IONOTROPIC RECEPTOR; KAINIC ACID RECEPTOR; METABOTROPIC RECEPTOR; N METHYL DEXTRO ASPARTIC ACID; QUISQUALIC ACID; UNCLASSIFIED DRUG;

EID: 0031423745     PISSN: 00283908     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0028-3908(97)00161-5     Document Type: Article
Times cited : (27)

References (21)
  • 1
    • 0028348997 scopus 로고
    • Resolution and regioselective protection of glutamic acid analogues. 1 - Resolution of diastereomeric α-boroxazolidone derivatives
    • Acher F. and Azerad R. (1994) Resolution and regioselective protection of glutamic acid analogues. 1 - Resolution of diastereomeric α-boroxazolidone derivatives. Tetrahedron Assymetry 5: 731-744.
    • (1994) Tetrahedron Assymetry , vol.5 , pp. 731-744
    • Acher, F.1    Azerad, R.2
  • 3
    • 0029240274 scopus 로고
    • Review: Neurotransmitter receptors 2. AMPA and kainate receptors
    • Bettler B. and Mulle C. (1995) Review: Neurotransmitter Receptors 2. AMPA and kainate receptors. Neuropharmacology 34: 123-139.
    • (1995) Neuropharmacology , vol.34 , pp. 123-139
    • Bettler, B.1    Mulle, C.2
  • 5
    • 0026080845 scopus 로고
    • Conformationally defined neurotransmitter analogues. Selective inhibition of glutamate uptake by one pyrrolidine-2,4-dicarboxylate diastereomer
    • Bridges R. J., Stanley M. S., Anderson M. W., Cotman C. W. and Chamberlin A. R. (1991) Conformationally defined neurotransmitter analogues. Selective inhibition of glutamate uptake by one pyrrolidine-2,4-dicarboxylate diastereomer. Journal of Medicinal Chemistry 34: 717-725.
    • (1991) Journal of Medicinal Chemistry , vol.34 , pp. 717-725
    • Bridges, R.J.1    Stanley, M.S.2    Anderson, M.W.3    Cotman, C.W.4    Chamberlin, A.R.5
  • 6
    • 0029045977 scopus 로고
    • Synthesis, resolution, and biological evaluation of the four stereoisomers of 4-methylglutamic acid: Selective probes of kainate receptors
    • Gu Z.-Q., Hesson D. P., Pelletier J. C., Maccecchini M.-L., Zhou L.-M. and Skolnick P. (1995) Synthesis, resolution, and biological evaluation of the four stereoisomers of 4-methylglutamic acid: selective probes of kainate receptors. Journal of Medicinal Chemistry 38: 2518-2520.
    • (1995) Journal of Medicinal Chemistry , vol.38 , pp. 2518-2520
    • Gu, Z.-Q.1    Hesson, D.P.2    Pelletier, J.C.3    Maccecchini, M.-L.4    Zhou, L.-M.5    Skolnick, P.6
  • 8
    • 0026530085 scopus 로고
    • The KA-2 subunit of excitatory amino acid receptors shows widespread expression in brain and forms ion channels with distantly related subunits
    • Herb A., Burnashev N., Werner P., Sakmann B., Wisden W. and Seeburg P. H. (1992) The KA-2 subunit of excitatory amino acid receptors shows widespread expression in brain and forms ion channels with distantly related subunits. Neuron 8: 775-785.
    • (1992) Neuron , vol.8 , pp. 775-785
    • Herb, A.1    Burnashev, N.2    Werner, P.3    Sakmann, B.4    Wisden, W.5    Seeburg, P.H.6
  • 11
    • 0029954379 scopus 로고    scopus 로고
    • Homomeric and heteromeric ion channels formed from the kainate-type subunits GluR6 and KA2 have very small, but different, unitary conductances
    • Howe J. R. (1996) Homomeric and heteromeric ion channels formed from the kainate-type subunits GluR6 and KA2 have very small, but different, unitary conductances. Journal of Neurophysiology 76: 510-519.
    • (1996) Journal of Neurophysiology , vol.76 , pp. 510-519
    • Howe, J.R.1
  • 16
    • 0028912822 scopus 로고
    • Neurotransmitter receptors I. The metabotropic glutamate receptors: Structure and functions
    • Pin J. P. and Duvoisin R. (1995) Neurotransmitter receptors I. The metabotropic glutamate receptors: structure and functions. Neuropharmacology 34: 1-26.
    • (1995) Neuropharmacology , vol.34 , pp. 1-26
    • Pin, J.P.1    Duvoisin, R.2
  • 18
    • 0028169790 scopus 로고
    • Selective block of recombinant glur6 receptors by NS-102, a novel non-NMDA receptor antagonist
    • Verdoorn T. A., Johansen T. H., Drejer J. and Nielsen E. Ø. (1994) Selective block of recombinant glur6 receptors by NS-102, a novel non-NMDA receptor antagonist. European Journal of Pharmacology 269: 43-49.
    • (1994) European Journal of Pharmacology , vol.269 , pp. 43-49
    • Verdoorn, T.A.1    Johansen, T.H.2    Drejer, J.3    Nielsen, E.Ø.4
  • 19
    • 0025810536 scopus 로고
    • Cloning of a putative high-affinity kainate receptor expressed predominantly in hippocampal CA3 cells
    • Werner P., Voigt M., Keinänen K., Wisden W. and Seeburg P. H. ( 1991 ) Cloning of a putative high-affinity kainate receptor expressed predominantly in hippocampal CA3 cells. Nature 351: 742-744.
    • (1991) Nature , vol.351 , pp. 742-744
    • Werner, P.1    Voigt, M.2    Keinänen, K.3    Wisden, W.4    Seeburg, P.H.5
  • 20
    • 0027471024 scopus 로고
    • Glutamate uptake system in the presynaptic vesicle: Glutamic acid analogs as inhibitors and alternate substrates
    • Winter H. C. and Ueda T. (1993) Glutamate uptake system in the presynaptic vesicle: glutamic acid analogs as inhibitors and alternate substrates. Neurochemical Research 18: 79-85.
    • (1993) Neurochemical Research , vol.18 , pp. 79-85
    • Winter, H.C.1    Ueda, T.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.