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Keating TA, Armstrong RW: A remarkable two-step synthesis of diverse 1,4-benzodia2epine-2,5-dlones using the Ugi four-component condensation. J Org Chem 1996, 61:8935-8939. Example of a short reaction sequence capable of enormous diversity.
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Overman LE, Tellew JE: Synthesis of 2-azatricyclo[5.2.1.04,10]decanes and 2,5-diazatricyclo[5.2.1.04,10] decanes by intramolecular azomethine ylide cycloadditions. J Org Chem 1996, 61:8338-8340. A solution-phase example employing the azomethine ylide cycloaddition to formulate complex products.
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